Efficient and novel one-pot synthesis of antifungal active 1-substituted-8-aryl-3-alkyl/aryl-4H-pyrazolo[4,5-f][1,2,4]triazolo[4,3-b][1,2, 4]triazepines using solid support

European Journal of Medicinal Chemistry

Volumn 46, Issue 2, 2011, Pages 631-635

  Gupta, Monika ^a   Paul, Satya ^a   Gupta, Rajive ^a  

^a UNIVERSITY OF JAMMU   (India)

Author keywords

Antifungal; Basic alumina; Microwave irradiation; N,N Dimethylformamide; p TsOH; Pyazolotriazolo triazepines

Indexed keywords

8 (4' CHLOROPHENYL) 3 METHYL 4H PYRAZOLO[4,5 F][1,2,4]TRIAZOLO[4,3 B][1,2,4]TRIAZEPINE; 8 PHENYL 3 METHYL 4H PYRAZOLO[4,5 F][1,2,4]TRIAZOLO[4,3 B][1,2,4]TRIAZEPINE; ANTIFUNGAL AGENT; FLUCONAZOLE; HETEROCYCLIC COMPOUND; N (4' BROMOPHENYL) 3,8 DIPHENYL 4H PYRAZOLO[4,5 F][1,2,4]TRIAZOLO[4,3 B][1,2,4]TRIAZEPINE; N (4' BROMOPHENYL) 8 (4' CHLOROPHENYL) 3 PHENYL 4H PYRAZOLO[4,5 F][1,2,4]TRIAZOLO[4,3 B][1,2,4]TRIAZEPINE; N (4' BROMOPHENYL) 8 (4' NITROPHENYL) 3 PHENYL 4H PYRAZOLO[4,5 F][1,2,4]TRIAZOLO[4,3 B][1,2,4]TRIAZEPINE; N (4' NITROPHENYL) 3,8 DIPHENYL 4H PYRAZOLO[4,5 F][1,2,4]TRIAZOLO[4,3 B][1,2,4]TRIAZEPINE; N (4' NITROPHENYL) 8 (4' NITROPHENYL) 3 PHENYL 4H PYRAZOLO[4,5 F][1,2,4]TRIAZOLO[4,3 B][1,2,4]TRIAZEPINE; N (4' NITROPHENYL) 8 BENZYL 3 PHENYL 4H PYRAZOLO[4,5 F][1,2,4]TRIAZOLO[4,3 B][1,2,4]TRIAZEPINE; N PHENYL 3,8 DIPHENYL 4H PYRAZOLO[4,5 F][1,2,4]TRIAZOLO[4,3 B][1,2,4]TRIAZEPINE; N PHENYL 8 BENZYL 3 (4' BROMOPHENYL) 4H PYRAZOLO[4,5 F][1,2,4]TRIAZOLO[4,3 B][1,2,4]TRIAZEPINE; N,N DIMETHYLFORMAMIDE; PYRAZOLONE DERIVATIVE; TRIAZEPINE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIFUNGAL ACTIVITY; ARTICLE; ASPERGILLUS FLAVUS; ASPERGILLUS NIGER; CATALYST; CONTROLLED STUDY; DRUG SCREENING; DRUG SYNTHESIS; ENERGY TRANSFER; MICROWAVE IRRADIATION; NONHUMAN; PENICILLIUM; RHIZOPUS;

ANTIFUNGAL AGENTS; ASPERGILLUS FLAVUS; ASPERGILLUS NIGER; AZEPINES; MICROBIAL SENSITIVITY TESTS; MICROWAVES; MOLECULAR STRUCTURE; PENICILLIUM; RHIZOPUS; STEREOISOMERISM; TRIAZOLES;

EID: 79151475534     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2010.11.043     Document Type: Article

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