A facile, click chemistry-based approach to assembling fluorescent chemosensors for protein tyrosine kinases

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 1, 2011, Pages 329-331

  Kamaruddin, Mohd Aizuddin ^a   Ung, Phuc ^b   Hossain, Mohammed Iqbal ^a   Jarasrassamee, Boonyarin ^a   O'Malley, William ^b   Thompson, Philip ^b   Scanlon, Denis ^c   Cheng, Heung Chin ^a   Graham, Bim ^b  

^a UNIVERSITY OF MELBOURNE   (Australia)

^b MONASH UNIVERSITY   (Australia)

^c UNIVERSITY OF MELBOURNE   (Australia)

Author keywords

Click chemistry; Fluorescence assays; Peptides; Tyrosine kinases

Indexed keywords

COPPER; IMATINIB; PROTEIN KINASE LYN; PROTEIN TYROSINE KINASE; STEROID RECEPTOR COACTIVATOR 1;

ARTICLE; CHEMICAL ANALYSIS; CHEMICAL REACTION; CHEMICAL STRUCTURE; ENZYME ACTIVITY; ENZYME PHOSPHORYLATION; FLUORESCENCE ANALYSIS; SCREENING; SYNTHESIS;

AMINO ACID SEQUENCE; BIOSENSING TECHNIQUES; CELL LINE, TUMOR; CLICK CHEMISTRY; ENZYME ASSAYS; FLUORESCENT DYES; HIGH-THROUGHPUT SCREENING ASSAYS; HUMANS; PEPTIDES; PHOSPHORYLATION; SRC-FAMILY KINASES; SUBSTRATE SPECIFICITY;

EID: 78650512710     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.11.005     Document Type: Article

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