ARTICLE;
CARBON NUCLEAR MAGNETIC RESONANCE;
CHEMICAL REACTION;
DRUG STRUCTURE;
DRUG SYNTHESIS;
NONHUMAN;
ONE POT SYNTHESIS;
PRIORITY JOURNAL;
PROTON NUCLEAR MAGNETIC RESONANCE;
ROOM TEMPERATURE;
Studies on the application of the Passerini reaction and enzymatic procedures to the synthesis of tripeptide mimetics
DOI 10.1016/j.tet.2007.05.044, PII S0040402007009064
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(2007)Tetrahedron, vol.63, Issue.32, pp. 7647-7653
Strategies for heterocyclic construction via novel multicomponent reactions based on isocyanides and nucleophilic carbenes
doi:10.1021/ar020258p
Nair V, Rajesh C, Vinod AU, Bindu S, Sreekanth AR, Mathen JS, Balagopal L (2003) Strategies for heterocyclic construction via novel multicomponent reactions based on isocyanides and nucleophilic carbenes. Acc Chem Res 36:899-907. doi:10.1021/ar020258p
Ugi I (1982) From isocyanides via four-component condensations to antibiotic syntheses. Angew Chem Int Ed Engl 21:810-819. doi:10.1002/1521- 3773(20000915)39:18<3168:AID-NIE3168>3.0.CO;2-U
Dihydrobenzopyrans, dihydrobenzothiopyrans, and tetrahydroquinolines for the treatment of COX-2-mediated disorders, WO2001049675
Rogier DJ Jr, Carter JS, Talley JJ (2001) Dihydrobenzopyrans, dihydrobenzothiopyrans, and tetrahydroquinolines for the treatment of COX-2-mediated disorders, WO2001049675. Chem Abstr 135:107252
The antimicrobial natural product chuangxinmycin and Some synthetic analogues are potent and selective inhibitors of bacterial tryptophanyl tRNA synthetase
doi:10.1016/S0960-894X(02)00604-2
Brown MJ, Carter PS, Fenwick AE, Fosberry AP, Hamprecht DW, Hibbs MJ, Arvest RL, Mensah L, Milner PH, O'Hanlon PJ, Pope AJ, Richardson CM, West A, Witty DR (2002) The antimicrobial natural product chuangxinmycin and Some synthetic analogues are potent and selective inhibitors of bacterial tryptophanyl tRNA synthetase. Bioorg Med Chem Lett 12:3171-3174. doi:10.1016/S0960-894X(02)00604-2
Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes
doi:10.1021/jm011066n
Quaglia W, Pigini M, Piergentili A, Giannella M, Gentili F, Marucci G, Carrieri A, Carotti A, Poggesi E, Leonardi A, Melchiorre C (2002) Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes. J Med Chem 45:1633-1643. doi:10.1021/jm011066n
Synthesis and pharmacological evaluation of thiopyran analogues of the dopamine D3 receptor-selective agonist (4aR,10bR)-(+)-trans- 3,4,4a,10b-tetrahydro-4-n-propyl-2H,5H [1] benzopyrano[4,3-b]- 1,4-oxazin-9-ol (PD 128907)
doi:10.1021/jm0000113
Van Vliet LA, Rodenhuis N, Dijkstra D, Wikstrom H, Pugsley TA, Serpa KA, Meltzer LT, Heffner TG, Wise LD, Lajiness ME, Huff RM, Svensson K, Sundell S, Lundmark M (2000) Synthesis and pharmacological evaluation of thiopyran analogues of the dopamine D3 receptor-selective agonist (4aR,10bR)-(+)-trans- 3,4,4a,10b-tetrahydro-4-n-propyl-2H,5H [1] benzopyrano[4,3-b]- 1,4-oxazin-9-ol (PD 128907). J Med Chem 43:2871-2882. doi:10.1021/jm0000113
Enantioselective organocatalytic tandem Michael-Aldol reactions: One-pot synthesis of chiral thiochromenes
DOI 10.1021/ja063328m
Wang W, Li H, Wang J, Zu LS (2006) Enantioselective organocatalytic tandem Michael-Aldol reactions: one-pot synthesis of chiral thiochromenes. J Am Chem Soc 128:10354-10355. doi:10.1021/ja063328m (Pubitemid 44265063)
Synthesis of substituted 2-iminothiopyrans from aryl ethylidene malononitriles
Samuel R, Asokan CV (2001) Synthesis of substituted 2-iminothiopyrans from aryl ethylidene malononitriles. Indian J Chem Sect B 40:834-836 (Pubitemid 32963700)
Synthesis of derivatives of 2-imino-5,6-dihydro-2H-thiopyran from 1- Heteroalkyl-1,3-butadienes and isothiocyanates
DOI 10.1016/S0040-4039(97)86431-3, PII S004040399800244X
Nedolya NA, Brandsma L (1998) Synthesis of derivatives of 2-imino-5,6-dihydro-2H-thiopyran from 1-heteroalkyl-1,3-butadienes and isothiocyanates. Tetrahedron Lett 39:2631-2634. doi:10.1016/S0040-4039(97)86431- 3 (Pubitemid 28224475)
A one-pot synthesis of functionalized thiazoles from acid chlorides, secondary amines, ethyl bromopyruvate, and ammonium thiocyanate
doi:10.1007/s11030-009-9114-3
Yavari I, Hossaini Z, Sabbaghan M, Ghazanfarpour-Darjani M (2009) A one-pot synthesis of functionalized thiazoles from acid chlorides, secondary amines, ethyl bromopyruvate, and ammonium thiocyanate. Mol Divers 13:295-300. doi:10.1007/s11030-009-9114-3
Diastereoselective synthesis of fused [1,3]thiazolo[1,3]oxazins and [1,3]oxazino[2,3- B][1,3]benzothiazoles
doi:10.1007/s11030-009-9128-x
Yavari I, Hossaini Z, Souri S (2009) Diastereoselective synthesis of fused [1,3]thiazolo[1,3]oxazins and [1,3]oxazino[2,3- b][1,3]benzothiazoles. Mol Divers 13:439-443. doi:10.1007/s11030-009-9128-x
One-pot synthesis of 4-hydroxy-3-phenyl-2h-pyrano[ 3,2-b]benzofuran-2-one derivatives
doi:10.1080/00397910802585886
Foroumadi A, Zamanian S, Samzadeh-Kermani A, Shafiee A (2009) One-pot synthesis of 4-hydroxy-3-phenyl-2h-pyrano[ 3,2-b]benzofuran-2-one derivatives. Synth Commun 39: 1722-1728. doi:10.1080/00397910802585886
Synthesis and cytotoxic activity of novel chromenes
doi:08-3057DP
Alizadeh BH, Ostad SN, Foroumadi A, Amini M, Dowlatabadi R, Navidpour L, Shafiee A (2008) Synthesis and cytotoxic activity of novel chromenes. Arkivok 13:45-56. doi:08-3057DP
