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Volumn 62, Issue 11, 2010, Pages 1534-1546

Factors affecting crystallization of hydrates

Author keywords

crystallization; hydrate; kinetics; salt; thermodynamics

Indexed keywords

INORGANIC SALT;

EID: 78649671797     PISSN: 00223573     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.2042-7158.2010.01186.x     Document Type: Review
Times cited : (81)

References (98)
  • 1
    • 84890662885 scopus 로고    scopus 로고
    • The importance of solvates
    • In: Hilfiker R., ed. Weinheim: Wiley-VCH Verlag GmbH & Co
    • Griesser UJ,. The importance of solvates. In:, Hilfiker R, ed. Polymorphism in the Pharmaceutical Industry. Weinheim: Wiley-VCH Verlag GmbH & Co., 2006: 211-257.
    • (2006) Polymorphism in the Pharmaceutical Industry , pp. 211-257
    • Griesser, U.J.1
  • 3
    • 0002095772 scopus 로고    scopus 로고
    • Structural aspects of hydrates and solvates
    • In: Brittain H.G., ed. New York: Marcel Dekker
    • Morris KR,. Structural aspects of hydrates and solvates. In:, Brittain HG, ed. Polymorphism in Pharmaceutical Solids. New York: Marcel Dekker, 1999: 125-181.
    • (1999) Polymorphism in Pharmaceutical Solids , pp. 125-181
    • Morris, K.R.1
  • 4
    • 0031958398 scopus 로고    scopus 로고
    • Formation of isomorphic desolvates: Creating a molecular vacuum
    • Stephenson GA, et al. Formation of isomorphic desolvates: creating a molecular vacuum. J Pharm Sci 1998; 87: 536-542.
    • (1998) J Pharm Sci , vol.87 , pp. 536-542
    • Stephenson, G.A.1
  • 5
    • 0014915329 scopus 로고
    • Crystal pseudopolymorphism of cephaloglycin and cephalexin
    • Pfeiffer RR, et al. Crystal pseudopolymorphism of cephaloglycin and cephalexin. J Pharm Sci 1970; 59: 1809-1812.
    • (1970) J Pharm Sci , vol.59 , pp. 1809-1812
    • Pfeiffer, R.R.1
  • 6
    • 0032726149 scopus 로고    scopus 로고
    • Solid-state behavior of cromolyn sodium hydrates
    • Chen LR, et al. Solid-state behavior of cromolyn sodium hydrates. J Pharm Sci 1999; 88: 1191-1200.
    • (1999) J Pharm Sci , vol.88 , pp. 1191-1200
    • Chen, L.R.1
  • 7
    • 23844505711 scopus 로고    scopus 로고
    • Effect of salt type on hygroscopicity of a new cephalosporin S-3578
    • Kawakami K, et al. Effect of salt type on hygroscopicity of a new cephalosporin S-3578. Pharm Res 2005; 22: 1365-1373.
    • (2005) Pharm Res , vol.22 , pp. 1365-1373
    • Kawakami, K.1
  • 8
    • 32644460308 scopus 로고    scopus 로고
    • A study of variable hydration states in topotecan hydrochloride
    • Vogt FG, et al. A study of variable hydration states in topotecan hydrochloride. J Pharm Biomed Anal 2006; 40: 1080-1088.
    • (2006) J Pharm Biomed Anal , vol.40 , pp. 1080-1088
    • Vogt, F.G.1
  • 9
    • 70349229288 scopus 로고    scopus 로고
    • Structural characterisation and dehydration behaviour of siramesine hydrochloride
    • Zimmermann A, et al. Structural characterisation and dehydration behaviour of siramesine hydrochloride. J Pharm Sci 2009; 98: 3596-3607.
    • (2009) J Pharm Sci , vol.98 , pp. 3596-3607
    • Zimmermann, A.1
  • 11
    • 0037296654 scopus 로고    scopus 로고
    • Three hydrates of the bisphosphonate risedronate, consisting of one molecular and two ionic structures
    • Gossman WL, et al. Three hydrates of the bisphosphonate risedronate, consisting of one molecular and two ionic structures. Acta Crystallogr C 2003; 59: m33-m36.
    • (2003) Acta Crystallogr C , vol.59
    • Gossman, W.L.1
  • 12
    • 0031658908 scopus 로고    scopus 로고
    • Physical characterization of nedocromil sodium hydrates
    • Khankari RL, et al. Physical characterization of nedocromil sodium hydrates. J Pharm Sci 2000; 87: 1052-1061.
    • (2000) J Pharm Sci , vol.87 , pp. 1052-1061
    • Khankari, R.L.1
  • 13
    • 33748181565 scopus 로고    scopus 로고
    • Cefdinir: A comparative study of anhydrous vs. monohydrate form: Microstructure and tabletting behavior
    • Cabri W, et al. Cefdinir: a comparative study of anhydrous vs. monohydrate form: microstructure and tabletting behavior. Eur J Pharm Biopharm 2006; 64: 212-221.
    • (2006) Eur J Pharm Biopharm , vol.64 , pp. 212-221
    • Cabri, W.1
  • 14
    • 0026045869 scopus 로고
    • Characterization of polymorphs of tranilast anhydrate and tranilast monohydrate when crystallized by two solvent change spherical crystallization techniques
    • Yoshiaki K, et al. Characterization of polymorphs of tranilast anhydrate and tranilast monohydrate when crystallized by two solvent change spherical crystallization techniques. J Pharm Sci 1991; 80: 472-478.
    • (1991) J Pharm Sci , vol.80 , pp. 472-478
    • Yoshiaki, K.1
  • 15
    • 0017861035 scopus 로고
    • Physical characterization of erythromycin: Anhydrate, monohydrate, and dihydrate crystalline solids
    • Allen PV, et al. Physical characterization of erythromycin: anhydrate, monohydrate, and dihydrate crystalline solids. J Pharm Sci 1978; 67: 1087-1093.
    • (1978) J Pharm Sci , vol.67 , pp. 1087-1093
    • Allen, P.V.1
  • 16
    • 0035680440 scopus 로고    scopus 로고
    • Characterization of the solubility and dissolution properties of several new rifampicin polymorphs, solvates, and hydrates
    • Henwood SQ, et al. Characterization of the solubility and dissolution properties of several new rifampicin polymorphs, solvates, and hydrates. Drug Dev Ind Pharm 2001; 27: 1017-1030.
    • (2001) Drug Dev Ind Pharm , vol.27 , pp. 1017-1030
    • Henwood, S.Q.1
  • 17
    • 33846212349 scopus 로고    scopus 로고
    • In-situ measurement of solvent mediated phase transformations during dissolution testing
    • Aaltonen J, et al. In-situ measurement of solvent mediated phase transformations during dissolution testing. J Pharm Sci 2006; 95: 2730-2737.
    • (2006) J Pharm Sci , vol.95 , pp. 2730-2737
    • Aaltonen, J.1
  • 18
    • 57349098391 scopus 로고    scopus 로고
    • Better understanding of dissolution behaviour of amorphous drugs by in situ solid-state analysis using Raman spectroscopy
    • Savolainen M, et al. Better understanding of dissolution behaviour of amorphous drugs by in situ solid-state analysis using Raman spectroscopy. Eur J Pharm Biopharm 2009; 71: 71-79.
    • (2009) Eur J Pharm Biopharm , vol.71 , pp. 71-79
    • Savolainen, M.1
  • 19
    • 77953171784 scopus 로고    scopus 로고
    • Understanding the behavior of amorphous pharmaceutical systems during dissolution
    • Alonzo DE, et al. Understanding the behavior of amorphous pharmaceutical systems during dissolution. Pharm Res 2010; 27: 608-618.
    • (2010) Pharm Res , vol.27 , pp. 608-618
    • Alonzo, D.E.1
  • 20
    • 77957741630 scopus 로고    scopus 로고
    • Design and characterization of a laminar flow-through dissolution apparatus: Comparison of hydrodynamic conditions to those of common dissolution techniques
    • doi:10.3109/10837450903499341. [epub ahead of print
    • Greco K, et al. Design and characterization of a laminar flow-through dissolution apparatus: comparison of hydrodynamic conditions to those of common dissolution techniques. Pharm Dev Technol 2010; doi:10.3109/10837450903499341. [epub ahead of print.
    • (2010) Pharm Dev Technol
    • Greco, K.1
  • 21
    • 62849110155 scopus 로고    scopus 로고
    • Solvent-mediated solid phase transformations of carbamazepine: Effects of simulated intestinal fluid and fasted state simulated intestinal fluid
    • Lehto P, et al. Solvent-mediated solid phase transformations of carbamazepine: effects of simulated intestinal fluid and fasted state simulated intestinal fluid. J Pharm Sci 2009; 98: 985-996.
    • (2009) J Pharm Sci , vol.98 , pp. 985-996
    • Lehto, P.1
  • 22
    • 0037372824 scopus 로고    scopus 로고
    • Effects of excipients on hydrate formation in wet masses containing theophylline
    • Airaksinen S, et al. Effects of excipients on hydrate formation in wet masses containing theophylline. J Pharm Sci 2003; 92: 516-528.
    • (2003) J Pharm Sci , vol.92 , pp. 516-528
    • Airaksinen, S.1
  • 23
    • 33947500641 scopus 로고    scopus 로고
    • Influence of polymorphic form, morphology and excipient interactions on the dissolution of carbamazepine compacts
    • Tian F, et al. Influence of polymorphic form, morphology and excipient interactions on the dissolution of carbamazepine compacts. J Pharm Sci 2007; 96: 584-594.
    • (2007) J Pharm Sci , vol.96 , pp. 584-594
    • Tian, F.1
  • 24
    • 33846799206 scopus 로고    scopus 로고
    • The influence of various excipients on the conversion kinetics of carbamazepine polymorphs in aqueous suspension
    • Tian F, et al. The influence of various excipients on the conversion kinetics of carbamazepine polymorphs in aqueous suspension. J Pharm Pharmacol 2006; 59: 193-201.
    • (2006) J Pharm Pharmacol , vol.59 , pp. 193-201
    • Tian, F.1
  • 25
    • 32644434551 scopus 로고    scopus 로고
    • Physical stability of crystal hydrates and their anhydrates in the presence of excipients
    • Salameh AK, Taylor LS,. Physical stability of crystal hydrates and their anhydrates in the presence of excipients. J Pharm Sci 2005; 95: 446-461.
    • (2005) J Pharm Sci , vol.95 , pp. 446-461
    • Salameh, A.K.1    Taylor, L.S.2
  • 26
    • 34247523344 scopus 로고    scopus 로고
    • Additive effects on the solvent-mediated anhydrate/hydrate phase transformation in a mixed solvent
    • Qu H, et al. Additive effects on the solvent-mediated anhydrate/hydrate phase transformation in a mixed solvent. Cryst Growth Des 2007; 7: 724-729.
    • (2007) Cryst Growth des , vol.7 , pp. 724-729
    • Qu, H.1
  • 27
    • 0036805062 scopus 로고    scopus 로고
    • Ibuprofen crystals with optimized properties
    • Rasenack N, Müller BW,. Ibuprofen crystals with optimized properties. Int J Pharm 2002; 245: 9-24.
    • (2002) Int J Pharm , vol.245 , pp. 9-24
    • Rasenack, N.1    Müller, B.W.2
  • 28
    • 0026677360 scopus 로고
    • Physicochemical characterization of a phase change produced during the wet granulation of chlorpromazine hydrochloride and its effects on tableting
    • Wong MWY, Mitchell AG,. Physicochemical characterization of a phase change produced during the wet granulation of chlorpromazine hydrochloride and its effects on tableting. Int J Pharm 1992; 88: 261-273.
    • (1992) Int J Pharm , vol.88 , pp. 261-273
    • Wong, M.W.Y.1    Mitchell, A.G.2
  • 29
    • 0024343174 scopus 로고
    • Piroxicam-pseudopolymorphism and the ability to agglomerate
    • [in German]
    • Huttenrauch R, Fricke S,. Piroxicam-pseudopolymorphism and the ability to agglomerate. Pharmazie 1989; 44: 726-727. [in German]
    • (1989) Pharmazie , vol.44 , pp. 726-727
    • Huttenrauch, R.1    Fricke, S.2
  • 30
    • 1242269729 scopus 로고    scopus 로고
    • Improved tableting properties of p-hydroxybenzoic acid by water of crystallization: A molecular insight
    • Sun C, Grant DJW,. Improved tableting properties of p-hydroxybenzoic acid by water of crystallization: a molecular insight. Pharm Res 2004; 21: 382-386.
    • (2004) Pharm Res , vol.21 , pp. 382-386
    • Sun, C.1    Grant, D.J.W.2
  • 31
  • 32
    • 0016588006 scopus 로고
    • Characterization of habits and crystalline modification of solids and their pharmaceutical applications
    • Haleblian JK,. Characterization of habits and crystalline modification of solids and their pharmaceutical applications. J Pharm Sci 1975; 64: 1269-1288.
    • (1975) J Pharm Sci , vol.64 , pp. 1269-1288
    • Haleblian, J.K.1
  • 34
    • 33847016492 scopus 로고    scopus 로고
    • Organic crystal hydrates: What are the important factors for the formation
    • Infantes L, et al. Organic crystal hydrates: what are the important factors for the formation. Cryst Eng Comm 2007; 9: 65-71.
    • (2007) Cryst Eng Comm , vol.9 , pp. 65-71
    • Infantes, L.1
  • 37
    • 0030591402 scopus 로고    scopus 로고
    • Influence of water activity in organic solvent + water mixtures on the nature of the crystallizing drug phase. 1. Theophylline
    • DOI 10.1016/0378-5173(95)04466-3
    • Zhu H, et al. Influence of water activity in organic solvent + water mixtures on the nature of the crystallizing drug phase. 1. Theophylline. Int J Pharm 1996; 135: 151-160. (Pubitemid 26260884)
    • (1996) International Journal of Pharmaceutics , vol.135 , Issue.1-2 , pp. 151-160
    • Zhu, H.1    Yuen, C.2    Grant, D.J.W.3
  • 38
    • 0030576612 scopus 로고    scopus 로고
    • Influence of water activity in organic solvent + water mixtures on the nature of the crystallizing drug phase. 2. Ampicillin
    • DOI 10.1016/0378-5173(96)04570-X
    • Zhu H, Grant DJW,. Influence of water activity in organic solvent + water mixtures on the nature of the crystallizing drug phase. 2. Ampicillin. Int J Pharm 1996; 139: 33-43. (Pubitemid 26276265)
    • (1996) International Journal of Pharmaceutics , vol.139 , Issue.1-2 , pp. 33-43
    • Zhu, H.1    Grant, D.J.W.2
  • 39
    • 33747368526 scopus 로고    scopus 로고
    • Solubility and stability of anhydrate/hydrate in solvent mixtures
    • Qu H, et al. Solubility and stability of anhydrate/hydrate in solvent mixtures. Int J Pharm 2006; 321: 101-107.
    • (2006) Int J Pharm , vol.321 , pp. 101-107
    • Qu, H.1
  • 40
    • 33749013855 scopus 로고    scopus 로고
    • Solvent-mediated phase transformation kinetics of an anhydrate/hydrate system
    • Qu H, et al. Solvent-mediated phase transformation kinetics of an anhydrate/hydrate system. Cryst Growth Des 2006; 6: 2053-2060.
    • (2006) Cryst Growth des , vol.6 , pp. 2053-2060
    • Qu, H.1
  • 41
    • 59049104133 scopus 로고    scopus 로고
    • Determination of hydrate transition temperature using transformation kinetics obtained by Raman spectroscopy
    • Wikström H, et al. Determination of hydrate transition temperature using transformation kinetics obtained by Raman spectroscopy. J Pharm Biomed Anal 2009; 49: 247-252.
    • (2009) J Pharm Biomed Anal , vol.49 , pp. 247-252
    • Wikström, H.1
  • 42
    • 34547774582 scopus 로고    scopus 로고
    • The nucleation of inosine: The impact of solution chemistry on the appearance of polymorphic and hydrated crystal forms
    • Chiarella RA, et al. The nucleation of inosine: the impact of solution chemistry on the appearance of polymorphic and hydrated crystal forms. Faraday Discuss 2007; 136: 179-193.
    • (2007) Faraday Discuss , vol.136 , pp. 179-193
    • Chiarella, R.A.1
  • 43
    • 65249165473 scopus 로고    scopus 로고
    • Mechanistic insight into the evaporative crystallization of two polymorphs of nitrofurantoin monohydrate
    • Tian F, et al. Mechanistic insight into the evaporative crystallization of two polymorphs of nitrofurantoin monohydrate. J Cryst Growth 2009; 311: 2580-2589.
    • (2009) J Cryst Growth , vol.311 , pp. 2580-2589
    • Tian, F.1
  • 44
    • 33748256291 scopus 로고    scopus 로고
    • Solubilities of and transformations between the anhydrous and hydrated forms of L-serine in water-methanol solutions
    • Luk C-WJ, Rousseau RW,. Solubilities of and transformations between the anhydrous and hydrated forms of L-serine in water-methanol solutions. Cryst Growth Des 2006; 6: 1808-1812.
    • (2006) Cryst Growth des , vol.6 , pp. 1808-1812
    • Luk, C.-W.1    Rousseau, R.W.2
  • 45
    • 0001732841 scopus 로고
    • Studies on formation and transformation of solid materials
    • Ostwald WZ,. Studies on formation and transformation of solid materials. Z Phys Chem 1897; 22: 289-330.
    • (1897) Z Phys Chem , vol.22 , pp. 289-330
    • Ostwald, W.Z.1
  • 46
    • 53349107543 scopus 로고    scopus 로고
    • Spectroscopic monitoring of carbamazepine crystallization and phase transformation in ethanol-water solution
    • Qu H, et al. Spectroscopic monitoring of carbamazepine crystallization and phase transformation in ethanol-water solution. Ind Eng Chem Res 2008; 47: 6991-6998.
    • (2008) Ind Eng Chem Res , vol.47 , pp. 6991-6998
    • Qu, H.1
  • 47
    • 34547735131 scopus 로고    scopus 로고
    • Crystallization of monohydrate citric acid. 1. in situ monitoring through the joint use of Raman spectroscopy and image analysis
    • Caillet A, et al. Crystallization of monohydrate citric acid. 1. In situ monitoring through the joint use of Raman spectroscopy and image analysis. Cryst Growth Des 2007; 7: 2080-2087.
    • (2007) Cryst Growth des , vol.7 , pp. 2080-2087
    • Caillet, A.1
  • 48
    • 53949112047 scopus 로고    scopus 로고
    • Kinetic study on hemipenta hydrate risedronate monosodium in batch crystallization by cooling mode
    • Nguyen TNP, Kim K-J,. Kinetic study on hemipenta hydrate risedronate monosodium in batch crystallization by cooling mode. Int J Pharm 2008; 364: 1-8.
    • (2008) Int J Pharm , vol.364 , pp. 1-8
    • Nguyen, T.N.P.1    Kim, K.-J.2
  • 49
    • 0037453790 scopus 로고    scopus 로고
    • Pseudopolymorphic crystallization of L-ornithine-L-aspartate by drawing out
    • Kim Y, et al. Pseudopolymorphic crystallization of L-ornithine-L- aspartate by drawing out. Ind Eng Chem Res 2003; 42: 883-889.
    • (2003) Ind Eng Chem Res , vol.42 , pp. 883-889
    • Kim, Y.1
  • 50
    • 33744832601 scopus 로고    scopus 로고
    • Effect of temperature on antisolvent crystallization and transformation behaviors of thiazole-derivative polymorphs
    • Kitamura M, Hironaka S,. Effect of temperature on antisolvent crystallization and transformation behaviors of thiazole-derivative polymorphs. Cryst Growth Des 2006; 6: 1214-1218.
    • (2006) Cryst Growth des , vol.6 , pp. 1214-1218
    • Kitamura, M.1    Hironaka, S.2
  • 51
    • 0036494081 scopus 로고    scopus 로고
    • Effects of solvent composition and temperature on polymorphism and crystallization behavior of thiazole-derivative
    • DOI 10.1016/S0022-0248(02)00828-X, PII S002202480200828X
    • Kitamura M, Nakamura K,. Effect of solvent composition and temperature on polymorphism and crystallization behavior of thiazole-derivative. J Cryst Growth 2002; 236: 676-686. (Pubitemid 34405250)
    • (2002) Journal of Crystal Growth , vol.236 , Issue.4 , pp. 676-686
    • Kitamura, M.1    Nakamura, K.2
  • 52
    • 0345014900 scopus 로고    scopus 로고
    • Monitoring of antisolvent addition crystallization with Raman spectroscopy
    • Falcon JA, Berglund KA,. Monitoring of antisolvent addition crystallization with Raman spectroscopy. Cryst Growth Des 2003; 3: 947-952.
    • (2003) Cryst Growth des , vol.3 , pp. 947-952
    • Falcon, J.A.1    Berglund, K.A.2
  • 53
    • 0042431697 scopus 로고    scopus 로고
    • Anti-solvent crystallization and transformation of thiazole-derivative polymorphs - I: Effects of addition rate and initial concentrations
    • Kitamura M, Sugimoto M,. Anti-solvent crystallization and transformation of thiazole-derivative polymorphs-I: effects of addition rate and initial concentrations. J Cryst Growth 2003; 257: 177-184.
    • (2003) J Cryst Growth , vol.257 , pp. 177-184
    • Kitamura, M.1    Sugimoto, M.2
  • 54
    • 0001266165 scopus 로고
    • The kinetics of solvent-mediated phase transformations
    • A
    • Cardew PT, Davey RJ,. The kinetics of solvent-mediated phase transformations. Proc R Soc Lond 1985; A 398: 415-428.
    • (1985) Proc R Soc Lond , vol.398 , pp. 415-428
    • Cardew, P.T.1    Davey, R.J.2
  • 55
    • 0000532131 scopus 로고
    • Rate controlling processes in solvent-mediated phase transformations
    • Davey RJ, Cardew PT,. Rate controlling processes in solvent-mediated phase transformations. J Cryst Growth 1986; 79: 648-653.
    • (1986) J Cryst Growth , vol.79 , pp. 648-653
    • Davey, R.J.1    Cardew, P.T.2
  • 56
    • 0025681708 scopus 로고
    • Effect of benzalkonium chloride on crystal growth and aqueous solubility of carbamazepine
    • Luhtala S, et al. Effect of benzalkonium chloride on crystal growth and aqueous solubility of carbamazepine. Acta Pharm Fennica 1990; 99: 9-68.
    • (1990) Acta Pharm Fennica , vol.99 , pp. 9-68
    • Luhtala, S.1
  • 57
    • 0027096942 scopus 로고
    • Effect of poloxamer 184 on crystal growth and aqueous solubility of carbamazepine
    • Luhtala S,. Effect of poloxamer 184 on crystal growth and aqueous solubility of carbamazepine. Acta Pharm Nord 1992; 4: 172-176.
    • (1992) Acta Pharm Nord , vol.4 , pp. 172-176
    • Luhtala, S.1
  • 58
    • 0842332474 scopus 로고    scopus 로고
    • Surfactant-facilitated crystallization of dihydrate carbamazepine during dissolution of anhydrous polymorph
    • Rodríguez-Hornedo N, Murphy D,. Surfactant-facilitated crystallization of dihydrate carbamazepine during dissolution of anhydrous polymorph. J Pharm Sci 2004; 93: 449-460.
    • (2004) J Pharm Sci , vol.93 , pp. 449-460
    • Rodríguez-Hornedo, N.1    Murphy, D.2
  • 59
    • 0026770590 scopus 로고
    • Effect of sodium lauryl sulphate and polysorbate 80 on crystal growth and aqueous solubility of carbamazepine
    • Luhtala S,. Effect of sodium lauryl sulphate and polysorbate 80 on crystal growth and aqueous solubility of carbamazepine. Acta Pharma Nord 1992; 4: 85-90.
    • (1992) Acta Pharma Nord , vol.4 , pp. 85-90
    • Luhtala, S.1
  • 60
    • 0033992376 scopus 로고    scopus 로고
    • Effect of binders on polymorphic transformation kinetics of carbamazepine in aqueous solution
    • Otsuka M, et al. Effect of binders on polymorphic transformation kinetics of carbamazepine in aqueous solution. Colloids Surf B 2000; 17: 145-152.
    • (2000) Colloids Surf B , vol.17 , pp. 145-152
    • Otsuka, M.1
  • 61
    • 0037413403 scopus 로고    scopus 로고
    • A compaction process to enhance dissolution of poorly water-soluble drugs using hydroxypropyl methylcellulose
    • Mitchell SA, et al. A compaction process to enhance dissolution of poorly water-soluble drugs using hydroxypropyl methylcellulose. Int J Pharm 2003; 250: 3-11.
    • (2003) Int J Pharm , vol.250 , pp. 3-11
    • Mitchell, S.A.1
  • 62
    • 35548973805 scopus 로고    scopus 로고
    • Crystallization of monohydrate citric acid. 2. Modeling through population balance equations
    • Caillet A, et al. Crystallization of monohydrate citric acid. 2. Modeling through population balance equations. Cryst Growth Des 2007; 7: 2088-2095.
    • (2007) Cryst Growth des , vol.7 , pp. 2088-2095
    • Caillet, A.1
  • 63
    • 35248813407 scopus 로고    scopus 로고
    • A population balance model of the solution-mediated phase transition of citric acid
    • Fevotte G, et al. A population balance model of the solution-mediated phase transition of citric acid. AIChE J 2007; 53: 2578-2589.
    • (2007) AIChE J , vol.53 , pp. 2578-2589
    • Fevotte, G.1
  • 64
    • 8844229530 scopus 로고    scopus 로고
    • Process modeling of the polymorphic transformation of L-glutamic acid
    • Ono T, et al. Process modeling of the polymorphic transformation of L-glutamic acid. Cryst Growth Des 2004; 6: 1161-1167.
    • (2004) Cryst Growth des , vol.6 , pp. 1161-1167
    • Ono, T.1
  • 65
    • 33646365349 scopus 로고    scopus 로고
    • In situ monitoring and modeling of the solvent-mediated polymorphic transformation of L-glutamic acid
    • Schöll J, et al. In situ monitoring and modeling of the solvent-mediated polymorphic transformation of L-glutamic acid. Cryst Growth Des 2006; 6: 881-891.
    • (2006) Cryst Growth des , vol.6 , pp. 881-891
    • Schöll, J.1
  • 66
    • 0015130813 scopus 로고
    • Isolation and characterization of some solid phases of fluprednisolone
    • Haleblian JK, et al. Isolation and characterization of some solid phases of fluprednisolone. J Pharm Sci 1971; 60: 1485-1488.
    • (1971) J Pharm Sci , vol.60 , pp. 1485-1488
    • Haleblian, J.K.1
  • 67
    • 77951689740 scopus 로고
    • Dissolution behavior of crystalline solvated and nonsolvated forms of some pharmaceuticals
    • Shefter E, Higuchi T,. Dissolution behavior of crystalline solvated and nonsolvated forms of some pharmaceuticals. J Pharm Sci 1963; 52: 781-791.
    • (1963) J Pharm Sci , vol.52 , pp. 781-791
    • Shefter, E.1    Higuchi, T.2
  • 69
    • 0141822419 scopus 로고
    • Polymorphs of nitrofurantoin. I. Preparation and x-ray crystal structures of two monohydrated forms of nitrofurantoin
    • Pienaar EW, et al. Polymorphs of nitrofurantoin. I. Preparation and x-ray crystal structures of two monohydrated forms of nitrofurantoin. J Crystall Spectr Res 1993; 23: 739-744.
    • (1993) J Crystall Spectr Res , vol.23 , pp. 739-744
    • Pienaar, E.W.1
  • 70
    • 0037945704 scopus 로고    scopus 로고
    • Crystal forms of LY334370 HCl: Isolation, solid-state characterization, and physicochemical properties
    • Reutzel-Edens SM, et al. Crystal forms of LY334370 HCl: isolation, solid-state characterization, and physicochemical properties. J Pharm Sci 2003; 92: 1196-1205.
    • (2003) J Pharm Sci , vol.92 , pp. 1196-1205
    • Reutzel-Edens, S.M.1
  • 71
    • 0347360187 scopus 로고    scopus 로고
    • Preparation and physicochemical properties of niclosamide anhydrate and two monohydrates
    • Van Tonder EC, et al. Preparation and physicochemical properties of niclosamide anhydrate and two monohydrates. Int J Pharm 2004; 269: 417-432.
    • (2004) Int J Pharm , vol.269 , pp. 417-432
    • Van Tonder, E.C.1
  • 72
    • 0008209306 scopus 로고    scopus 로고
    • Polymorphism and pseudopolymorphism of the antibacterial nitrofurantoin
    • Caira MR, et al. Polymorphism and pseudopolymorphism of the antibacterial nitrofurantoin. Mol Cryst Liq Cryst Sci Technol Mol Cryst Liq Cryst 1996; 279: 241-264.
    • (1996) Mol Cryst Liq Cryst Sci Technol Mol Cryst Liq Cryst , vol.279 , pp. 241-264
    • Caira, M.R.1
  • 73
    • 0027289727 scopus 로고
    • Effect of environmental humidity on the transformation pathway of nitrofurantoin modifications during grinding and the physicochemical properties of ground products
    • Otsuka M, Matsuda Y,. Effect of environmental humidity on the transformation pathway of nitrofurantoin modifications during grinding and the physicochemical properties of ground products. J Pharm Pharmacol 1993; 45: 406-413.
    • (1993) J Pharm Pharmacol , vol.45 , pp. 406-413
    • Otsuka, M.1    Matsuda, Y.2
  • 75
    • 34249980663 scopus 로고    scopus 로고
    • Hyphenated spectroscopy as a polymorph screening tool
    • Aaltonen J, et al. Hyphenated spectroscopy as a polymorph screening tool. J Pharm Biomed Anal 2007; 44: 477-483.
    • (2007) J Pharm Biomed Anal , vol.44 , pp. 477-483
    • Aaltonen, J.1
  • 76
    • 0026501543 scopus 로고
    • Rotating-disk dissolution kinetics of nitrofurantoin anhydrate and monohydrate at various temperatures
    • Otsuka M, et al. Rotating-disk dissolution kinetics of nitrofurantoin anhydrate and monohydrate at various temperatures. Pharm Res 1992; 9: 307-311.
    • (1992) Pharm Res , vol.9 , pp. 307-311
    • Otsuka, M.1
  • 77
    • 0025118436 scopus 로고
    • Characterization of nitrofurantoin anhydrate and monohydrate, and their dissolution behaviors
    • Otsuka M, et al. Characterization of nitrofurantoin anhydrate and monohydrate, and their dissolution behaviors. Chem Pharm Bull 1990; 38: 2667-2670.
    • (1990) Chem Pharm Bull , vol.38 , pp. 2667-2670
    • Otsuka, M.1
  • 78
    • 61549111851 scopus 로고    scopus 로고
    • Towards an understanding of the factors influencing anhydrate-to-hydrate transformation kinetics in aqueous environments
    • Wikström H, et al. Towards an understanding of the factors influencing anhydrate-to-hydrate transformation kinetics in aqueous environments. Cryst Growth Des 2008; 8: 2684-2693.
    • (2008) Cryst Growth des , vol.8 , pp. 2684-2693
    • Wikström, H.1
  • 79
    • 74049124218 scopus 로고    scopus 로고
    • Crystallization of a polymorphic hydrate system
    • Tian F, et al. Crystallization of a polymorphic hydrate system. J Pharm Sci 2010; 99: 753-763.
    • (2010) J Pharm Sci , vol.99 , pp. 753-763
    • Tian, F.1
  • 80
    • 77951671779 scopus 로고    scopus 로고
    • Insight into crystallization mechanisms of polymorphic hydrate systems
    • Tian F, et al. Insight into crystallization mechanisms of polymorphic hydrate systems. Chem Eng Technol 2010 33: 833-838.
    • (2010) Chem Eng Technol , vol.33 , pp. 833-838
    • Tian, F.1
  • 81
    • 27944487022 scopus 로고    scopus 로고
    • Occurrence of pharmaceutically acceptable anions and cations in the Cambridge Structural Database
    • Haynes DA, et al. Occurrence of pharmaceutically acceptable anions and cations in the Cambridge Structural Database. J Pharm Sci 2005; 94: 2111-2120.
    • (2005) J Pharm Sci , vol.94 , pp. 2111-2120
    • Haynes, D.A.1
  • 82
    • 0023032232 scopus 로고
    • Salt selection for basic drugs
    • Gould PL,. Salt selection for basic drugs. Int J Pharm 1986; 33: 201-217.
    • (1986) Int J Pharm , vol.33 , pp. 201-217
    • Gould, P.L.1
  • 83
    • 0017623487 scopus 로고
    • Pharmaceutical salts
    • Berge SM, et al. Pharmaceutical salts. J Pharm Sci 1977; 66: 1-19.
    • (1977) J Pharm Sci , vol.66 , pp. 1-19
    • Berge, S.M.1
  • 84
    • 34548032742 scopus 로고    scopus 로고
    • Salt formation to improve drug solubility
    • Serajuddin ATM,. Salt formation to improve drug solubility. Adv Drug Deliv Rev 2007; 59: 603-616.
    • (2007) Adv Drug Deliv Rev , vol.59 , pp. 603-616
    • Serajuddin, A.T.M.1
  • 86
    • 0026457855 scopus 로고
    • Physicochemical properties of salts of P-aminosalicylic acid. I. Correlation of crystal structure and hydrate stability
    • Forbes RT, et al. Physicochemical properties of salts of P-aminosalicylic acid. I. Correlation of crystal structure and hydrate stability. Pharm Res 1992; 9: 1428-1435.
    • (1992) Pharm Res , vol.9 , pp. 1428-1435
    • Forbes, R.T.1
  • 87
    • 0029798062 scopus 로고    scopus 로고
    • Physicochemical characterization of nedocromil bivalent metal salt hydrates. 1. Nedocromil magnesium
    • Zhu H, et al. Physicochemical characterization of nedocromil bivalent metal salt hydrates. 1. Nedocromil magnesium. J Pharm Sci 1996; 85: 1026-1034.
    • (1996) J Pharm Sci , vol.85 , pp. 1026-1034
    • Zhu, H.1
  • 88
    • 0030975430 scopus 로고    scopus 로고
    • Physicochemical characterization of nedocromil bivalent metal salt hydrates. 2. Nedocromil zinc
    • Zhu H, et al. Physicochemical characterization of nedocromil bivalent metal salt hydrates. 2. Nedocromil zinc. J Pharm Sci 1997; 86: 418-428.
    • (1997) J Pharm Sci , vol.86 , pp. 418-428
    • Zhu, H.1
  • 89
    • 61549104954 scopus 로고    scopus 로고
    • Structural investigations of hydrate, anhydrate, free base and hydrochloride forms of morphine and naloxone
    • Guguta C, et al. Structural investigations of hydrate, anhydrate, free base and hydrochloride forms of morphine and naloxone. Cryst Growth Des 2008; 8: 4150-4158.
    • (2008) Cryst Growth des , vol.8 , pp. 4150-4158
    • Guguta, C.1
  • 90
    • 0028016246 scopus 로고
    • Crystallinity, hygroscopicity and dissolution of moricizine hydrochloride hemihydrate
    • Wu LS, et al. Crystallinity, hygroscopicity and dissolution of moricizine hydrochloride hemihydrate. J Pharm Biomed Anal 1994; 12: 1043-1046.
    • (1994) J Pharm Biomed Anal , vol.12 , pp. 1043-1046
    • Wu, L.S.1
  • 91
    • 0037945704 scopus 로고    scopus 로고
    • Crystal forms of LY334370 HCl: Isolation, solid-state characterization, and physicochemical properties
    • Reutzel SM, et al. Crystal forms of LY334370 HCl: isolation, solid-state characterization, and physicochemical properties. J Pharm Sci 2003; 92: 1196-1205.
    • (2003) J Pharm Sci , vol.92 , pp. 1196-1205
    • Reutzel, S.M.1
  • 92
    • 32644490018 scopus 로고    scopus 로고
    • Physico-chemical characterisation and intrinsic dissolution studies of a new hydrate form of diclofenac sodium: Comparison with anhydrous form
    • Bartolomei M, et al. Physico-chemical characterisation and intrinsic dissolution studies of a new hydrate form of diclofenac sodium: comparison with anhydrous form. J Pharm Biomed Anal 2006; 40: 1105-1113.
    • (2006) J Pharm Biomed Anal , vol.40 , pp. 1105-1113
    • Bartolomei, M.1
  • 93
    • 0036746781 scopus 로고    scopus 로고
    • Hydrate formation during wet granulation studied by spectroscopic methods and multivariate analysis
    • Jørgensen AC, et al. Hydrate formation during wet granulation studied by spectroscopic methods and multivariate analysis. Pharm Res 2002; 19: 1285-1291.
    • (2002) Pharm Res , vol.19 , pp. 1285-1291
    • Jørgensen, A.C.1
  • 94
    • 0035897679 scopus 로고    scopus 로고
    • Theoretical approaches to physical transformations of active pharmaceutical ingredients during manufacturing processes
    • Morris KR, et al. Theoretical approaches to physical transformations of active pharmaceutical ingredients during manufacturing processes. Adv Drug Deliv Rev 2001; 48: 91-114.
    • (2001) Adv Drug Deliv Rev , vol.48 , pp. 91-114
    • Morris, K.R.1
  • 95
    • 1842789824 scopus 로고    scopus 로고
    • Evaluation of drug physical form during granulation, tabletting and storage
    • Williams AC, et al. Evaluation of drug physical form during granulation, tabletting and storage. Int J Pharm 2004; 275: 29-39.
    • (2004) Int J Pharm , vol.275 , pp. 29-39
    • Williams, A.C.1
  • 96
    • 35348859452 scopus 로고    scopus 로고
    • Hydrate modifications of the non-steroidal anti-inflammatory drug diclofenac sodium: Solid-state characterisation of a trihydrate form
    • Bartolomei M, et al. Hydrate modifications of the non-steroidal anti-inflammatory drug diclofenac sodium: solid-state characterisation of a trihydrate form. J Pharm Biomed Anal 2007; 45: 443-449.
    • (2007) J Pharm Biomed Anal , vol.45 , pp. 443-449
    • Bartolomei, M.1
  • 97
    • 15744390959 scopus 로고    scopus 로고
    • Diclofenac sodium multisource prolonged release tablets - A comparative study on the dissolution profiles
    • Bertocchi P, et al. Diclofenac sodium multisource prolonged release tablets-a comparative study on the dissolution profiles. J Pharm Biomed Anal 2005; 37: 679-685.
    • (2005) J Pharm Biomed Anal , vol.37 , pp. 679-685
    • Bertocchi, P.1
  • 98
    • 61449120999 scopus 로고    scopus 로고
    • Influence of the solid form of siramesine hydrochloride on its behaviour in aqueous environments
    • Zimmermann A, et al. Influence of the solid form of siramesine hydrochloride on its behaviour in aqueous environments. Pharm Res 2009; 26: 846-854.
    • (2009) Pharm Res , vol.26 , pp. 846-854
    • Zimmermann, A.1


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