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Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 19, 2010, Pages 5895-5899

Novel amides and esters prodrugs of olmesartan: Synthesis, bioconversion, and pharmacokinetic evaluation

(14) Park, Jin Hun a,e,f Chang, Jeong Soo c El Gamal, Mohammed I a,b Choi, Won Kyoung a Lee, Woong San a Chung, Hye Jin a Kim, Hyun Il d Cho, Young Jin d Lee, Bong Sang d Jeon, Hong Ryeol d Lee, Yong Sup e,f Choi, Young Wook c Lee, Jaehwi c Oh, Chang Hyun a,b

a Korea Institute of Science and Technology (South Korea)

b University of Science and Technology (UST) (South Korea)

c Chung Ang University (South Korea)

d CTC Bio Inc (South Korea)

e Kyung Hee University (South Korea)

f Kyung Hee University (South Korea)

Author keywords

Amide; Antihypertensive; Ester; Olmesartan; Olmesartan medoxomil; Pharmacokinetics; Prodrug

Indexed keywords

AMIDE; ANTIHYPERTENSIVE AGENT; ESTER DERIVATIVE; OLMESARTAN;

ANIMAL EXPERIMENT; ANTIHYPERTENSIVE ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG METABOLISM; DRUG SCREENING; DRUG STABILITY; DRUG SYNTHESIS; IN VITRO STUDY; MALE; NONHUMAN; PHARMACOLOGICAL PARAMETERS; RAT;

ADMINISTRATION, ORAL; AMIDES; ANIMALS; ESTERS; IMIDAZOLES; MALE; PRODRUGS; RATS; RATS, SPRAGUE-DAWLEY; TETRAZOLES;

RATTUS;

EID: 77957561249 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.07.089 Document Type: Article

Times cited : (19)

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