Synthesis and pharmacological activity of 9-R-2-halogenophenylimidazo[1,2- a]benzimidazoles

Pharmaceutical Chemistry Journal

Volumn 44, Issue 7, 2010, Pages 345-351

  Anisimova, V A ^a   Spasov, A A ^b,c   Tolpygin, I E ^a   Minkin, V I ^a   Chernikov, M V ^b,c   Yakovlev, D S ^b,c   Stukovina, A Yu ^b,c   Goryagin, I I ^b,c   Grechko, O Yu ^b   Kirillova, N V ^b   Kosolapov, V A ^b   Tibir'Kova, E V ^b   Salaznikova, O A ^b   Naumenko, L V ^a   Gurova, N A ^b  

^a SOUTHERN FEDERAL UNIVERSITY   (Russian Federation)

^b VOLGOGRAD STATE MEDICAL UNIVERSITY   (Russian Federation)

^c INSTITUTE OF BIOMEDICAL CHEMISTRY   (Russian Federation)

Author keywords

2 a benzimidazole; 5 HT2 antagonist activity; 5 HT3 antagonist activity; Antiarrhythmic activity; Antioxidant activity; Antiplatelet activity; Hemorheological activity; Imidazo 1; P2Y1 antagonist activity

Indexed keywords

2,9 HALOGENOPHENYLIMIDAZO[1,2 ALPHA]BENZIMIDAZOLE; BENZIMIDAZOLE DERIVATIVE; HISTAMINE H1 RECEPTOR ANTAGONIST; KAPPA OPIATE RECEPTOR AGONIST; PURINERGIC P2Y1 RECEPTOR; RADICAL; SEROTONIN 2 ANTAGONIST; SEROTONIN 3 ANTAGONIST; UNCLASSIFIED DRUG;

ANTIARRHYTHMIC ACTIVITY; ANTIOXIDANT ACTIVITY; ARTICLE; BLOOD RHEOLOGY; NONHUMAN; RAT;

EID: 78649471894     PISSN: 0091150X     EISSN: 15739031     Source Type: Journal    
DOI: 10.1007/s11094-010-0465-y     Document Type: Article

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