-
1
-
-
10744221981
-
Tamoxifen DNA Damage Detected in Human Endometrium Using Accelerator Mass Spectrometry
-
EA Martin K Brown M Gaskell F Al-Azzawi RC Garner DJ Boocock, et al. 2003 Tamoxifen DNA damage deteted in human endometrium using accelerator mass spectrometry Cancer Res 63 8461 8465 1:CAS:528:DC%2BD3sXpvVagur8%3D (Pubitemid 37549502)
-
(2003)
Cancer Research
, vol.63
, Issue.23
, pp. 8461-8465
-
-
Martin, E.A.1
Brown, K.2
Gaskell, M.3
Al-Azzawi, F.4
Garner, R.C.5
Boocock, D.J.6
Mattock, E.7
Pring, D.W.8
Dingley, K.9
Turteltaub, K.W.10
Smith, L.L.11
White, I.N.H.12
-
2
-
-
34248350428
-
Medicinal chemistry and emerging strategies applied to the development of selective estrogen receptor modulators (SERMs)
-
DOI 10.2174/092986707780598023
-
MA Musa MOF Khan JS Cooperwood 2007 Medicinal chemistry and emerging strategies applied to the development of selective estrogen receptor modulators (SERMs) Curr Med Chem 14 1249 1261 10.2174/092986707780598023 1:CAS:528:DC%2BD2sXltFejsrc%3D (Pubitemid 46739325)
-
(2007)
Current Medicinal Chemistry
, vol.14
, Issue.11
, pp. 1249-1261
-
-
Musa, M.A.1
Khan, M.O.F.2
Cooperwood, J.S.3
-
3
-
-
14044265107
-
The efficacy of tamoxifen in estrogen receptor-positive breast cancer cells is enhanced by a medical nutriment
-
DOI 10.1089/cbr.2004.19.746
-
Z Marcsek Z Kocsis M Jakab B Szende A Tompa 2004 The efficacy of tamoxifen in estrogen receptor-positive breast cancer cells is enhanced by a medical nutriment Cancer Biother Radiopharm 19 746 753 10.1089/cbr.2004.19.746 1:CAS:528:DC%2BD2MXhs1Cjsr0%3D (Pubitemid 40279583)
-
(2004)
Cancer Biotherapy and Radiopharmaceuticals
, vol.19
, Issue.6
, pp. 746-753
-
-
Marcsek, Z.1
Kocsis, Z.2
Jakab, M.3
Szende, B.4
Tompa, A.5
-
4
-
-
0030751284
-
The role of β-glucuronidase in drug disposition and drug targeting in humans
-
B Sperker JT Backman HK Kroemer 1997 The role of beta-glucuronidase in drug disposition and drug targeting in humans J Clin Pharmacol 33 18 31 1:CAS:528:DyaK2sXltlShsbo%3D (Pubitemid 27303115)
-
(1997)
Clinical Pharmacokinetics
, vol.33
, Issue.1
, pp. 18-31
-
-
Sperker, B.1
Backman, J.T.2
Kroemer, H.K.3
-
5
-
-
0001144402
-
Characterization of novel anthracycline prodrugs activated by human β-glucuronidase for use in antibody-directed enzyme prodrug therapy
-
DOI 10.1016/0006-2952(96)00248-1
-
PHJ Houba RGG Leenders E Boven JW Scheeren HM Pinedo HJ Haisma 1996 Characterization of novel anthracycline prodrugs activated by human β-glucuronidase for use in antibody-directed enzyme prodrug therapy Biochem Pharmacol 9 455 463 10.1016/0006-2952(96)00248-1 (Pubitemid 26233589)
-
(1996)
Biochemical Pharmacology
, vol.52
, Issue.3
, pp. 455-463
-
-
Houba, P.H.J.1
Leenders, R.G.G.2
Boven, E.3
Scheeren, J.W.4
Pinedo, H.M.5
Haisma, H.J.6
-
6
-
-
44749093733
-
Pyrrolo[2,1-c][1,4]benzodiazepine-β-glucuronide prodrugs with a potential for selective therapy of solid tumors by PMT and ADEPT strategies
-
10.1016/j.bmcl.2008.05.038 1:CAS:528:DC%2BD1cXnt1Ogsr0%3D
-
A Kamal V Tekumalla P Raju VGM Naidu PV Diwan R Sistla 2008 Pyrrolo[2,1-c][1,4]benzodiazepine-β-glucuronide prodrugs with a potential for selective therapy of solid tumors by PMT and ADEPT strategies Bioorg Med Chem Lett 18 3769 3773 10.1016/j.bmcl.2008.05.038 1:CAS:528:DC%2BD1cXnt1Ogsr0%3D
-
(2008)
Bioorg Med Chem Lett
, vol.18
, pp. 3769-3773
-
-
Kamal, A.1
Tekumalla, V.2
Raju, P.3
Naidu, V.G.M.4
Diwan, P.V.5
Sistla, R.6
-
7
-
-
0035812971
-
Fluorogenic assay for β-glucuronidase using microchip-based capillary electrophoresis
-
DOI 10.1016/S0378-4347(01)00313-9, PII S0378434701003139
-
DE Starkey A Han JJ Bao CH Ahn KR Wehmeyer MC Prenger, et al. 2001 Fluorogenic assay for β-glucuronidase using microchip-based capillary electrophorrsis J Chromatogr 762 33 41 10.1016/S0378-4347(01)00313-9 1:CAS:528:DC%2BD3MXmvVygt7s%3D (Pubitemid 32885580)
-
(2001)
Journal of Chromatography B: Biomedical Sciences and Applications
, vol.762
, Issue.1
, pp. 33-41
-
-
Starkey, D.E.1
Han, A.2
Bao, J.J.3
Ahn, C.H.4
Wehmeyer, K.R.5
Prenger, M.C.6
Halsall, H.B.7
Heineman, W.R.8
-
8
-
-
0022841821
-
Beta-Glucuronidase levels in patients with fibrocystic breast disease
-
10.1007/BF01807334 1:STN:280:DyaL2s3kt12qtw%3D%3D
-
JP Minton Z Walaszek W Schooley WM Hanausek TE Webb 1986 Beta-Glucuronidase levels in patients with fibrocystic breast disease Breast Cancer Res Treat 8 217 222 10.1007/BF01807334 1:STN:280:DyaL2s3kt12qtw%3D%3D
-
(1986)
Breast Cancer Res Treat
, vol.8
, pp. 217-222
-
-
Minton, J.P.1
Walaszek, Z.2
Schooley, W.3
Hanausek, W.M.4
Webb, T.E.5
-
9
-
-
0029904131
-
Synthesis, biodistribution, and estrogen receptor scintigraphy of indium- 111-diethylenetriaminepentaacetic acid-tamoxifen analogue
-
DOI 10.1021/js960049w
-
SE Delpassand JD Yang S Wallace A CherIf MS QuadrI J Price, et al. 1996 Synthesis, biodistribution and estrogen receptor scintigraphy of Indium-111-diethylenetriamine pentaacetic acid-tamoxifen analogue J Pharm Sci 85 553 559 10.1021/js960049w 1:CAS:528:DyaK28XivVCks7k%3D (Pubitemid 26179651)
-
(1996)
Journal of Pharmaceutical Sciences
, vol.85
, Issue.6
, pp. 553-559
-
-
Delpassand, E.S.1
Yang, D.J.2
Wallace, S.3
Cherif, A.4
Quadri, S.M.5
Price, J.6
Joubert, A.7
Inoue, T.8
Podoloff, D.A.9
-
12
-
-
0017184389
-
A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding
-
10.1016/0003-2697(76)90527-3 1:CAS:528:DyaE28XksVehtrY%3D
-
MM Bradford 1976 A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding Anal Biochem 72 248 254 10.1016/0003-2697(76)90527-3 1:CAS:528: DyaE28XksVehtrY%3D
-
(1976)
Anal Biochem
, vol.72
, pp. 248-254
-
-
Bradford, M.M.1
-
13
-
-
0037025065
-
Sensitive liquid chromatographic method using fluorescence detection for the determination of estradiol 3- and 17-glucuronides in rat and human liver microsomal incubations: Formation kinetics
-
DOI 10.1016/S1570-0232(02)00188-5, PII S1570023202001885
-
KM Alkharfy RF Frye 2002 Sensitive liquid chromatographic method using fluorescence detection for the determination of estradiol 3- and 17-glucuronides in rat and human liver microsomal incubations: formation kinetics J Chromatogr B Analyt Technol Biomed Life Sci 1 33 38 10.1016/S1570-0232(02)00188-5 (Pubitemid 34607421)
-
(2002)
Journal of Chromatography B: Analytical Technologies in the Biomedical and Life Sciences
, vol.774
, Issue.1
, pp. 33-38
-
-
Alkharfy, K.M.1
Frye, R.F.2
-
14
-
-
0345003995
-
Optimization of β-D-glucuronide synthesis using UDP-glucuronyl transferase
-
DOI 10.1016/S0141-0229(98)00137-9, PII S0141022998001379
-
DE Stevenson U Hubl 1999 Optimization of β-glucuronide synthesis using UDP-glucuronyl transferase Enzyme Microbial Technol 24 388 396 10.1016/S0141-0229(98)00137-9 1:CAS:528:DyaK1MXisFKgtrw%3D (Pubitemid 29182642)
-
(1999)
Enzyme and Microbial Technology
, vol.24
, Issue.7
, pp. 388-396
-
-
Stevenson, D.E.1
Hubl, U.2
-
15
-
-
0032966716
-
Optimisation of UDP-glucuronyl transferase-catalysed synthesis of testosterone-β-D-glucuronide by inhibition of contaminating β-glucuronidase
-
DOI 10.1023/A:1008857331429
-
DE Stevenson 1999 Optimisation of UDP-glucuronyl transferase-catalysed synthesis of testosterone-β-D-glucuronide by inhibition of contaminating -glucuronidase Biotechnol Tech 13 17 21 10.1023/A:1008857331429 1:CAS:528:DyaK1MXitVKhsLg%3D (Pubitemid 29114564)
-
(1999)
Biotechnology Techniques
, vol.13
, Issue.1
, pp. 17-21
-
-
Stevenson, D.E.1
-
16
-
-
0034103121
-
Identification of tamoxifen and metabolites in human male urine by GC/MS
-
DOI 10.1002/1099-0801(200005)14:3<180::AID-BMC958>3.0.CO;2-T
-
R Mihailescu HY Aboul-Enein MD Efstatide 2000 Identification of tamoxifen and metabolites in human male urine by GC/MS Biomed Chromatogr 14 180 183 10.1002/1099-0801(200005)14:3<180::AID-BMC958>3.0.CO;2-T 1:CAS:528:DC%2BD3cXjsF2murc%3D (Pubitemid 30255904)
-
(2000)
Biomedical Chromatography
, vol.14
, Issue.3
, pp. 180-183
-
-
Mihailescu, R.1
Aboul-Enein, H.Y.2
Efstatide, M.D.3
-
18
-
-
37149047201
-
131I labeling of tamoxifen and biodistribution studies in rats
-
DOI 10.1016/j.apradiso.2007.08.005, PII S0969804307002485
-
131I labeling of tamoxifen and biodistribution studies in rats Appl Radiat Isot 66 178 187 10.1016/j.apradiso.2007.08.005 1:CAS:528: DC%2BD2sXhsVKkurnI (Pubitemid 350256950)
-
(2008)
Applied Radiation and Isotopes
, vol.66
, Issue.2
, pp. 178-187
-
-
Biber Muftuler, F.Z.1
Unak, P.2
Teksoz, S.3
Acar, C.4
Yolcular, S.5
Yurekli, Y.6
-
19
-
-
33646503033
-
Synthesis of an estradiol glucuronide derivative and investigation of its radiopharmaceutical potential
-
10.1016/j.apradiso.2006.02.001 1:CAS:528:DC%2BD28XltVeru7s%3D
-
FZ Biber P Unak T Ertay EI Medine F Zihnioglu C TascI, et al. 2006 Synthesis of an estradiol glucuronide derivative and investigation of its radiopharmaceutical potential Appl Radiat Isot 64 778 788 10.1016/j.apradiso. 2006.02.001 1:CAS:528:DC%2BD28XltVeru7s%3D
-
(2006)
Appl Radiat Isot
, vol.64
, pp. 778-788
-
-
Biber, F.Z.1
Unak, P.2
Ertay, T.3
Medine, E.I.4
Zihnioglu, F.5
Tasci, C.6
-
21
-
-
0029904131
-
Synthesis, biodistribution, and estrogen receptor scintigraphy of indium- 111-diethylenetriaminepentaacetic acid-tamoxifen analogue
-
DOI 10.1021/js960049w
-
ES Delpassand DG Yang S Wallace A Cherif SM Quadri G Price, et al. 1996 Synthesis, biodistribution, and estrogen receptor scintigraphy of indium-111-diethyleneaminpentaacetic acid-tamoxifen analogue J Pharm Sci 85 553 559 10.1021/js960049w 1:CAS:528:DyaK28XivVCks7k%3D (Pubitemid 26179651)
-
(1996)
Journal of Pharmaceutical Sciences
, vol.85
, Issue.6
, pp. 553-559
-
-
Delpassand, E.S.1
Yang, D.J.2
Wallace, S.3
Cherif, A.4
Quadri, S.M.5
Price, J.6
Joubert, A.7
Inoue, T.8
Podoloff, D.A.9
-
22
-
-
0020530005
-
An antiestrogen binding protein in human tissues
-
1:CAS:528:DyaL3sXhtlOrtLo%3D
-
OL Kon 1983 An antiestrogen binding protein in human tissues J Biol Chem 258 3173 3177 1:CAS:528:DyaL3sXhtlOrtLo%3D
-
(1983)
J Biol Chem
, vol.258
, pp. 3173-3177
-
-
Kon, O.L.1
-
23
-
-
0023205362
-
Sex steroid receptors in the stomach, liver, pancreas, and gastrointestinal tract of the baboon
-
WB Winborn PJ Sheridan HC McGill 1987 Sex steroid in the stomach, liver, pancreas, and gastrointestinal tract of the baboon Gastroenterology 92 23 32 1:CAS:528:DyaL2sXmtFCjuw%3D%3D (Pubitemid 17207657)
-
(1987)
Gastroenterology
, vol.92
, Issue.1
, pp. 23-32
-
-
Winborn, W.B.1
Sheridan, P.J.2
McGill Jr., H.C.3
-
24
-
-
0028919090
-
Estrogen receptors in human nontarget tissues: Biological and clinical implications
-
1:CAS:528:DyaK2MXltlKhu7k%3D
-
DR Ciocca LM Vargas 1995 Estrogen receptors in human nontarget tissues: biological and clinical implications Endocr Rev 16 35 62 1:CAS:528: DyaK2MXltlKhu7k%3D
-
(1995)
Endocr Rev
, vol.16
, pp. 35-62
-
-
Ciocca, D.R.1
Vargas, L.M.2
-
26
-
-
33646519774
-
Attempts to develop a new nuclear measurement technique of β-glucuronidase levels in biological samples
-
10.1007/s10582-003-0104-x 1:CAS:528:DC%2BD3sXmsV2nsro%3D
-
T Unak U AvcIbaşI Y YIldIrIm B Cetinkaya 2003 Attempts to develop a new nuclear measurement technique of β-glucuronidase levels in biological samples Czechoslovak J Phys 53 A797 A802 10.1007/s10582-003-0104-x 1:CAS:528:DC%2BD3sXmsV2nsro%3D
-
(2003)
Czechoslovak J Phys
, vol.53
-
-
Unak, T.1
Avcibaşi, U.2
Yildirim, Y.3
Cetinkaya, B.4
-
27
-
-
0019506819
-
Clinical pharmacology of tamoxifen in patients with breast cancer: Correlation with clinical data
-
DOI 10.1002/1097-0142(19810815)48:4<876::AID-CNCR2820480403>3.0. CO;2-Q
-
C Fabian L Sternson M El-serafi L Cain E Hearne 1981 Clinical pharmacology of Tamoxifen in patients with breast cancer: correlation with clinical data Cancer 48 876 882 10.1002/1097-0142(19810815)48:4<876::AID- CNCR2820480403>3.0.CO;2-Q 1:STN:280:DyaL38%2FgtFygsw%3D%3D (Pubitemid 11049082)
-
(1981)
Cancer
, vol.48
, Issue.4
, pp. 876-882
-
-
Fabian, C.1
Sternson, L.2
El-Serafi, M.3
Hearne, E.4
-
28
-
-
0035255412
-
Synthesis and biological evaluation of two new radiolabelled estrogens: (125I)(E)-3-methoxy-17α-iodovinylestra-1,3,5(10),6-tetraen-17β-ol and (125I)(Z)-3-methoxy-17α-iodovinylestra-1,3,5(10),6-tetraen-17β-ol
-
10.1016/S0969-8043(99)00258-4
-
MC Silva P Luciana L Gano ML SáMelo E Inohae M Shuntaro, et al. 2001 Synthesis and biological evaluation of two new radiolabelled estrogens: (125I)(E)-3-methoxy-17α-iodovinylestra-1,3,5(10),6-tetraen-17β-ol and (125I)(Z)-3-methoxy-17α-iodovinylestra-1,3,5(10),6-tetraen-17β-ol Appl Radiat Isot 54 227 239 10.1016/S0969-8043(99)00258-4
-
(2001)
Appl Radiat Isot
, vol.54
, pp. 227-239
-
-
Silva, M.C.1
Luciana, P.2
Gano, L.3
Sámelo, M.L.4
Inohae, E.5
Shuntaro, M.6
-
29
-
-
0025007461
-
Amino and iodotamoxifens: Synthesis, estrogen receptor affinity and biodistribution
-
LA Strickland YZ Ponce DH Hunter PL Zabel JE Powe G Morrissey, et al. 1990 Amino and iodotamoxifens: synthesis estrogen receptor affinity and biodistribution Drug Des Deliv 6 195 212 1:CAS:528:DyaK3MXit1SrtrY%3D (Pubitemid 20302003)
-
(1990)
Drug Design and Delivery
, vol.6
, Issue.3
, pp. 195-212
-
-
Strickland, L.A.1
Ponce, Y.Z.2
Hunter, D.H.3
Zabel, P.L.4
Powe, J.E.5
Morrissey, G.6
Driedger, A.A.7
Chamberlain, M.J.8
Tustanoff, E.R.9
|