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Volumn 27, Issue 10, 2010, Pages 2063-2074

Development of PLGA-based injectable delivery systems for hydrophobic fenretinide

Author keywords

controlled release; fenretinide; hydrophobic drug; in situ implant; s o w PLGA microparticle

Indexed keywords

1 METHYL 2 PYRROLIDINONE; DICHLOROMETHANE; FENRETINIDE; METHANOL; POLYGLACTIN; POLYSORBATE 80;

EID: 77957331565     PISSN: 07248741     EISSN: 1573904X     Source Type: Journal    
DOI: 10.1007/s11095-010-0202-y     Document Type: Article
Times cited : (54)

References (36)
  • 1
    • 0018292530 scopus 로고
    • New Long-Acting Injectable Microcapsule Contraceptive System
    • 114054 1:CAS:528:DyaL3cXhtFWmug%3D%3D
    • LR Beck DR Cowsar DH Lewis JW Gibson CE Flowers 1979 New Long-Acting Injectable Microcapsule Contraceptive System Am J Obstet Gynecol 135 419 26 114054 1:CAS:528:DyaL3cXhtFWmug%3D%3D
    • (1979) Am J Obstet Gynecol , vol.135 , pp. 419-26
    • Beck, L.R.1    Cowsar, D.R.2    Lewis, D.H.3    Gibson, J.W.4    Flowers, C.E.5
  • 3
    • 0036000111 scopus 로고    scopus 로고
    • Recent advances in the stabilization of proteins encapsulated in injectable PLGA delivery systems
    • DOI 10.1615/CritRevTherDrugCarrierSyst.v19.i1.20
    • SP Schwendeman 2002 Recent advances in the stabilization of proteins encapsulated in injectable PLGA delivery systems Crit Rev Ther Drug 19 73 98 10.1615/CritRevTherDrugCarrierSyst.v19.i1.20 1:CAS:528:DC%2BD38XksFaltL0%3D (Pubitemid 34521249)
    • (2002) Critical Reviews in Therapeutic Drug Carrier Systems , vol.19 , Issue.1 , pp. 73-98
    • Schwendeman, S.P.1
  • 4
    • 9244253168 scopus 로고    scopus 로고
    • Biodegradable poly(lactic-co-glycolic acid) microparticles for injectable delivery of vaccine antigens
    • DOI 10.1016/j.addr.2004.09.003, PII S0169409X04002091
    • WL Jiang RK Gupta MC Deshpande SP Schwendeman 2005 Biodegradable poly(lactic-co-glycolic acid) microparticles for injectable delivery of vaccine antigens Adv Drug Deliver Rev 57 391 410 10.1016/j.addr.2004.09.003 1:CAS:528:DC%2BD2cXhtVSntbrO (Pubitemid 39550967)
    • (2005) Advanced Drug Delivery Reviews , vol.57 , Issue.3 SPEC. ISS. , pp. 391-410
    • Jiang, W.1    Gupta, R.K.2    Deshpande, M.C.3    Schwendeman, S.P.4
  • 5
    • 55649104973 scopus 로고    scopus 로고
    • Principles of encapsulating hydrophobic drugs in PLA/PLGA microparticles
    • 10.1016/j.ijpharm.2008.04.042 18621492 1:CAS:528:DC%2BD1cXhtlOnurjF
    • C Wischke SP Schwendeman 2008 Principles of encapsulating hydrophobic drugs in PLA/PLGA microparticles Int J Pharm 364 298 327 10.1016/j.ijpharm.2008. 04.042 18621492 1:CAS:528:DC%2BD1cXhtlOnurjF
    • (2008) Int J Pharm , vol.364 , pp. 298-327
    • Wischke, C.1    Schwendeman, S.P.2
  • 6
    • 0028948839 scopus 로고
    • A Theoretical Basis for a Biopharmaceutic Drug Classification-the Correlation of in-Vitro Drug Product Dissolution and in-Vivo Bioavailability
    • 10.1023/A:1016212804288 7617530 1:CAS:528:DyaK2MXksVGqur8%3D
    • GL Amidon H Lennernas VP Shah JR Crison 1995 A Theoretical Basis for a Biopharmaceutic Drug Classification-the Correlation of in-Vitro Drug Product Dissolution and in-Vivo Bioavailability Pharm Res 12 413 20 10.1023/A: 1016212804288 7617530 1:CAS:528:DyaK2MXksVGqur8%3D
    • (1995) Pharm Res , vol.12 , pp. 413-20
    • Amidon, G.L.1    Lennernas, H.2    Shah, V.P.3    Crison, J.R.4
  • 7
    • 12244275011 scopus 로고    scopus 로고
    • BCNU-loaded poly(D, L-lactide-co-glycolide) wafer and antitumor activity against XF-498 human CNS tumor cells in vitro
    • DOI 10.1016/S0378-5173(02)00543-4, PII S0378517302005434
    • H Seong TK An G Khang SU Choi CO Lee HB Lee 2003 BCNU-loadedpoly(D, L-lactide-co-glycolide) wafer and antitumor activity against XF-498 human CNS tumor cells in vitro Int J Pharm 251 1 12 10.1016/S0378-5173(02)00543-4 12527170 1:CAS:528:DC%2BD3sXis1Whsg%3D%3D (Pubitemid 36071455)
    • (2003) International Journal of Pharmaceutics , vol.251 , Issue.1-2 , pp. 1-12
    • Seong, H.1    An, T.K.2    Khang, G.3    Choi, S.-U.4    Lee, C.O.5    Lee, H.B.6
  • 8
    • 34247564699 scopus 로고    scopus 로고
    • Intratumoral delivery of paclitaxel-loaded poly(lactic-co-glycolic acid) microspheres for Hep-2 laryngeal squamous cell carcinoma xenografts
    • DOI 10.1097/CAD.0b013e328012bccd, PII 0000181320070400000011
    • M Xie L Zhou T Hu M Yao 2007 Intratumoral delivery of paclitaxel-loaded poly(lactic-co-glycolic acid) microspheres for Hep-2 laryngeal squamous cell carcinoma xenografts Anticancer Drugs 18 459 66 10.1097/CAD.0b013e328012bccd 17351398 1:CAS:528:DC%2BD2sXis1anurY%3D (Pubitemid 46712409)
    • (2007) Anti-Cancer Drugs , vol.18 , Issue.4 , pp. 459-466
    • Xie, M.1    Zhou, L.2    Hu, T.3    Yao, M.4
  • 10
    • 33748606380 scopus 로고    scopus 로고
    • Mechanisms of fenretinide-induced apoptosis
    • DOI 10.1007/s10495-006-9289-3
    • N Hail HJ Kim R Lotan 2006 Mechanisms of fenretinide-induced apoptosis Apoptosis 11 1677 94 10.1007/s10495-006-9289-3 16850162 1:CAS:528: DC%2BD28XptF2rurg%3D (Pubitemid 44376243)
    • (2006) Apoptosis , vol.11 , Issue.10 , pp. 1677-1694
    • Hail Jr., N.1    Kim, H.J.2    Lotan, R.3
  • 11
    • 0022973551 scopus 로고
    • N-(4-Hydroxyphenyl)-All-Trans-Retinamide Pharmacokinetics in Female Rats and Mice
    • 2877832 1:CAS:528:DyaL2sXislensA%3D%3D
    • TA Hultin CM May RC Moon 1986 N-(4-Hydroxyphenyl)-All-Trans-Retinamide Pharmacokinetics in Female Rats and Mice Drug Metab Dispos 14 714 7 2877832 1:CAS:528:DyaL2sXislensA%3D%3D
    • (1986) Drug Metab Dispos , vol.14 , pp. 714-7
    • Hultin, T.A.1    May, C.M.2    Moon, R.C.3
  • 12
    • 77957347110 scopus 로고    scopus 로고
    • U.S. National Institutes of Health
    • U.S. National Institutes of Health. www.clinicaltrials.gov.
  • 13
    • 0141919699 scopus 로고    scopus 로고
    • Lipofuscin and macular degeneration
    • DOI 10.1301/nr.2003.oct.342-346
    • G Wolf 2003 Lipofuscin and macular degeneration Nutr Rev 61 342 6 10.1301/nr.2003.oct.342-346 14604266 (Pubitemid 37243712)
    • (2003) Nutrition Reviews , vol.61 , Issue.10 , pp. 342-346
    • Wolf, G.1
  • 14
    • 33644795859 scopus 로고    scopus 로고
    • Reductions in serum vitamin A arrest accumulation of toxic retinal fluorophores: A potential therapy for treatment of lipofuscin-based retinal diseases
    • DOI 10.1167/iovs.05-0820
    • RA Radu Y Han TV Bui S Nusinowitz D Bok J Lichter K Widder GH Travis NL Mata 2005 Reductions in serum vitamin A arrest accumulation of toxic retinal fluorophores: a potential therapy for treatment of lipofuscin-based retinal diseases Invest Ophthalmol Vis Sci 46 4393 401 10.1167/iovs.05-0820 16303925 (Pubitemid 44264531)
    • (2005) Investigative Ophthalmology and Visual Science , vol.46 , Issue.12 , pp. 4393-4401
    • Radu, R.A.1    Han, Y.2    Bui, T.V.3    Nusinowitz, S.4    Bok, D.5    Lichter, J.6    Widder, K.7    Travis, G.H.8    Mata, N.L.9
  • 17
    • 35548984440 scopus 로고    scopus 로고
    • Fenretinide-polyvinylalcohol conjugates: New systems allowing fenretinide intravenous administration
    • DOI 10.1021/bm7005592
    • I Orienti G Zuccari V Bergamante R Carosio R Gotti M Cilli PG Montaldo 2007 Fenretinide-polyvinylalcohol conjugates: New systems allowing fenretinide intravenous administration Biomacromolecules 8 3258 62 10.1021/bm7005592 17883277 1:CAS:528:DC%2BD2sXhtVKgtbvO (Pubitemid 350011650)
    • (2007) Biomacromolecules , vol.8 , Issue.10 , pp. 3258-3262
    • Orienti, I.1    Zuccari, G.2    Bergamante, V.3    Carosio, R.4    Gotti, R.5    Cilli, M.6    Montaldo, P.G.7
  • 18
    • 36448993341 scopus 로고    scopus 로고
    • Antitumor activity of 4-(N-hydroxyphenyl)retinamide conjugated with poly(l-glutamic acid) against ovarian cancer xenografts
    • DOI 10.1016/j.ygyno.2007.07.077, PII S0090825807005409
    • C Zou M Brewer X Cao R Zang J Lin Y Deng C Li 2007 Antitumor activity of 4-(N-hydroxyphenyl)retinamide conjugated with poly(L-glutamic acid) against ovarian cancer xenografts Gynecol Oncol 107 441 9 10.1016/j.ygyno.2007.07.077 17854871 1:CAS:528:DC%2BD2sXhtlyrt73F (Pubitemid 350167464)
    • (2007) Gynecologic Oncology , vol.107 , Issue.3 , pp. 441-449
    • Zou, C.1    Brewer, M.2    Cao, X.3    Zang, R.4    Lin, J.5    Deng, Y.6    Li, C.7
  • 19
    • 67349123353 scopus 로고    scopus 로고
    • Enhanced in vivo antitumor efficacy of fenretinide encapsulated in polymeric micelles
    • 10.1016/j.ijpharm.2009.01.019 19429294 1:CAS:528:DC%2BD1MXltlSjsLo%3D
    • T Okuda S Kawakami Y Higuchi T Satoh Y Oka M Yokoyama F Yamashita M Hashida 2009 Enhanced in vivo antitumor efficacy of fenretinide encapsulated in polymeric micelles Int J Pharm 373 100 6 10.1016/j.ijpharm.2009.01.019 19429294 1:CAS:528:DC%2BD1MXltlSjsLo%3D
    • (2009) Int J Pharm , vol.373 , pp. 100-6
    • Okuda, T.1    Kawakami, S.2    Higuchi, Y.3    Satoh, T.4    Oka, Y.5    Yokoyama, M.6    Yamashita, F.7    Hashida, M.8
  • 21
    • 0032951672 scopus 로고    scopus 로고
    • Biocompatibility of a biodegradable in situ forming implant system in rhesus monkeys
    • DOI 10.1002/(SICI)1097-4636(19990605)45:3<231::AID-JBM11>3.0.CO;2-H
    • MA Royals SM Fujita GL Yewey J Rodriguez PC Schultheiss RL Dunn 1999 Biocompatibility of a biodegradable in situ forming implant system in rhesus monkeys J Biomed Mater Res 45 231 9 10.1002/(SICI)1097-4636(19990605)45: 3<231::AID-JBM11>3.0.CO;2-H 10397981 1:CAS:528:DyaK1MXisVeqtbY%3D (Pubitemid 29165939)
    • (1999) Journal of Biomedical Materials Research , vol.45 , Issue.3 , pp. 231-239
    • Royals, M.A.1    Fujita, S.M.2    Yewey, G.L.3    Rodriguez, J.4    Schultheiss, P.C.5    Dunn, R.L.6
  • 23
    • 37849034324 scopus 로고    scopus 로고
    • Effects of process and formulation parameters on characteristics and internal morphology of poly(D, L-lactide-co-glycolide) microspheres formed by the solvent evaporation method
    • 10.1016/j.ejpb.2007.06.008 17651954 1:CAS:528:DC%2BD1cXlsF2msw%3D%3D
    • SR Mao Y Shi L Li J Xu A Schaper T Kissel 2008 Effects of process and formulation parameters on characteristics and internal morphology of poly(D, L-lactide-co-glycolide) microspheres formed by the solvent evaporation method Eur J Pharm Biopharm 68 214 23 10.1016/j.ejpb.2007.06.008 17651954 1:CAS:528:DC%2BD1cXlsF2msw%3D%3D
    • (2008) Eur J Pharm Biopharm , vol.68 , pp. 214-23
    • Mao, S.R.1    Shi, Y.2    Li, L.3    Xu, J.4    Schaper, A.5    Kissel, T.6
  • 24
    • 0024452570 scopus 로고
    • Plasma Retinol Level Reduction by the Synthetic Retinoid Fenretinide-a One-Year Follow-up-Study of Breast-Cancer Patients
    • 2529028 1:STN:280:DyaK3c%2Fgt12quw%3D%3D
    • F Formelli R Carsana A Costa F Buranelli T Campa G Dossena A Magni M Pizzichetta 1989 Plasma Retinol Level Reduction by the Synthetic Retinoid Fenretinide-a One-Year Follow-up-Study of Breast-Cancer Patients Cancer Res 49 6149 52 2529028 1:STN:280:DyaK3c%2Fgt12quw%3D%3D
    • (1989) Cancer Res , vol.49 , pp. 6149-52
    • Formelli, F.1    Carsana, R.2    Costa, A.3    Buranelli, F.4    Campa, T.5    Dossena, G.6    Magni, A.7    Pizzichetta, M.8
  • 25
    • 0035868837 scopus 로고    scopus 로고
    • Safety of the synthetic retinoid fenretinide: Long-term results from a controlled clinical trial for the prevention of contralateral breast cancer
    • 11250995 1:CAS:528:DC%2BD3MXisFygs78%3D
    • T Camerini L Mariani G De Palo E Marubini MG Di Mauro A Decensi A Costa U Veronesi 2001 Safety of the synthetic retinoid fenretinide: Long-term results from a controlled clinical trial for the prevention of contralateral breast cancer J Clin Oncol 19 1664 70 11250995 1:CAS:528:DC%2BD3MXisFygs78%3D
    • (2001) J Clin Oncol , vol.19 , pp. 1664-70
    • Camerini, T.1    Mariani, L.2    De Palo, G.3    Marubini, E.4    Di Mauro, M.G.5    Decensi, A.6    Costa, A.7    Veronesi, U.8
  • 26
    • 0034002855 scopus 로고    scopus 로고
    • Controlled release of β-estradiol from PLAGA microparticles: The effect of organic phase solvent on encapsulation and release
    • DOI 10.1016/S0168-3659(99)00219-9, PII S0168365999002199
    • DT Birnbaum JD Kosmala DB Henthorn L Brannon-Peppas 2000 Controlled release of beta-estradiol from PLAGA microparticles: The effect of organic phase solvent on encapsulation and release J Control Release 65 375 87 10.1016/S0168-3659(99)00219-9 10699296 1:CAS:528:DC%2BD3cXhtl2qsbw%3D (Pubitemid 30122940)
    • (2000) Journal of Controlled Release , vol.65 , Issue.3 , pp. 375-387
    • Birnbaum, D.T.1    Kosmala, J.D.2    Henthorn, D.B.3    Brannon-Peppas, L.4
  • 27
    • 0029561449 scopus 로고
    • Prediction of solvent removal profile and effect on properties for peptide-loaded PLGA microspheres prepared by solvent extraction/evaporation method
    • 10.1016/0168-3659(95)00076-3 1:CAS:528:DyaK2MXhtVSgt7vO
    • W-I Li K Anderson R Mehta P DeLuca 1995 Prediction of solvent removal profile and effect on properties for peptide-loaded PLGA microspheres prepared by solvent extraction/evaporation method J Control Release 37 199 10.1016/0168-3659(95)00076-3 1:CAS:528:DyaK2MXhtVSgt7vO
    • (1995) J Control Release , vol.37 , pp. 199
    • Li, W.-I.1    Anderson, K.2    Mehta, R.3    Deluca, P.4
  • 28
    • 0023904637 scopus 로고
    • Solvent Selection in the Preparation of Poly(Dl-Lactide) Microspheres Prepared by the Solvent Evaporation Method
    • 10.1016/0378-5173(88)90073-7 1:CAS:528:DyaL1cXhvFaksL8%3D
    • R Bodmeier JW Mcginity 1988 Solvent Selection in the Preparation of Poly(Dl-Lactide) Microspheres Prepared by the Solvent Evaporation Method Int J Pharm 43 179 86 10.1016/0378-5173(88)90073-7 1:CAS:528:DyaL1cXhvFaksL8%3D
    • (1988) Int J Pharm , vol.43 , pp. 179-86
    • Bodmeier, R.1    McGinity, J.W.2
  • 29
    • 0022473091 scopus 로고
    • Formation and characterization of cisplatin loaded poly(d, l-lactide) microspheres for chemoembolization
    • 10.1002/jps.2600750805 3772745 1:CAS:528:DyaL2sXnt1yiug%3D%3D
    • G Spenlehauer M Veillard JP Benoit 1986 Formation and characterization of cisplatin loaded poly(d, l-lactide) microspheres for chemoembolization J Pharm Sci 75 750 5 10.1002/jps.2600750805 3772745 1:CAS:528:DyaL2sXnt1yiug%3D%3D
    • (1986) J Pharm Sci , vol.75 , pp. 750-5
    • Spenlehauer, G.1    Veillard, M.2    Benoit, J.P.3
  • 30
    • 84913460925 scopus 로고
    • Continuous release pharmaceutical compositions
    • FG Hutchinson 1986 Continuous release pharmaceutical compositions European Patent EP 58 481
    • (1986) European Patent EP , vol.58 , pp. 481
    • Hutchinson, F.G.1
  • 31
    • 0023943907 scopus 로고
    • Controlled-Release of Leuprolide Acetate from Polylactic Acid or Copoly(Lactic Glycolic) Acid Microcapsules-Influence of Molecular-Weight and Copolymer Ratio of Polymer
    • 3138032 1:CAS:528:DyaL1cXks1Wgt7o%3D
    • Y Ogawa M Yamamoto S Takada H Okada T Shimamoto 1988 Controlled-Release of Leuprolide Acetate from Polylactic Acid or Copoly(Lactic Glycolic) Acid Microcapsules-Influence of Molecular-Weight and Copolymer Ratio of Polymer Chem Pharm Bull 36 1502 7 3138032 1:CAS:528:DyaL1cXks1Wgt7o%3D
    • (1988) Chem Pharm Bull , vol.36 , pp. 1502-7
    • Ogawa, Y.1    Yamamoto, M.2    Takada, S.3    Okada, H.4    Shimamoto, T.5
  • 32
    • 41249098853 scopus 로고    scopus 로고
    • Evaluation of in vivo-in vitro release of dexamethasone from PLGA microspheres
    • 10.1016/j.jconrel.2008.01.004 18282629 1:CAS:528:DC%2BD1cXkt1OrtL4%3D
    • BS Zolnik DJ Burgess 2008 Evaluation of in vivo-in vitro release of dexamethasone from PLGA microspheres J Control Release 127 137 45 10.1016/j.jconrel.2008.01.004 18282629 1:CAS:528:DC%2BD1cXkt1OrtL4%3D
    • (2008) J Control Release , vol.127 , pp. 137-45
    • Zolnik, B.S.1    Burgess, D.J.2
  • 33
    • 23144436866 scopus 로고    scopus 로고
    • Stabilized nanoparticles of phytosterol by rapid expansion from supercritical solution into aqueous solution
    • 10.1208/pt050456 15760053
    • M Turk R Lietzow 2004 Stabilized nanoparticles of phytosterol by rapid expansion from supercritical solution into aqueous solution AAPS PharmSciTech 5 e56 10.1208/pt050456 15760053
    • (2004) AAPS PharmSciTech , vol.5 , pp. 56
    • Turk, M.1    Lietzow, R.2
  • 35
    • 0033032661 scopus 로고    scopus 로고
    • Phase inversion dynamics of PLGA solutions related to drug delivery
    • DOI 10.1016/S0168-3659(98)00158-8, PII S0168365998001588
    • PD Graham KJ Brodbeck AJ McHugh 1999 Phase inversion dynamics of PLGA solutions related to drug delivery J Controlled Release 58 233 45 10.1016/S0168-3659(98)00158-8 1:CAS:528:DyaK1MXhsVentL8%3D (Pubitemid 29112894)
    • (1999) Journal of Controlled Release , vol.58 , Issue.2 , pp. 233-245
    • Graham, P.D.1    Brodbeck, K.J.2    McHugh, A.J.3
  • 36
    • 0842332476 scopus 로고    scopus 로고
    • Determination of Water-Soluble Acid Distribution in Poly(lactide-co- glycolide)
    • DOI 10.1002/jps.10524
    • AG Ding SP Schwendeman 2004 Determination of water-soluble acid distribution in poly(lactide-co-glycolide) J Pharm Sci 93 322 31 10.1002/jps.10524 14705190 1:CAS:528:DC%2BD2cXhsFagu7g%3D (Pubitemid 38174255)
    • (2004) Journal of Pharmaceutical Sciences , vol.93 , Issue.2 , pp. 322-331
    • Ding, A.G.1    Schwendeman, S.P.2


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