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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 5, 2011, Pages 1338-1341

Chroman and tetrahydroquinoline ureas as potent TRPV1 antagonists

(14) Schmidt, Robert G a Bayburt, Erol K a Latshaw, Steven P a Koenig, John R a Daanen, Jerome F a McDonald, Heath A a Bianchi, Bruce R a Zhong, Chengmin a Joshi, Shailen a Honore, Prisca a Marsh, Kennan C a Lee, Chih Hung a Faltynek, Connie R a Gomtsyan, Arthur a

a ABBOTT LABORATORIES (United States)

Author keywords

Chromanyl urea; Pain; Tetrahydroquinolinyl urea; TRPV1 antagonists

Indexed keywords

A 784168; ANALGESIC AGENT; CELECOXIB; CHROMAN DERIVATIVE; CYTOCHROME P450 3A4; DICLOFENAC; NITROGEN; QUINOLINE DERIVATIVE; UNCLASSIFIED DRUG; VANILLOID RECEPTOR 1 ANTAGONIST;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; ATOM; BLOOD BRAIN BARRIER; CHRONIC PAIN; CONTROLLED STUDY; DRUG EFFICACY; DRUG SCREENING; DRUG SYNTHESIS; IN VITRO STUDY; NONHUMAN; PAIN; RAT;

CHROMANS; HUMANS; INHIBITORY CONCENTRATION 50; MOLECULAR STRUCTURE; QUINOLINES; TRPV CATION CHANNELS; UREA;

EID: 79951726098 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2011.01.056 Document Type: Article

Times cited : (42)

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