Ring-chain tautomerism in 2,2-bis(2-thienyl)-tetrahydrofurans: Preparation of [butene-2H5]-tiagabine

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 53, Issue 9, 2010, Pages 598-600

  Herberta, John M ^a   Mathersa, Trevor W ^a  

^a Sanof Aventis   (United Kingdom)

Author keywords

2,2 bis(2 thienyl)tetrahydrofuran; Deuterium; Gabitril; Piperidines

Indexed keywords

SYNTHESIS (CHEMICAL);

2,2-BIS(2-THIENYL)TETRAHYDROFURAN; BUTENE-2; BUTYROLACTONES; GABITRIL; PIPERIDINE; RING OPENS; RING-CHAIN TAUTOMERISM; TETRA-HYDROFURAN; TETRAHYDROFURANS; THIENYL;

BUTENES;

1,1 BIS(3 METHYL 2 THIENYL)BUTANE 1,4 DIOL; 2,2 BIS(2 THIENYL)TETRAHYDROFURAN; 2,2 BIS(3 METHYL 2 THIENYL)TETRAHYDROFURAN; 4,4 BIS(3 METHYL 2 THIENYL) 3 BUTEN 1 OL; RADIOPHARMACEUTICAL AGENT; TETRAHYDROFURAN DERIVATIVE; TIAGABINE BUTENE 2 H 5; UNCLASSIFIED DRUG;

ARTICLE; CYCLIZATION;

EID: 77956927802     PISSN: 03624803     EISSN: 10991344     Source Type: Journal    
DOI: 10.1002/jlcr.1787     Document Type: Article

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