Recent Advances in the Discovery and Development of Potential Antidiabetic Agents

Annual Reports in Medicinal Chemistry

Volumn 27, Issue C, 1992, Pages 219-226

  Colca, Jerry R ^a   Tanis, Steven P ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 77956843172     PISSN: 00657743     EISSN: None     Source Type: Book Series    
DOI: 10.1016/S0065-7743(08)60421-2     Document Type: Article

References (95)

1. Bransome, E.D., Diabetes Care, 15(Suppl. 1), 1991, 1.
2. DeFronzo, R.A., Ferrannini, E., Koivisto, V., Am. J. Med, 74, 1983, 52.
3. Reaven, G.M., Diabetes, 37, 1988, 1595.
4. DeFronzo, R.A., Diabetes, 37, 1988, 667.
5. Olefsky, J.M., Garvey, W.T., Henry, R.R., Matthei, S., Freidenberg, G.R., Am. J. Med., 85, 1988, 86.
6. DeFronzo, R.A., Bonadonna, R.C., Ferrannini, E., Diabetes Care, 15, 1992, 318.
7. Warram, J.H., Martin, B.C., Krolewski, A.S., Soeldner, J.S., Kahn, C.R., Ann. Intern. Med., 113, 1990, 909.
8. Kahn, S.E., Porte, D., Am. J. Med., 85, 1988, 4.
9. Taylor, R., Br. Med. Bull., 45, 1989, 73.
10. Boyd, A.E. 3rd, Aguilar, B.L., Bryan, J., Kunze, D.L., Moss, L., Nelson, D.A., Rajan, A.S., Raef, H., Xiang, H.D., Yaney, G.C., Recent Prog. Horm. Res., 47, 1991, 299.
11. Angel, I., Niddam, R., Langer, S.Z., J. Pharmacol. Exp. Ther., 254, 1990, 877.
12. Yamanaka, K., Kigoshi, S., Muramatsu, I., Eur. J. Pharmacol., 106, 1984, 625.
13. Kawazu, S., Suzuki, M., Negishi, K., Watanabe, T., Ishii, J., Diabetes, 36, 1987, 216.
14. Kawazu, S., Suzuki, M., Negishi, K., Ishii, J., Sando, H., Katagiri, H., Kanazawa, Y., Yamanouchi, S., Akanuma, Y., Kajinuma, H., Suzuki, K., Watanabe, K., Itoh, T., Kobayashi, T., Kosaka, K., Diabetes, 36, 1987, 221.
15. Kameda, K., Koyama, I., Abiko, Y., Biochim. Biophys. Acta, 677, 1981, 263.
16. Koh, G., Seino, Y., Tsuda, K., Nishi, S., Ishida, H., Takeda, J., Fukumoto, H., Taminato, T., Imura, H., Life Sci., 40, 1987, 1113.
17. Chapleo, C.B., Myers, P.L., Butler, R.C.M., Doxey, J.C., Roach, A.G., Roach, C.F.C., J. Med. Chem., 26, 1983, 823.
18. Chapleo, C.B., Myers, P.L., Butler, R.C.M., Davis, J.A., Doxey, J.C., Higgins, S.D., Myers, M., Roach, A.G., Smith, C.F.C., Stillings, M.R., Welbourn, A.P., J. Med. Chem., 27, 1984, 570.
19. Fagan, G.P., Chapleo, C.P., Lane, A.C., Myers, M., Roach, A.G., Roach, C.F.C., Stillings, M.R., Welbourn, A.P., J. Med. Chem., 31, 1988, 944.
20. D. Biggs, S. Langer, C. Morel, andM. Servin, U.S. Patent 4, 904, 684(1990).
21. Angel, I., Schoemaker, H., Azerhad, R., Bidet, S., Duval, N., Langer, S.Z., Int. J. Obesity, 14(Suppl. 2), 1990, 50 (Abstract IF12).
22. Ostenson, C.G., Pigon, J., Doxey, J.C., Efendic, S., J. Clin. Endocrin. Metab., 67, 1988, 1054.
23. Shinkai, H., Toi, K., Kumashiro, I., Seto, Y., Fukuma, M., Dan, K., Toyoshima, S., J. Med. Chem., 31, 1988, 2092.
24. Shinkai, H., Nishikawa, M., Sato, Y., Toi, K., Kumashiro, I., Seto, Y., Fukuma, M., Dan, K., Toyoshima, S., J. Med. Chem., 32, 1989, 1436.
25. Shinkai, H., Sato, Y., Bailey, C.J., Flatt, P.R., (eds.) New Antidiabetic Drugs, 1990, Smith-Gordon, London, 249.
26. Y. Sato, M. Nishikawa, H. Shinkai, andE. Sukegawa, Diabetes Res. Clin. Practice, in press(1992).
27. Geisen, K., Arzneim-Forsch/Drug Res., 38, 1988, 1120.
28. Yen, T.T., Dininger, N.B., Broderick, C.L., Gill, A.M., Arch. Int. Pharmacodyn., 308, 1990, 137.
29. R. Saperstein, R.M. Tolman, and E.E. Slater, U.S. Patent 4, 978, 667(1990).
30. Kreymann, B., Gitatei, M.A., Williams, G., Bloom, S.R., Lancet, II, 1987, 1300.
31. Fehmann, H.C., Habener, J.F., Endocrinology, 130, 1992, 159.
32. Steiner, K.E., Lien, E.L., Prog. Med. Chem., 24, 1987, 209.
33. Larsen, E.R., Clark, D.A., Stevenson, R.W., Ann. Rep. Med. Chem., 25, 1989, 205.
34. Colca, J.R., Morton, D.R., Bailey, C.J., Flatt, P.R., (eds.) New Antidiabetic Drugs, 1990, Smith-Gordon, London, 255.
35. Drugs of the Future, 15, 1990, 1080.
36. Drugs of the Future, 16, 1991, 853.
37. Suter, S.L., Nolan, J.J., Wallace, P., Gumbiner, B., Olefsky, J.M., Diabetes Care, 15, 1992, 193.
38. Kuzuya, T., Iwamoto, Y., Kosaka, K., Takebe, K., Yamanouchi, T., Kasuga, M., Kajinuma, H., Akanuma, Y., Yoshida, S., Shigeta, Y., Diabetes Res. Clin. Pract., 11, 1991, 147.
39. Stevenson, R.W., McPherson, R.K., Genereux, P.E., Danbury, B.H., Kreutter, D.K., Metabolism, 40, 1991, 1268.
40. Clark, D.A., Goldestein, S.W., Volkmann, R.A., Eggler, J.F., Holland, G.F., Hulin, B., Stevenson, R.W., Kreutter, D.K., Gibbs, E.M., Krupp, M.N., Merrigan, P., Kelbaugh, P.L., Andrews, E.G., Tickner, D.L., Suleske, R.T., Lamphere, C.H., Rajeckas, F.J., Kappeler, W.H., McDermott, R.E., Hutson, N.J., Johnson, M.R., J. Med. Chem., 34, 1991, 319.
41. Hofmann, C., Lorenz, K., Colca, J.R., Endocrinol., 129, 1991, 1915.
42. Hofmann, C.A., Edwards, C.W. III, Hillman, R.M., Colca, J.R., Endocrinol., 130, 1992, 735.
43. Gibbs, E.M., Genereux, P.E., Kreutter, D.K., Diabetologia, 32, 1989, 491A.
44. Colca, J.R., Dailey, C.F., Palazuk, B.J., Hillman, R.M., Dinh, D.M., Melchior, G.W., Spilman, C.H., Diabetes, 40, 1991, 1669.
45. Ikeda, H., Taketomi, S., Sugiyama, Y., Sodha, T., Meguro, K., Fujita, T., Arzneim-Forsch/Drug Res., 40, 1990, 156.
46. Sugiyama, Y., Taketomi, S., Shimura, Y., Ikeda, H., Fujita, T., Arzneim-Forsch/Drug Res., 40, 1990, 263.
47. Sugiyama, Y., Shimura, Y., Ikeda, H., Arzneim-Forsch/Drug Res., 40, 1990, 436.
48. Stevenson, R.W., Hutson, N.J., Krupp, M.N., Volkmann, R.M., Holland, G.F., Eggler, J.F., Clark, D.A., McPherson, R.K., Hall, K.L., Danbury, B.H., Gibbs, E.M., Kreutter, D.K., Diabetes, 39, 1990, 1218.
49. R.K. Dubey, T.A. Kotchen, M.A. Boegehold, and H.Y. Zhang, FASEB, abstract in press(1992).
50. Momose, Y., Meguro, K., Ikeda, H., Hatanaga, C., Ot, S., Sohda, T., Chem. Pharm. Bull., 39, 1991, 1440.
51. Sohda, T., Momose, Y., Meguro, K., Kawamatsu, Y., Sugiyama, Y., Ikeda, H., Arzneim-Forsch/Drug Res., 40, 1990, 37.
52. D.A. Clark, S.W. Goldstein, andB. Hulin, U.S. Patent 5, 036, 079(1991).
53. D.A. Clark, S.W. Goldstein, andB. Hulin, WO 9103474(1991).
54. D.A. Clark, and M.R. Johnson, U.S. Patent 4, 968, 707(1990).
55. B.C. C. Cantello, and P.T. Duff, European Patent 415, 605A(1991).
56. R.M. Hindley, R. Southgate, and P.T. Duff, European Patent 419, 035A(1991).
57. Zask, A., Jirkovsky, I., Nowicki, J.W., McCaleb, M.L., J. Med. Chem., 33, 1990, 1418.
58. A. Zask, andI. Jirkovsky, U.S. Patent 4, 997, 948(1991).
59. Dow, R.L., Bechle, B.M., Chou, T.T., Clark, D.A., Hulin, B., Stevenson, R.W., J. Med. Chem., 34, 1991, 1538.
60. S.W. Goldstein, U.S. Patent 5, 037, 842(1991).
61. J.W. Ellingboe, J.F. Bagli, and T.R. Alessi, U.S. Patent 4, 966, 975(1990).
62. T.R. Alessi, T.M. Dolak, J.W. Ellingboe, and L.J. Lombardo, U.S. Patent 4, 897, 405(1990).
63. T.R. Alessi, and T.M. Dolak, U.S. Patent 4, 895, 862(1990).
64. Kees, K.L., Cheeseman, R.S., Prozialeck, D.H., Steiner, K.E., J. Med. Chem., 32, 1989, 11.
65. Steiner, K.E., McCaleb, M.L., Kees, K.L., Bailey, C.J., Flatt, P.R., (eds.) New Antidiabetic Drugs, 1990, Smith-Gordon, London, 237.
66. Kees, K.L., Smith, T.M., McCaleb, M.L., Prozialeck, D.H., Cheeseman, R.S., Christos, T.E., Patt, W.C., Steiner, K.E., J. Med. Chem., 35, 1992, 944.
67. Yen, T.T., Schmiegel, K.K., Gold, G., Williams, G.D., Dininger, N.B., Broderick, C.L., Gill, A.M., Arch. Int. Pharmacodyn., 310, 1991, 162.
68. G.A. Youngdale, WO 8909224(1989).
69. R.A. Johnson, G.L. Bundy, G.A. Youngdale, D.R. Morton, and D.P. Wallach, U.S. Patent 4, 917, 826(1990).
70. Dominianni, S.J., Yen, T.T., J. Med. Chem., 32, 1989, 2301.
71. Yen, T.T., Dominianni, S.J., Harris, R.A., Stephens, T.W., Bailey, C.J., Flatt, P.R., (eds.) New Antidiabetic Drugs, 1990, Smith-Gordon, London, 245.
72. G. Balasubramanian, GB 2, 226, 562A(1990).
73. Reitz, A.B., Tuman, R.W., Marchione, C.S., Jordan, A.D. Jr., Bowden, C.R., Maryanoff, B.E., J. Med. Chem., 32, 1989, 2110.
74. Arch, J.R.S., Ainsworth, A.T., Cawthorne, M.A., Piercy, V., Sennitt, M.V., Thody, V.E., Wilson, C., Wilson, S., Nature, 309, 1984, 163.
75. Wilson, C.S., Wilson, V., Piercy, M., Sennitt, M.V., J.R. S. Arch, Eur. J. Pharmacol., 100, 1984, 309.
76. Thurlby, P.L., Ellis, R.D.M., Can. J. Physiol. Pharmacol., 64, 1986, 1111.
77. Henry, C., Buckert, A., Schutz, Y., Jequeir, E., Felber, J.P., Int. J. Obesity, 12, 1988, 227.
78. Golay, A., Felber, J.P., Jequier, E., DeFronzo, R.A., Ferrannini, E., Diabet. /Metab. Rev., 4, 1988, 727.
79. Watts, N.B., Spanheimer, R.G., DiGirolamo, M., Gebhart, S.S.P., Musey, V.C., Siddiq, Y.K., Phillips, L.S., Arch. Int. Med., 150, 1990, 803.
80. Challiss, J., Budohoski, L., Newsholme, E.A., Sennitt, M.V., Cawthorne, M.A., Biochem. Biophys. Res. Comm., 128, 1985, 928.
81. Hollenga, C., Haas, M., Deinum, J.T., Zaagsma, J., Horm. Metabol. Res., 22, 1990, 171.
82. Holloway, B.R., Howe, R., Rao, B.S., Stribling, D., Int. J. Obesity, 14(Suppl. 2), 1990, 51 (Abstract IF-15).
83. Holloway, B.R., Mayers, R., Jackson, J., Briscoe, M., Int. J. Obesity, 14(Suppl. 2), 1990, 142 (Abstract 2P-85).
84. Zaagsma, J., Nahorski, S.R., TIPS, 11, 1990, 3.
85. Selby, P.L., Sherratt, H.S.A., TIPS, 10, 1989, 495.
86. von-Herrath, M., Holzer, H., Z. Lebensm. Unters. Forsil., 186, 1988, 427.
87. Regen, D.M., Pilkis, S.J., Kraus-Friedmann, N., (eds.) Hormonal Control of Gluconeogenesis, III, 1986, CRC Press, Boca Raton, Florida, 101.
88. Leighton, B., Cooper, G.J.S., Nature, 335, 1988, 632.
89. Young, D.A., Deems, R.O., Deacon, R.W., McIntosh, R.H., Foley, J.E., Amer. J. Physiol., 259, 1990, E457.
90. Gill, A.M., Yen, T.T., Life Sciences, 48, 1990, 703.
91. Moore, C.X., Cooper, G.J.S., Biochem. Biophys. Res. Comm., 179, 1991, 1.
92. Taylor, R., Clin. Endocrinol., 34, 1991, 159.
93. Haring, H.U., Diabetologia, 34, 1991, 848.
94. Houslay, M.D., Wakelman, M.J.O., Pyne, N.J., TIBS II, 1986, 393.
95. Saltiel, A.R., J. Bioenerg. Biomembranes, 23, 1991, 29.