On the existence of a possible A2A-D2-β- arrestin2 complex: A2A agonist modulation of D2 agonist-induced β-arrestin2 recruitment

Journal of Molecular Biology

Volumn 406, Issue 5, 2011, Pages 687-699

  Borroto Escuela, Dasiel O ^a   Romero Fernandez, Wilber ^a   Tarakanov, Alexander O ^b   Ciruela, Francisco ^c   Agnati, Luigi F ^d   Fuxe, Kjell ^a  

^a KAROLINSKA INSTITUTE   (Sweden)

^b ST PETERSBURG INSTITUTE FOR INFORMATICS AND AUTOMATION   (Russian Federation)

^c UNIVERSITY OF BARCELONA   (Spain)

^d IRCCS   (Italy)

Author keywords

allosteric modulation; G protein coupled receptors; heteromerization; internalization; receptor protein interaction

Indexed keywords

2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A2A RECEPTOR; ADENOSINE A2A RECEPTOR AGONIST; BETA ARRESTIN 2; DOPAMINE 2 RECEPTOR; DOPAMINE 2 RECEPTOR STIMULATING AGENT; G PROTEIN COUPLED RECEPTOR; PROTEIN KINASE B; SCAFFOLD PROTEIN; 2 (4 (2 CARBOXYETHYL)PHENETHYLAMINO) 5' N ETHYLCARBOXAMIDOADENOSINE; 2-(4-(2-CARBOXYETHYL)PHENETHYLAMINO)-5'-N-ETHYLCARBOXAMIDOADENOSINE; ADENOSINE; ADENOSINE A2 RECEPTOR AGONIST; BETA ARRESTIN; DRUG DERIVATIVE; PHENETHYLAMINE DERIVATIVE; RETINA S ANTIGEN;

ARTICLE; BIOINFORMATICS; BIOLUMINESCENCE RESONANCE ENERGY TRANSFER; INTERNALIZATION; PRIORITY JOURNAL; PROTEIN PHOSPHORYLATION; PROTEIN PROTEIN INTERACTION; CELL LINE; CHEMICAL STRUCTURE; DRUG POTENTIATION; HUMAN; METABOLISM; PROTEIN BINDING; PROTEIN MULTIMERIZATION; PROTEIN QUATERNARY STRUCTURE;

ADENOSINE; ADENOSINE A2 RECEPTOR AGONISTS; ARRESTINS; CELL LINE; HUMANS; MODELS, MOLECULAR; PHENETHYLAMINES; PROTEIN BINDING; PROTEIN MULTIMERIZATION; PROTEIN STRUCTURE, QUATERNARY; RECEPTOR, ADENOSINE A2A; RECEPTORS, DOPAMINE D2;

EID: 79951771675     PISSN: 00222836     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jmb.2011.01.022     Document Type: Article

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