CGP-37157 inhibits the sarcoplasmic reticulum Ca 2+ ATPase and activates ryanodine receptor channels in striated muscle

Molecular Pharmacology

Volumn 79, Issue 1, 2011, Pages 141-147

  Neumann, Jake T ^a   Diaz Sylvester, Paula L ^a   Fleischer, Sidney ^b   Copello, Julio A ^a  

^a SOUTHERN ILLINOIS UNIVERSITY SCHOOL OF MEDICINE   (United States)

^b VANDERBILT UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

7 CHLORO 5 (2 CHLOROPHENYL) 1,5 DIHYDRO 4,1 BENZOTHIAZEPIN 2(3H) ONE; ADENOSINE TRIPHOSPHATASE (CALCIUM); RUTHENIUM RED; RYANODINE RECEPTOR; SARCOPLASMIC RETICULUM CALCIUM TRANSPORTING ADENOSINE TRIPHOSPHATASE;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CALCIUM TRANSPORT; CONCENTRATION RESPONSE; CORRELATION ANALYSIS; DRUG ACTIVITY; ENZYME ACTIVITY; HEART MUSCLE; LIPID BILAYER; MICROSOME; NONHUMAN; PRIORITY JOURNAL; SARCOPLASMIC RETICULUM; SKELETAL MUSCLE;

ANIMALS; CALCIUM; CALCIUM-TRANSPORTING ATPASES; CLONAZEPAM; MUSCLE, STRIATED; RABBITS; RYANODINE RECEPTOR CALCIUM RELEASE CHANNEL; SARCOPLASMIC RETICULUM; THIAZEPINES;

EID: 78651329211     PISSN: 0026895X     EISSN: 15210111     Source Type: Journal    
DOI: 10.1124/mol.110.067165     Document Type: Article

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