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Volumn 404, Issue 1-2, 2011, Pages 75-82

Unintended potential impact of perfect sink conditions on PLGA degradation in microparticles

Author keywords

Controlled release; Microparticles; PLGA; Release conditions; Sink conditions

Indexed keywords

CARBAMAZEPINE; IBUPROFEN; POLYGLACTIN; RESOMER RG 504H; UNCLASSIFIED DRUG;

EID: 78650678085     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2010.10.054     Document Type: Article
Times cited : (36)

References (42)
  • 1
    • 0343247711 scopus 로고    scopus 로고
    • Biodegradation and biocompatibility of PLA and PLGA microspheres
    • J.M. Anderson, and M.S. Shive Biodegradation and biocompatibility of PLA and PLGA microspheres Adv. Drug Del. Rev. 28 1997 5 24
    • (1997) Adv. Drug Del. Rev. , vol.28 , pp. 5-24
    • Anderson, J.M.1    Shive, M.S.2
  • 2
    • 0035997340 scopus 로고    scopus 로고
    • A novel in vitro delivery system for assessing the biological integrity of protein upon release from PLGA microspheres
    • A. Aubert-Pouëssel, D.C. Bibby, M.C. Venier-Julienne, F. Hindré, and J.P. Benoit A novel in vitro delivery system for assessing the biological integrity of protein upon release from PLGA microspheres Pharm. Res. 19 2002 1046 1051
    • (2002) Pharm. Res. , vol.19 , pp. 1046-1051
    • Aubert-Pouëssel, A.1    Bibby, D.C.2    Venier-Julienne, M.C.3    Hindré, F.4    Benoit, J.P.5
  • 3
    • 0032904287 scopus 로고    scopus 로고
    • Modulation of rifampicin release from spray-dried microspheres using combinations of poly-(dl-lactide)
    • D.F. Bain, D.L. Munday, and A. Smith Modulation of rifampicin release from spray-dried microspheres using combinations of poly-(dl-lactide) J. Microencapsul. 16 1999 369 385
    • (1999) J. Microencapsul. , vol.16 , pp. 369-385
    • Bain, D.F.1    Munday, D.L.2    Smith, A.3
  • 4
    • 0038537239 scopus 로고    scopus 로고
    • PLG microsphere size controls drug release rate through several competing factors
    • C. Berkland, K. Kim, and D.W. Pack PLG microsphere size controls drug release rate through several competing factors Pharm. Res. 20 2003 1055 1062
    • (2003) Pharm. Res. , vol.20 , pp. 1055-1062
    • Berkland, C.1    Kim, K.2    Pack, D.W.3
  • 5
    • 0033026897 scopus 로고    scopus 로고
    • PH and osmotic pressure inside biodegradable microspheres during erosion
    • A. Brunner, K. Maeder, and A. Goepferich pH and osmotic pressure inside biodegradable microspheres during erosion Pharm. Res. 16 1999 847 853
    • (1999) Pharm. Res. , vol.16 , pp. 847-853
    • Brunner, A.1    Maeder, K.2    Goepferich, A.3
  • 6
    • 1842555130 scopus 로고    scopus 로고
    • Assuring quality and performance of sustained and controlled release parenterals
    • D. Burgess, D. Crommelin, A. Hussain, and M. Chen Assuring quality and performance of sustained and controlled release parenterals Eur. J. Pharm. Sci. 21 2004 679 690
    • (2004) Eur. J. Pharm. Sci. , vol.21 , pp. 679-690
    • Burgess, D.1    Crommelin, D.2    Hussain, A.3    Chen, M.4
  • 7
    • 0036845762 scopus 로고    scopus 로고
    • Assuring quality and performance of sustained and controlled release parenterals: AAPS workshop report, co-sponsored by FDA and USP
    • D. Burgess, A.S. Hussain, T.S. Ingallinera, and M.L. Chen Assuring quality and performance of sustained and controlled release parenterals: AAPS workshop report, co-sponsored by FDA and USP Pharm. Res. 19 2002 1761 1768
    • (2002) Pharm. Res. , vol.19 , pp. 1761-1768
    • Burgess, D.1    Hussain, A.S.2    Ingallinera, T.S.3    Chen, M.L.4
  • 8
    • 0028944513 scopus 로고
    • Testing of "in vitro" dissolution behaviour of microparticulate drug delivery systems
    • C.B. Conti, I. Genta, P. Giunchedi, and T. Modena Testing of "in vitro" dissolution behaviour of microparticulate drug delivery systems Drug Dev. Ind. Pharm. 21 1995 1223 1233
    • (1995) Drug Dev. Ind. Pharm. , vol.21 , pp. 1223-1233
    • Conti, C.B.1    Genta, I.2    Giunchedi, P.3    Modena, T.4
  • 9
    • 33644984488 scopus 로고    scopus 로고
    • Methods to assess in vitro drug release from injectable polymeric particulate systems
    • S. D'Souza, and P.P. DeLuca Methods to assess in vitro drug release from injectable polymeric particulate systems Pharm. Res. 23 2006 460 474
    • (2006) Pharm. Res. , vol.23 , pp. 460-474
    • D'Souza, S.1    Deluca, P.P.2
  • 10
    • 27744494863 scopus 로고    scopus 로고
    • Development of a dialysis in vitro release method for biodegradable microspheres
    • S. D'Souza, and P.P. DeLuca Development of a dialysis in vitro release method for biodegradable microspheres AAPS PharmSciTech 6 2005 323 328
    • (2005) AAPS PharmSciTech , vol.6 , pp. 323-328
    • D'Souza, S.1    Deluca, P.P.2
  • 11
    • 0034036366 scopus 로고    scopus 로고
    • Influence of particle size and dissolution conditions on the degradation properties of polylactide-co-glycolide particles
    • M. Dunne, O.I. Corrigan, and Z. Ramtoola Influence of particle size and dissolution conditions on the degradation properties of polylactide-co-glycolide particles Biomaterials 21 2000 1659 1668
    • (2000) Biomaterials , vol.21 , pp. 1659-1668
    • Dunne, M.1    Corrigan, O.I.2    Ramtoola, Z.3
  • 12
    • 33646188402 scopus 로고    scopus 로고
    • Effects of the type of release medium on drug release from PLGA-based microparticles: Experiment and theory
    • N. Faisant, J. Akiki, F. Siepmann, J.P. Benoit, and J. Siepmann Effects of the type of release medium on drug release from PLGA-based microparticles: experiment and theory Int. J. Pharm. 314 2006 189 197
    • (2006) Int. J. Pharm. , vol.314 , pp. 189-197
    • Faisant, N.1    Akiki, J.2    Siepmann, F.3    Benoit, J.P.4    Siepmann, J.5
  • 13
    • 0037619257 scopus 로고    scopus 로고
    • Biocompatibility of implantable synthetic polymeric drug carriers: Focus on brain biocompatibility
    • E. Fournier, C. Passirani, C.N. Montero-Menei, and J.P. Benoit Biocompatibility of implantable synthetic polymeric drug carriers: focus on brain biocompatibility Biomaterials 24 2003 3311 3331
    • (2003) Biomaterials , vol.24 , pp. 3311-3331
    • Fournier, E.1    Passirani, C.2    Montero-Menei, C.N.3    Benoit, J.P.4
  • 14
    • 11844289546 scopus 로고    scopus 로고
    • Controlled release from bioerodible polymers: Effect of drug type and polymer composition
    • A. Frank, S.K. Rath, and S.S. Venkatraman Controlled release from bioerodible polymers: effect of drug type and polymer composition J. Control. Release 102 2005 333 344
    • (2005) J. Control. Release , vol.102 , pp. 333-344
    • Frank, A.1    Rath, S.K.2    Venkatraman, S.S.3
  • 15
    • 4444246813 scopus 로고    scopus 로고
    • Polymer microspheres for controlled drug release
    • S. Freiberg, and X.X. Zhu Polymer microspheres for controlled drug release Int. J. Pharm. 282 2004 1 18
    • (2004) Int. J. Pharm. , vol.282 , pp. 1-18
    • Freiberg, S.1    Zhu, X.X.2
  • 16
    • 0034006495 scopus 로고    scopus 로고
    • Visual evidence of acidic environment within degrading poly(lactic-co-glycolic acid) (PLGA) microspheres
    • K. Fu, D.W. Pack, A.M. Klibanov, and R. Langer Visual evidence of acidic environment within degrading poly(lactic-co-glycolic acid) (PLGA) microspheres Pharm. Res. 17 2000 100 106
    • (2000) Pharm. Res. , vol.17 , pp. 100-106
    • Fu, K.1    Pack, D.W.2    Klibanov, A.M.3    Langer, R.4
  • 17
    • 0029256583 scopus 로고
    • Hydrolytic degradation of devices based on poly(dl-lactic acid) size dependence
    • I. Grizzi, S.L. Garreau, and M. Vert Hydrolytic degradation of devices based on poly(dl-lactic acid) size dependence Biomaterials 16 1995 305 311
    • (1995) Biomaterials , vol.16 , pp. 305-311
    • Grizzi, I.1    Garreau, S.L.2    Vert, M.3
  • 18
    • 33847185185 scopus 로고    scopus 로고
    • Pore closing and opening in biodegradable polymers and their effect on the controlled release of proteins
    • J. Kang, and S.P. Schwendeman Pore closing and opening in biodegradable polymers and their effect on the controlled release of proteins Mol. Pharm. 4 2007 104 118
    • (2007) Mol. Pharm. , vol.4 , pp. 104-118
    • Kang, J.1    Schwendeman, S.P.2
  • 19
    • 33845281956 scopus 로고
    • Poly(lactide-co-glycolide) decomposition kinetics in vivo and in vitro
    • R.A. Kenley, M.O. Lee, T.R. Mahoney, and L.M. Sanders Poly(lactide-co-glycolide) decomposition kinetics in vivo and in vitro Macromolecules 20 1987 2398 2403
    • (1987) Macromolecules , vol.20 , pp. 2398-2403
    • Kenley, R.A.1    Lee, M.O.2    Mahoney, T.R.3    Sanders, L.M.4
  • 20
    • 33646176224 scopus 로고    scopus 로고
    • How porosity and size affect the drug release mechanisms from PLGA-based microparticles
    • D. Klose, F. Siepmann, K. Elkharraz, S. Krenzlin, and J. Siepmann How porosity and size affect the drug release mechanisms from PLGA-based microparticles Int. J. Pharm. 314 2006 198 206
    • (2006) Int. J. Pharm. , vol.314 , pp. 198-206
    • Klose, D.1    Siepmann, F.2    Elkharraz, K.3    Krenzlin, S.4    Siepmann, J.5
  • 21
    • 40949133332 scopus 로고    scopus 로고
    • PLGA-based drug delivery systems: Importance of the type of drug and device geometry
    • D. Klose, F. Siepmann, K. Elkharraz, and J. Siepmann PLGA-based drug delivery systems: Importance of the type of drug and device geometry Int. J. Pharm. 354 2008 95 103
    • (2008) Int. J. Pharm. , vol.354 , pp. 95-103
    • Klose, D.1    Siepmann, F.2    Elkharraz, K.3    Siepmann, J.4
  • 22
    • 70449710805 scopus 로고    scopus 로고
    • Drug release from PLGA-based microparticles: Effects of the "microparticle:bulk fluid" ratio
    • D. Klose, F. Siepmann, J.F. Willart, M. Descamps, and J. Siepmann Drug release from PLGA-based microparticles: effects of the "microparticle:bulk fluid" ratio Int. J. Pharm. 383 2010 123 131
    • (2010) Int. J. Pharm. , vol.383 , pp. 123-131
    • Klose, D.1    Siepmann, F.2    Willart, J.F.3    Descamps, M.4    Siepmann, J.5
  • 23
    • 19244381301 scopus 로고    scopus 로고
    • A novel in vitro release technique for peptide containing biodegradable microspheres
    • J.W. Kostanski, and P.P. DeLuca A novel in vitro release technique for peptide containing biodegradable microspheres AAPS PharmSciTech. 1 2000 E4
    • (2000) AAPS PharmSciTech. , vol.1 , pp. 4
    • Kostanski, J.W.1    Deluca, P.P.2
  • 24
    • 10044272241 scopus 로고    scopus 로고
    • Mapping neutral microclimate pH in PLGA microspheres
    • L. Li, and S.P. Schwendeman Mapping neutral microclimate pH in PLGA microspheres J. Control. Release 101 2005 163 173
    • (2005) J. Control. Release , vol.101 , pp. 163-173
    • Li, L.1    Schwendeman, S.P.2
  • 25
    • 0031808578 scopus 로고    scopus 로고
    • Evaluation of a novel phase separation technique for the encapsulation of water-soluble drugs in biodegradable polymer
    • T.K. Mandal Evaluation of a novel phase separation technique for the encapsulation of water-soluble drugs in biodegradable polymer Drug Dev. Ind. Pharm. 24 1998 623 629
    • (1998) Drug Dev. Ind. Pharm. , vol.24 , pp. 623-629
    • Mandal, T.K.1
  • 26
    • 45249109321 scopus 로고    scopus 로고
    • In vitro and in vivo considerations associated with parenteral sustained release products: A review based upon information presented and points expressed at the 2007 Controlled Release Society Annual Meeting
    • M. Martinez, M. Rathbone, D. Burgess, and M. Huynh In vitro and in vivo considerations associated with parenteral sustained release products: a review based upon information presented and points expressed at the 2007 Controlled Release Society Annual Meeting J. Control. Release 129 2008 79 87
    • (2008) J. Control. Release , vol.129 , pp. 79-87
    • Martinez, M.1    Rathbone, M.2    Burgess, D.3    Huynh, M.4
  • 27
    • 76749157815 scopus 로고    scopus 로고
    • Breakout session summary from AAPS/CRS joint workshop on critical variables in the in vitro and in vivo performance of parenteral sustained release products
    • M.N. Martinez, M.J. Rathbone, D. Burgess, and M. Huynh Breakout session summary from AAPS/CRS joint workshop on critical variables in the in vitro and in vivo performance of parenteral sustained release products J. Control. Release 142 2010 2 7
    • (2010) J. Control. Release , vol.142 , pp. 2-7
    • Martinez, M.N.1    Rathbone, M.J.2    Burgess, D.3    Huynh, M.4
  • 29
    • 0034580276 scopus 로고    scopus 로고
    • Synthetic biodegradable polymers as orthopedic devices
    • J.C. Middleton, and A.J. Tipton Synthetic biodegradable polymers as orthopedic devices Biomaterials 21 2000 2335 2346
    • (2000) Biomaterials , vol.21 , pp. 2335-2346
    • Middleton, J.C.1    Tipton, A.J.2
  • 30
    • 0343683341 scopus 로고    scopus 로고
    • Preparation of microspheres by the solvent evaporation technique
    • P.B. O'Donnell, and J.W. McGinity Preparation of microspheres by the solvent evaporation technique Adv. Drug Del. Rev. 28 1997 25 42
    • (1997) Adv. Drug Del. Rev. , vol.28 , pp. 25-42
    • O'Donnell, P.B.1    McGinity, J.W.2
  • 31
    • 0028319146 scopus 로고
    • Degradation of poly(image-lactic acid) microspheres: Effect of molecular weight
    • T.G. Park Degradation of poly(image-lactic acid) microspheres: effect of molecular weight J. Control. Release 30 1994 161 173
    • (1994) J. Control. Release , vol.30 , pp. 161-173
    • Park, T.G.1
  • 32
    • 0033846774 scopus 로고    scopus 로고
    • Polymer and microsphere blending to alter the release of a peptide from PLGA microspheres
    • H.B. Ravivarapu, K. Burton, and P.P. DeLuca Polymer and microsphere blending to alter the release of a peptide from PLGA microspheres Eur. J. Pharm. Biopharm. 50 2000 263 270
    • (2000) Eur. J. Pharm. Biopharm. , vol.50 , pp. 263-270
    • Ravivarapu, H.B.1    Burton, K.2    Deluca, P.P.3
  • 33
    • 0028808125 scopus 로고
    • Effects of H+ liberated from hydrolytic cleavage of polyester microcapsules on their permeability and degradability
    • H. Sah, and Y.W. Chien Effects of H+ liberated from hydrolytic cleavage of polyester microcapsules on their permeability and degradability J. Pharm. Sci. 84 1995 1353 1359
    • (1995) J. Pharm. Sci. , vol.84 , pp. 1353-1359
    • Sah, H.1    Chien, Y.W.2
  • 34
    • 0027327772 scopus 로고
    • Influence of manufacturing parameters on the size characteristics and the release profiles of nifedipine from poly(-lactide-co-glycolide) microspheres
    • S.P. Sansdrap, and A.J. Moës Influence of manufacturing parameters on the size characteristics and the release profiles of nifedipine from poly(-lactide-co-glycolide) microspheres Int. J. Pharm. 98 1993 157 164
    • (1993) Int. J. Pharm. , vol.98 , pp. 157-164
    • Sansdrap, S.P.1    Moës, A.J.2
  • 35
    • 33947180013 scopus 로고    scopus 로고
    • A short term (accelerated release) approach to evaluate peptide release from PLGA depot-formulations
    • M. Shameem, H. Lee, and P.P. DeLuca A short term (accelerated release) approach to evaluate peptide release from PLGA depot-formulations AAPS PharmSci. 1 1999 E7
    • (1999) AAPS PharmSci. , vol.1 , pp. 7
    • Shameem, M.1    Lee, H.2    Deluca, P.P.3
  • 36
    • 22944480893 scopus 로고    scopus 로고
    • How autocatalysis accelerates drug release from PLGA-based microparticles: A quantitative treatment
    • J. Siepmann, K. Elkharraz, F. Siepmann, and D. Klose How autocatalysis accelerates drug release from PLGA-based microparticles: a quantitative treatment Biomacromolecules 6 2005 2312 2319
    • (2005) Biomacromolecules , vol.6 , pp. 2312-2319
    • Siepmann, J.1    Elkharraz, K.2    Siepmann, F.3    Klose, D.4
  • 37
    • 0141800053 scopus 로고    scopus 로고
    • FIP/AAPS guidelines to dissolution/in vitro release testing of novel/special dosage forms
    • M. Siewert, J. Dressman, C.K. Brown, and V.P. Shah FIP/AAPS guidelines to dissolution/in vitro release testing of novel/special dosage forms AAPS PharmSciTech. 4 2003 pE7
    • (2003) AAPS PharmSciTech. , vol.4 , pp. 7
    • Siewert, M.1    Dressman, J.2    Brown, C.K.3    Shah, V.P.4
  • 38
    • 12844273562 scopus 로고    scopus 로고
    • Reduction in the initial-burst release by surface crosslinking of PLGA microparticles containing hydrophilic or hydrophobic drugs
    • A.J. Thote, J.T. Chappell, R.B. Gupta, and R. Kumar Reduction in the initial-burst release by surface crosslinking of PLGA microparticles containing hydrophilic or hydrophobic drugs Drug Dev. Ind. Pharm. 31 2005 43 57
    • (2005) Drug Dev. Ind. Pharm. , vol.31 , pp. 43-57
    • Thote, A.J.1    Chappell, J.T.2    Gupta, R.B.3    Kumar, R.4
  • 39
    • 72149091750 scopus 로고    scopus 로고
    • Physicochemical property profiles of marketed drugs, clinical candidates and bioactive compounds
    • C. Tyrchan, N. Blomberg, O. Engkvist, T. Kogej, and S. Muresan Physicochemical property profiles of marketed drugs, clinical candidates and bioactive compounds Bioorg. Med. Chem. Lett. 19 2009 6943 6947
    • (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 6943-6947
    • Tyrchan, C.1    Blomberg, N.2    Engkvist, O.3    Kogej, T.4    Muresan, S.5
  • 40
    • 2542461982 scopus 로고    scopus 로고
    • In vitro degradation of three-dimensional porous poly(d,l-lactide-co- glycolide) scaffolds for tissue engineering
    • L. Wu, and J. Ding In vitro degradation of three-dimensional porous poly(d,l-lactide-co-glycolide) scaffolds for tissue engineering Biomaterials 25 2004 5821 5830
    • (2004) Biomaterials , vol.25 , pp. 5821-5830
    • Wu, L.1    Ding, J.2
  • 41
    • 40949156307 scopus 로고    scopus 로고
    • Solubilisation of drugs in worm-like micelles of block copolymers of ethylene oxide and 1,2-butylene oxide in aqueous solution
    • Z. Zhou, C. Chaibundit, A. D'Emanuele, K. Lennon, D. Attwood, and C. Booth Solubilisation of drugs in worm-like micelles of block copolymers of ethylene oxide and 1,2-butylene oxide in aqueous solution Int. J. Pharm. 354 2008 82 87
    • (2008) Int. J. Pharm. , vol.354 , pp. 82-87
    • Zhou, Z.1    Chaibundit, C.2    D'Emanuele, A.3    Lennon, K.4    Attwood, D.5    Booth, C.6
  • 42
    • 33646676075 scopus 로고    scopus 로고
    • Elevated temperature accelerated release testing of PLGA microspheres
    • B.S. Zolnik, P.E. Leary, and D. Burgess Elevated temperature accelerated release testing of PLGA microspheres J. Control. Release 112 2006 293 300
    • (2006) J. Control. Release , vol.112 , pp. 293-300
    • Zolnik, B.S.1    Leary, P.E.2    Burgess, D.3


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