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Tetrahedron Letters

Volumn 52, Issue 15, 2011, Pages 1807-1810

Synthesis of two isotopically labeled versions of NEDD8-activating enzyme (NAE) inhibitor

(3) Li, Yuexian a Plesescu, Mihaela a Prakash, Shimoga R a

a MILLENNIUM PHARMACEUTICALS INC (United States)

Author keywords

14C 6 chloro 7 deazapurine; D 8 (S) 1 aminoindan; MLN4924; NAE inhibitor

Indexed keywords

9 DEXTRO 3 PHENYLPROPANOIC ACID; CARBON 14; ENZYME INHIBITOR; MLN 4924; NEDD8 ACTIVATING ENZYME INHIBITOR; PROPIONIC ACID DERIVATIVE; SULFUR ACID DERIVATIVE; THIOUREA; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; CYCLIZATION; DRUG ACTIVITY; DRUG SYNTHESIS; HYDROLYSIS; ISOTOPE LABELING; NONHUMAN; STRUCTURE ACTIVITY RELATION;

EID: 79952538394 PISSN: 00404039 EISSN: None Source Type: Journal
DOI: 10.1016/j.tetlet.2011.02.033 Document Type: Article

Times cited : (6)

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