Syntheses and biological evaluation of new triazole-spirochromone conjugates as inhibitors of Mycobacterium tuberculosis

Tetrahedron Letters

Volumn 52, Issue 18, 2011, Pages 2387-2389

  Muthukrishnan, M ^a   Mujahid, M ^a   Yogeeswari, P ^b   Sriram, D ^b  

^a NATIONAL CHEMICAL LABORATORY   (India)

^b BIRLA INSTITUTE OF TECHNOLOGY AND SCIENCE   (India)

Author keywords

Antitubercular activity; Click chemistry; Mycobacterium tuberculosis; Spirochromones

Indexed keywords

AMMONIUM CHLORIDE; CHROMONE DERIVATIVE; SODIUM AZIDE; TRIAZOLE DERIVATIVE;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL STRAIN; DRUG INHIBITION; DRUG SYNTHESIS; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; STRUCTURE ACTIVITY RELATION;

MYCOBACTERIUM TUBERCULOSIS;

EID: 79953283288     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2011.02.099     Document Type: Article

References (34)

1. WHO Global Tuberculosis Control Report, 2009.
2. M.T. Gutierrez-Lugo, and C.A. Bewley J. Med. Chem. 51 2008 2606
3. C.V. Smith, V. Sharma, and J.C. Sacchettini Tuberculosis 84 2004 45
4. E.L. Corbett, C.J. Watt, N. Walker, D. Maher, B.G. Williams, M.C. Raviglione, and C. Dye Arch. Intern. Med. 163 2003 1009
5. R. Long Can. Med. Assoc. J. 163 2000 425
6. A. Pozniak J. Tuberc. Lung Dis. 4 2000 993
7. R.J. O'Brien, and P.P. Nunn Am. J. Respir. Crit. Care Med. 162 2001 1055
8. B.E. Laughon Curr. Top. Med. Chem. 7 2007 463
9. K. Duncan, and C.E. Barry III Curr. Opin. Microbiol. 7 2004 460
10. R. Ranjithkumar, S. Perumal, P. Senthilkumar, P. Yogeeswari, and D. Sriram J. Med. Chem. 51 2008 5731
11. R. Frank Curr. Opin. Biotechnol. 15 2004 573
12. J.Y. Ortholand, and A. Ganesan Curr. Opin. Chem. Biol. 8 2004 271
13. G. Mehta, and V. Singh Chem. Soc. Rev. 31 2002 324
14. M.A. Koch, M. Schuffenhauer, M. Scheck, S. Wetzel, M. Casaulta, A. Odermatt, P. Ertl, and H. Waldmann Proc. Natl. Acad. Sci. U.S.A. 102 2005 17272
15. G. Zinzalla, L.G. Milroy, and S.V. Ley Org. Biomol. Chem. 4 2006 1977
16. D.A. Horton, G.T. Bourne, and M.L. Smythe Chem. Rev. 103 2003 893
17. G.P. Ellis Chromenes, Chromanones and Chromones The Chemistry of Heterocyclic Compounds Vol. 31 1977 Wiley New York
18. J. Hepworth A.R. Katrizky, C.W. Rees, Comprehensive Heterocyclic Chemistry Vol. 3 1984 Pergamon Oxford, UK 737 883
19. M. Muthukrishnan, U.M.V. Basavanag, and V.G. Puranik Tetrahedron Lett. 50 2009 2643
20. M. Muthukrishnan, and O.V. Singh Synth. Commun. 38 2008 3875
21. M. Muthukrishnan, P.S. Patil, S.V. More, and R.A. Joshi Mendeleev Commun. 2005 100
22. O.V. Singh, M. Muthukrishnan, and R. Gopan Synth. Commun. 35 2005 2723
23. O.V. Singh, M. Muthukrishnan, and M. Sundaravadivelu Indian J. Chem., Sect. B 44 2005 2575
24. H.C. Kolb, M.G. Finn, and K.B. Sharpless Angew. Chem., Int. Ed. 40 2001 2004
25. M. Meldel, and C.W. Tornoe Chem. Rev. 108 2008 2952
26. G.C. Tron, T. Pirali, R.A. Billington, P.L. Canonico, G. Sorba, and A.A. Genazzani Med. Res. Rev. 28 2008 278
27. C.W. Tornoe, C. Christensen, and M. Meldal J. Org. Chem. 67 2002 3057
28. J. Yoon, and J.S. Ryu Bioorg. Med. Chem. Lett. 20 2010 3930
29. H.C. Kolb, and K.B. Sharpless Drug Discovery Today 8 2003 1128
30. H.J. Kabbe Synthesis 1978 886
31. V.S. Moskvina, Y.L. Garazd, M.M. Garazd, A.V. Turov, and V.P. Khilya Chem. Heterocycl. Compd. 43 2007 421
32. +.
33. F. Himo, T. Lovell, R. Hilgraf, V.V. Rostovtsev, L. Noodleman, K.B. Sharpless, and V.V. Fokin J. Am. Chem. Soc. 127 2005 210
34. NCCLS-National Committee for Clinical Laboratory Standards, Antimycobacterial susceptibility testing for Mycobacterium tuberculosis. Proposed standard M24-T; Villanova, PA, 1995.