Design, synthesis and acaricidal activity of novel strobilurin derivatives containing pyrimidine moieties

Pest Management Science

Volumn 66, Issue 11, 2010, Pages 1208-1214

  Chai, Bao Shan ^a,b   Liu, Chang Ling ^a   Li, Hui Chao ^a   He, Xiao Min ^a   Luo, Yan Mei ^a   Huang, Guang ^a   Zhang, Hong ^a   Chang, Jun Biao ^b  

^a SHENYANG RESEARCH INSTITUTE OF CHEMICAL INDUSTRY   (China)

^b ZHENGZHOU UNIVERSITY   (China)

Author keywords

Acaricidal activity; Intermediate derivatisation method; Pyrimidine; Strobilurin derivatives

Indexed keywords

ACARICIDE; LEAD; METHACRYLIC ACID DERIVATIVE; PYRIMIDINE; PYRIMIDINE DERIVATIVE;

ACARICIDE; BIOASSAY; CHEMICAL CONTROL; MASS SPECTROMETRY; NUCLEAR MAGNETIC RESONANCE; STROBILURIN; X-RAY DIFFRACTION;

ANIMAL; ARTICLE; CHEMISTRY; MASS SPECTROMETRY; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PEST CONTROL; SYNTHESIS; TETRANYCHIDAE;

ACARICIDES; ANIMALS; LEAD; MAGNETIC RESONANCE SPECTROSCOPY; MASS SPECTROMETRY; METHACRYLATES; PEST CONTROL; PYRIMIDINES; TETRANYCHIDAE;

TETRANYCHUS CINNABARINUS;

EID: 77958487970     PISSN: 1526498X     EISSN: 15264998     Source Type: Journal    
DOI: 10.1002/ps.1997     Document Type: Article

References (22)

1. Londershausen M, Review: Approaches to new parasiticides. Pest Manag Sci 48: 269-292 (1996).
2. Corran AJ, Renwick A and Dunbar SJ, Approaches to in vitro lead generation for fungicide invention. Pest Manag Sci 54: 338-344 (1998).
3. Jeschke P, Lieb F, Velten R and Wiese WB, Natural products and their role in the design of active ingredients for modern crop protection. ACS Symposium Series (Natural Products for Pest Management), pp. 128-141 (2006).
4. Lindell SD, Pattenden LC and Shannon J, Combinatorial chemistry in the agrosciences. Bioorg Med Chem 17: 4035-4046 (2009).
5. Bordás B, Komíves T and Lopata A, Ligand-based computer-aided pesticide design. A review of applications of the CoMFA and CoMSIA methodologies. Pest Manag Sci 59: 393-400 (2003).
6. Holmwood G and Schindler M, Protein structure based rational design of ecdysone agonists. Bioorg Med Chem 17: 4064-4070 (2009).
7. Liu CL, New agrochemical candidates from intermediate derivatization method based on bioisosteric replacement, Frontiers of Modern Chemical Engineering, Metallurgy and Material Technologies-7th Academic Conference of Chemical, Metallurgy and Material Engineering Department, CAE, ed. by Wang JK. Chemical Industry Press Publishers, Beijing, China, pp. 86-94 (2009).
8. Liu CL, Innovation of pesticide discovery methods and candidate compounds (in Chinese). High-Technology and Industrialization 9: 79-81 (2008).
9. Liu CL, Li M, Guan AY, Zhang H, Li ZN and Ye TX, Preparation of coumarin derivatives for preventing diseases and pests in crop plants. CN Patent 1869032 (2006).
10. Liu CL, Li M, Zhang H, Li L, Zhang MX, Guan AY, et al, Preparation of azoles as agrochemical insecticides and germicides. World Patent WO 2005080344 (2005).
11. Liu CL, Li M, Li ZN, Geng LW, Zhang H, Zhou DF, et al, Preparation of arylethers as fungicides and pesticides. World Patent WO 2006125370 (2005).
12. Liu CL, Li M, Guan AY, Zhang H and Li ZM, Design, synthesis and fungicidal activity of novel (E)-methyl 2-{2-[(coumarin-7-yloxy)methyl]phenyl}-3-methoxyacrylates. Nat Prod Commun 2: 845-848 (2007).
13. Li M, Liu CL, Li L, Yang H, Li ZN, Zhang H, et al, Design, synthesis and biological activities of new strobilurin derivatives containing substituted pyrazoles. Pest Manag Sci 66: 107-112 (2010).
14. Li HC, Liu CL, Chai BS, Li M, Li ZN and Yang JC, Design, synthesis and fungicidal activity of novel strobilurin analogues containing substituted N-phenylpyrimidin-2-amines. Nat Prod Commun 4: 1209-1214 (2009).
15. Li M, Liu CL, Yang JC, Li L, Li ZN, Zhang H, et al, Design, synthesis and biological activity of new strobilurin derivatives with a 1H-pyrazol-5-oxy side chain. Nat Prod Commun 4: 1215-1220 (2009).
16. Li HC, Chai BS, Li ZN, Yang JC and Liu CL, Synthesis and fungicidal activity of novel strobilurin analogues containing substituted N-phenylpyrimidin-2-amines. Chin Chem Lett 20: 1287-1290 (2009).
17. Li M, Liu CL, Yang JC, Zhang JB, Li ZN, Zhang H, et al, Synthesis and biological activity of new (E)-α-(methoxyimino)benzeneacetate derivatives containing a substituted pyrazole ring. J Ag Food Chem 58: 2664-2667 (2010).
18. Tomlin CDS (ed.), Fluacrypyrim, The Pesticide Manual, 14th edition. British Crop Protection Council, Alton, Hants, UK, pp. 471-472 (2006).
19. Marini AM, Settimo FD, Salerno S, Motta CL, Simorini F, Taliani S, et al, Synthesis and in vitro antiproliferative activity of new substituted benzo[3', 2':5, 6]thiopyrano[4, 3-d]pyrimidines. J Heterocycl Chem 45: 745-749 (2008).
20. Liu CL, Chai BS, Zhang H, Li HC, Wang JF, Peng YW, et al, Substituted pyrimidine ether compounds and their use. World Patent WO 2008145052 (2008).
21. SMART, SAINT, SHELXTL and SADABS. Bruker AXS Inc., Madison, WI (1998).
22. Sheldrick GM, SHELXS-97 and SHELXL-97. University of Göttingen, Göttingen, Germany (1997).