Rigid backbone moiety of KNI-272, a highly selective HIV protease inhibitor: Methanol, acetone and dimethylsulfoxide solvated forms of 3-[3-benzyl-2-hydroxy-9-(isoquinolin-5-yloxy)-6-methyl-sulfanylmethyl-5, 8-dioxo-4,7-diazanonanoyl]-N-tert-butyl-1,3-thiazolidine-4-carboxamide

Acta Crystallographica Section B: Structural Science

Volumn 60, Issue 4, 2004, Pages 433-437

  Doi, Mitsunobu ^a   Kimura, Tooru ^b   Ishida, Toshimasa ^a   Kiso, Yoshiaki ^b  

^a OSAKA MEDICAL COLLEGE   (Japan)

^b KYOTO PHARMACEUTICAL UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

ACETONE; CONFORMATIONS; CRYSTAL STRUCTURE; ENZYME INHIBITION; METHANOL;

HYDROXYMETHYLCARBONYL (HMC); ISOQUINOLINE RING; KYNOSTATIN (KNI)-272 PROTEASE INHIBITORS;

ENZYME KINETICS;

HUMAN IMMUNODEFICIENCY VIRUS;

ACETONE; DIMETHYL SULFOXIDE; KYNOSTATIN 272; METHANOL; OLIGOPEPTIDE; PROTEINASE INHIBITOR; SOLVENT;

ARTICLE; CHEMICAL STRUCTURE; CHEMISTRY; CONFORMATION; X RAY CRYSTALLOGRAPHY;

ACETONE; CRYSTALLOGRAPHY, X-RAY; DIMETHYL SULFOXIDE; HIV PROTEASE INHIBITORS; METHANOL; MODELS, MOLECULAR; MOLECULAR CONFORMATION; MOLECULAR STRUCTURE; OLIGOPEPTIDES; SOLVENTS;

EID: 7944226840     PISSN: 01087681     EISSN: None     Source Type: Journal    
DOI: 10.1107/S0108768104013047     Document Type: Article

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