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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 1, 2011, Pages 584-587

Identification of novel pyrrolopyrazoles as protein kinase C β II inhibitors

(16) Li, Hui a Hong, Yufeng a Nukui, Seiji a Lou, Jihong a Johnson, Sarah a Scales, Stephanie a Botrous, Iriny a Tompkins, Eileen a Yin, Chunfeng a Zhou, Ru a He, Mingying a Jensen, Jordan a Bouzida, Djamal a Alton, Gordon a Lafontaine, Jennifer a Grant, Stephan a

a PFIZER INC (United States)

Author keywords

Diabetic complications; Kinase inhibitor; Protein kinase C; Pyrrolopyrazole

Indexed keywords

PROTEIN KINASE C BETA INHIBITOR; PYRROLOPYRAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CELL PERMEABILIZATION; COLUMN CHROMATOGRAPHY; DRUG ACTIVITY; DRUG SYNTHESIS; HIGH THROUGHPUT SCREENING; HUMAN; HUMAN CELL; HYDROGEN BOND;

HIGH-THROUGHPUT SCREENING ASSAYS; PROTEIN KINASE C; PROTEIN KINASE INHIBITORS; PYRAZOLES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 78650513218 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.10.032 Document Type: Article

Times cited : (13)

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