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Binding studies of luzopeptin A to DNA revealed that the compound is a bifunctional intercalator and that it favors DNA regions containing alternating A and T residues
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50'S of quinoxapeptin A against DNA polymerase a,b, g and d are equal to 2563, 615, 1798 and 494 nM, respectively). This activity is comparable to that reported for luzopeptins.
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