Synthesis and evaluation of anti-tubercular activity of new dithiocarbamate sugar derivatives

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 3, 2011, Pages 899-903

  Horita, Yasuhiro ^a,c   Takii, Takemasa ^a   Kuroishi, Ryuji ^a   Chiba, Taku ^b   Ogawa, Kenji ^c   Kremer, Laurent ^d   Sato, Yasuo ^e   Lee, Yoosa ^a   Hasegawa, Tomohiro ^a   Onozaki, Kikuo ^a  

^a NAGOYA CITY UNIVERSITY   (Japan)

^b KINJO GAKUIN UNIVERSITY   (Japan)

^c National Hospital Organization Higashinagoya National Hospital   (Japan)

^d UNIVERSITÉ DE MONTPELLIER   (France)

^e MEIJI DAIRIES CORPORATION   (Japan)

Author keywords

Dithiocarbamate; Mycobacterium tuberculosis; N Acetyl glucosamine; Pyrrolidine

Indexed keywords

2 ACETAMIDO 2 DEOXY BETA GLUCOPYRANOSYL N,N DIMETHYLDITHIOCARBAMATE; 2 ACETAMIDO 2 DEOXY BETA GLUCOPYRANOSYLPYRROLIDINE DITHIOCARBAMATE; DITHIOCARBAMIC ACID DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIBIOTIC RESISTANCE; ARTICLE; BACTERICIDAL ACTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; MINIMUM INHIBITORY CONCENTRATION; MULTIDRUG RESISTANCE; MYCOBACTERIUM AVIUM; MYCOBACTERIUM BOVIS; MYCOBACTERIUM SMEGMATIS; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; STAPHYLOCOCCUS AUREUS;

ANTITUBERCULAR AGENTS; CARBOHYDRATES; DRUG RESISTANCE, BACTERIAL; MICROBIAL SENSITIVITY TESTS; MYCOBACTERIUM TUBERCULOSIS; OXIDOREDUCTASES; THIOCARBAMATES; THIOGLUCOSIDES;

ESCHERICHIA COLI; MYCOBACTERIUM AVIUM; MYCOBACTERIUM BOVIS BCG; MYCOBACTERIUM SMEGMATIS; MYCOBACTERIUM TUBERCULOSIS; STAPHYLOCOCCUS AUREUS;

EID: 78751702936     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.12.084     Document Type: Article

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