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Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 13, 2010, Pages 3906-3910

Design, synthesis and anticancer activity of piperazine hydroxamates and their histone deacetylase (HDAC) inhibitory activity

(12) Chetan, Bhadaliya a Bunha, Mahesh a Jagrat, Monika a Sinha, Barij Nayan a Saiko, Philipp a Graser, Geraldine b Szekeres, Thomas b Raman, Ganapathy c Rajendran, Praveen c Moorthy, Dhatchana c Basu, Arijit a Jayaprakash, Venkatesan a

a BIRLA INSTITUTE OF TECHNOLOGY (India)

b UNIVERSITY OF VIENNA (Austria)

c Orchid Research Laboratories Limited (India)

Author keywords

Histone deacetylase inhibitors; Hydroxamates; Piperazine linker; RR pharmacophore

Indexed keywords

ANTINEOPLASTIC AGENT; HISTONE DEACETYLASE 8; HISTONE DEACETYLASE INHIBITOR; PIPERAZINE HYDROXAMATE; UNCLASSIFIED DRUG; ZINC BINDING PROTEIN;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL CULTURE; CELL STRAIN HL 60; DRUG DESIGN; DRUG SCREENING; DRUG SYNTHESIS; HUMAN; HUMAN CELL; HUMAN TISSUE; IC 50; LEUKEMIA CELL LINE; PHARMACOPHORE; PROMYELOCYTIC LEUKEMIA;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL PROLIFERATION; CELL SURVIVAL; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; DRUG SCREENING ASSAYS, ANTITUMOR; HISTONE DEACETYLASE INHIBITORS; HISTONE DEACETYLASES; HUMANS; HYDROXAMIC ACIDS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; PIPERAZINES; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 77954315435 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.05.020 Document Type: Article

Times cited : (61)

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