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Clotet, B.1
Katlama, C.2
Lazzarin, A.3
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47
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77957328176
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Etravirine (ETR; TMC125) has no effect on fetal development in rats and rabbits
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Abstract TUPE0013
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Raoof A, Lachau-Durand S, Verbeeck J, et al. Etravirine (ETR; TMC125) has no effect on fetal development in rats and rabbits. 17th International AIDS Conference. 3-8 August 2008, Mexico City, Mexico. Abstract TUPE0013.
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17th International AIDS Conference. 3-8 August 2008, Mexico City, Mexico
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Raoof, A.1
Lachau-Durand, S.2
Verbeeck, J.3
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48
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59849126824
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Successful use of darunavir, etravirine, enfuvirtide and tenofovir/emtricitabine in pregnant woman with multiclass HIV resistance
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Furco A, Gosrani B, Nicholas S, et al. Successful use of darunavir, etravirine, enfuvirtide and tenofovir/emtricitabine in pregnant woman with multiclass HIV resistance. AIDS 2009; 23:434-435.
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AIDS
, vol.23
, pp. 434-435
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Furco, A.1
Gosrani, B.2
Nicholas, S.3
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49
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77957334287
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Safety and pharmacokinetics of etravirine in pregnant HIV-infected women
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Abstract PE4.1/6
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Izurieta P, Kakuda TN, Clark A, Feys C, Witek J. Safety and pharmacokinetics of etravirine in pregnant HIV-infected women. 12th European AIDS Conference, 11-14 November 2009, Cologne, Germany. Abstract PE4.1/6.
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12th European AIDS Conference, 11-14 November 2009, Cologne, Germany
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Izurieta, P.1
Kakuda, T.N.2
Clark, A.3
Feys, C.4
Witek, J.5
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50
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77649254869
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Resistance profile of etravirine: Combined analysis of baseline genotypic and phenotypic data from the DUET studies
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Vingerhoets J, Tambuyzer L, Azijn H, et al. Resistance profile of etravirine: combined analysis of baseline genotypic and phenotypic data from the DUET studies. AIDS 2010; 24:503-514.
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(2010)
AIDS
, vol.24
, pp. 503-514
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Vingerhoets, J.1
Tambuyzer, L.2
Azijn, H.3
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51
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58149505548
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HIV-1 genotype algorithms for prediction of etravirine susceptibility: Novel mutations and weighting factors identified through correlations to phenotype
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Benhamida J, Chappey C, Coakley E, Parkin N. HIV-1 genotype algorithms for prediction of etravirine susceptibility: novel mutations and weighting factors identified through correlations to phenotype. Antivir Ther 2008; 13 Suppl 3:A142.
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(2008)
Antivir Ther
, vol.13
, Issue.SUPPL. 3
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Benhamida, J.1
Chappey, C.2
Coakley, E.3
Parkin, N.4
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52
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62849127651
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Prediction of the virological response to etravirine in clinical practice: Comparison of three genotype algorithms
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Cotte L, Trabaud MA, Tardy JC, et al. Prediction of the virological response to etravirine in clinical practice: comparison of three genotype algorithms. J Med Virol 2009; 81:672-677.
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(2009)
J Med Virol
, vol.81
, pp. 672-677
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Cotte, L.1
Trabaud, M.A.2
Tardy, J.C.3
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53
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54749118543
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Effects of different meal compositions and fasted state on the oral bioavailability of etravirine
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Schöller-Gyüre M, Boffito M, Pozniak AL, et al. Effects of different meal compositions and fasted state on the oral bioavailability of etravirine. Pharmacotherapy 2008; 28:1215-1222.
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(2008)
Pharmacotherapy
, vol.28
, pp. 1215-1222
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Schöller-Gyüre, M.1
Boffito, M.2
Pozniak, A.L.3
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55
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77957333438
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Pharmacokinetics of TMC125 in once-daily and twice-daily regimens in HIV-1-negative volunteers
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Abstract A-1427
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Schöller-Gyüre M, Kakuda TN, De Smedt G, et al. Pharmacokinetics of TMC125 in once-daily and twice-daily regimens in HIV-1-negative volunteers. 47th Interscience Conference on Antimicrobial Agents and Chemotherapy. 17-20 September 2007, Chicago, IL, USA. Abstract A-1427.
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47th Interscience Conference on Antimicrobial Agents and Chemotherapy. 17-20 September 2007, Chicago, IL, USA
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Schöller-Gyüre, M.1
Kakuda, T.N.2
De Smedt, G.3
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56
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77957363599
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Pharmacokinetics (PK) of once-daily etravirine (ETR) without and with once-daily darunavir/ritonavir (DRV/r) in antiretroviral-naive HIV-1-infected adults
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Abstract O413
-
Lalezari J, DeJesus E, Osiyemi O, et al. Pharmacokinetics (PK) of once-daily etravirine (ETR) without and with once-daily darunavir/ritonavir (DRV/r) in antiretroviral-naive HIV-1-infected adults. 9th International Congress on Drug Therapy and HIV Infection. 9-13 November 2008, Glasgow, UK. Abstract O413.
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9th International Congress on Drug Therapy and HIV Infection. 9-13 November 2008, Glasgow, UK
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Lalezari, J.1
DeJesus, E.2
Osiyemi, O.3
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57
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77957367636
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Pharmacokinetics and dose selection of etravirine in HIV-infected children between 6 and 17 years, inclusive
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Abstract S-167
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Konigs C, Feiterna-Sperling C, Esposito S, et al. Pharmacokinetics and dose selection of etravirine in HIV-infected children between 6 and 17 years, inclusive. 16th Conference on Retroviruses and Opportunistic Infections. 8-11 February 2009, Montreal, QC, Canada. Abstract S-167.
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16th Conference on Retroviruses and Opportunistic Infections. 8-11 February 2009, Montreal, QC, Canada
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Konigs, C.1
Feiterna-Sperling, C.2
Esposito, S.3
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58
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69849107159
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Clinical pharmacokinetics and pharmacodynamics of etravirine
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Schöller-Gyüre M, Kakuda TN, Raoof A, et al. Clinical pharmacokinetics and pharmacodynamics of etravirine. Clin Pharmacokinet 2009; 48:561-574.
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(2009)
Clin Pharmacokinet
, vol.48
, pp. 561-574
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Schöller-Gyüre, M.1
Kakuda, T.N.2
Raoof, A.3
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59
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77957341685
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Mass balance of 14C-labelled TMC125 in healthy volunteers
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Abstract 78
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Schöller-Gyüre M, Raoof A, Mannens G, et al. Mass balance of 14C-labelled TMC125 in healthy volunteers. 8th International Workshop on Clinical Pharmacology of HIV Therapy. 16-18 April 2007, Budapest, Hungary. Abstract 78.
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8th International Workshop on Clinical Pharmacology of HIV Therapy. 16-18 April 2007, Budapest, Hungary
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Schöller-Gyüre, M.1
Raoof, A.2
Mannens, G.3
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60
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57049148690
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Minimal pharmacokinetic interaction between the human immunodeficiency virus nonnucleoside reverse transcriptase inhibitor etravirine and the integrase inhibitor raltegravir in healthy subjects
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Anderson MS, Kakuda TN, Hanley W, et al. Minimal pharmacokinetic interaction between the human immunodeficiency virus nonnucleoside reverse transcriptase inhibitor etravirine and the integrase inhibitor raltegravir in healthy subjects. Antimicrob Agents Chemother 2008; 52:4228-4232.
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(2008)
Antimicrob Agents Chemother
, vol.52
, pp. 4228-4232
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Anderson, M.S.1
Kakuda, T.N.2
Hanley, W.3
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62
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77957341947
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An open, randomized, two-period, crossover study in two cohorts to investigate the effect of steady-state TMC125 (etravirine) and the combination of TMC125/darunavir/ritonavir on the steady-state pharmacokinetics of oral maraviroc in healthy subjects
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Abstract P4.3/02
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Davis J, Schöller-Gyüre M, Kakuda TN, et al. An open, randomized, two-period, crossover study in two cohorts to investigate the effect of steady-state TMC125 (etravirine) and the combination of TMC125/darunavir/ ritonavir on the steady-state pharmacokinetics of oral maraviroc in healthy subjects. 11th European AIDS Conference. 24-27 October 2007, Madrid, Spain. Abstract P4.3/02.
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11th European AIDS Conference. 24-27 October 2007, Madrid, Spain
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Davis, J.1
Schöller-Gyüre, M.2
Kakuda, T.N.3
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63
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68049094896
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No significant interaction between TMC125 and didanosine (ddI) in healthy volunteers
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Abstract WePe3.3C16
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Schöller M, Hoetelmans R, Bollen S, et al. No significant interaction between TMC125 and didanosine (ddI) in healthy volunteers. 3rd International AIDS Society Conference on HIV Pathogenesis and Treatment. 24-27 July 2005, Rio de Janeiro, Brazil. Abstract WePe3.3C16.
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3rd International AIDS Society Conference on HIV Pathogenesis and Treatment. 24-27 July 2005, Rio de Janeiro, Brazil
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Schöller, M.1
Hoetelmans, R.2
Bollen, S.3
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64
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77957353251
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Pharmacokinetics and safety of adding TMC125 to stable regimens of saquinavir, lopinavir, ritonavir, and NRTI in HIV+ adults
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Abstract 575b
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Harris M, Zala C, Ramirez S, et al. Pharmacokinetics and safety of adding TMC125 to stable regimens of saquinavir, lopinavir, ritonavir, and NRTI in HIV+ adults. 13th Conference on Retroviruses and Opportunistic Infections. 5-8 February 2006, Denver, CO, USA. Abstract 575b.
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13th Conference on Retroviruses and Opportunistic Infections. 5-8 February 2006, Denver, CO, USA
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Harris, M.1
Zala, C.2
Ramirez, S.3
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65
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58149489322
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Pharmacokinetics of elvitegravir and etravirine following coadministration of ritonavir-boosted elvitegravir and etravirine
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Ramanathan S, Kakuda TN, Mack R, West S, Kearney BP. Pharmacokinetics of elvitegravir and etravirine following coadministration of ritonavir-boosted elvitegravir and etravirine. Antivir Ther 2008; 13:1011-1017.
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(2008)
Antivir Ther
, vol.13
, pp. 1011-1017
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Ramanathan, S.1
Kakuda, T.N.2
Mack, R.3
West, S.4
Kearney, B.P.5
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66
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70349540810
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Effect of TMC125 on sildenafil pharmacokinetics
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Abstract 45
-
Schöller-Gyüre M, Debroye C, Vyncke V, et al. Effect of TMC125 on sildenafil pharmacokinetics. 7th International Workshop of Clinical Pharmacology. 20-22 April 2006, Lisbon, Portugal. Abstract 45.
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7th International Workshop of Clinical Pharmacology. 20-22 April 2006, Lisbon, Portugal
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Schöller-Gyüre, M.1
Debroye, C.2
Vyncke, V.3
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67
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66949111695
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Pharmacokinetic interaction between the non-nucleoside reverse transcriptase inhibitor (NNRTI) TMC125 and atorvastatin in HIV-negative volunteers
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Abstract WEPEA106
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Schöller-Gyüre M, Kakuda TN, De Smedt G, et al. Pharmacokinetic interaction between the non-nucleoside reverse transcriptase inhibitor (NNRTI) TMC125 and atorvastatin in HIV-negative volunteers. 4th IAS Conference on HIV Pathogenesis, Treatment and Prevention. 22-25 July 2007, Sydney, Australia. Abstract WEPEA106.
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4th IAS Conference on HIV Pathogenesis, Treatment and Prevention. 22-25 July 2007, Sydney, Australia
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Schöller-Gyüre, M.1
Kakuda, T.N.2
De Smedt, G.3
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68
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77957364646
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No pharmacokinetic interaction between TMC125 (etravirine; ETR) and paroxetine in HIV-negative volunteers
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Abstract P4.3/01
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Schöller-Gyüre M, Kakuda TN, Bollen S, et al. No pharmacokinetic interaction between TMC125 (etravirine; ETR) and paroxetine in HIV-negative volunteers. 11th European AIDS Conference. 24-27 October 2007, Madrid, Spain. Abstract P4.3/01.
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11th European AIDS Conference. 24-27 October 2007, Madrid, Spain
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Schöller-Gyüre, M.1
Kakuda, T.N.2
Bollen, S.3
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69
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51649083570
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A pharmacokinetic study of etravirine (TMC125) co-administered with ranitidine and omeprazole in HIV-negative volunteers
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Schöller-Gyüre M, Kakuda TN, De Smedt G, et al. A pharmacokinetic study of etravirine (TMC125) co-administered with ranitidine and omeprazole in HIV-negative volunteers. Br J Clin Pharmacol 2008; 66:508-516.
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Br J Clin Pharmacol
, vol.66
, pp. 508-516
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Schöller-Gyüre, M.1
Kakuda, T.N.2
De Smedt, G.3
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70
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34547780413
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Pharmacokinetics of darunavir/ritonavir and TMC125 alone and co-administered in HIV-negative volunteers
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Schöller-Gyüre M, Kakuda T, Sekar V, et al. Pharmacokinetics of darunavir/ritonavir and TMC125 alone and co-administered in HIV-negative volunteers. Antivir Ther 2007; 12:789-796.
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Antivir Ther
, vol.12
, pp. 789-796
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Schöller-Gyüre, M.1
Kakuda, T.2
Sekar, V.3
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71
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33747845304
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Pharmacokinetic interactions between HIV antiretroviral therapy and drugs used to treat opioid dependence
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Maas B, Kerr T, Fairbairn N, Montaner J, Wood E. Pharmacokinetic interactions between HIV antiretroviral therapy and drugs used to treat opioid dependence. Expert Opin Drug Metab Toxicol 2006; 2:533-543.
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Expert Opin Drug Metab Toxicol
, vol.2
, pp. 533-543
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Maas, B.1
Kerr, T.2
Fairbairn, N.3
Montaner, J.4
Wood, E.5
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72
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39149138092
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Pharmacokinetic and pharmacodynamic study of the concomitant administration of methadone and TMC125 in HIV-negative volunteers
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Schöller-Gyüre M, Van den Brink W, Kakuda TN, et al. Pharmacokinetic and pharmacodynamic study of the concomitant administration of methadone and TMC125 in HIV-negative volunteers. J Clin Pharmacol 2008; 48:322-329.
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J Clin Pharmacol
, vol.48
, pp. 322-329
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Schöller-Gyüre, M.1
Van Den Brink, W.2
Kakuda, T.N.3
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