메뉴 건너뛰기




Volumn 65, Issue 7, 2010, Pages 1441-1447

Bactericidal activity of besifloxacin against staphylococci, Streptococcus pneumoniae and Haemophilus influenzae

Author keywords

Bactericidal activity; Fluoroquinolones; Time kill

Indexed keywords

ANTIINFECTIVE AGENT; AZITHROMYCIN; BESIFLOXACIN; CIPROFLOXACIN; GATIFLOXACIN; MOXIFLOXACIN; TOBRAMYCIN; UNCLASSIFIED DRUG; 7-(3-AMINOHEXAHYDRO-1H-AZEPIN-1-YL)-8-CHLORO-1-CYCLOPROPYL-6-FLUORO-1,4-DIHYDRO-4-OXO-3-QUINOLINECARBOXYLIC ACID; AMINOGLYCOSIDE; AZEPINE DERIVATIVE; BACTERIAL DNA; BETA LACTAM; MACROLIDE; QUINOLONE DERIVATIVE;

EID: 77954188913     PISSN: 03057453     EISSN: 14602091     Source Type: Journal    
DOI: 10.1093/jac/dkq127     Document Type: Article
Times cited : (47)

References (27)
  • 1
    • 0002431230 scopus 로고
    • Mechanisms of action and resistance to quinolone antimicrobial agents
    • Wolfson JS, Hooper DC, eds. Washington, DC: ASM Press
    • Wolfson JS, Hooper DC, Swartz MN. Mechanisms of action and resistance to quinolone antimicrobial agents. In: Wolfson JS, Hooper DC, eds. Quinolone Antimicrobial Agents. Washington, DC: ASM Press, 1989; 5-34.
    • (1989) Quinolone Antimicrobial Agents , pp. 5-34
    • Wolfson, J.S.1    Hooper, D.C.2    Swartz, M.N.3
  • 2
    • 67749108274 scopus 로고    scopus 로고
    • Besifloxacin, a novel fluoroquinolone, has broad-spectrum in vitro activity against aerobic and anaerobic bacteria
    • Haas W, Pillar CP, Zurenko GE et al. Besifloxacin, a novel fluoroquinolone, has broad-spectrum in vitro activity against aerobic and anaerobic bacteria. Antimicrob Agents Chemother 2009; 53: 3552-60.
    • (2009) Antimicrob Agents Chemother , vol.53 , pp. 3552-3560
    • Haas, W.1    Pillar, C.P.2    Zurenko, G.E.3
  • 7
    • 0029743055 scopus 로고    scopus 로고
    • Comparative antimicrobial activity and post-antibiotic effect of azithromycin, clarithromycin and roxithromycin against some respiratory pathogens
    • Ferrara A, Dos SC, Cimbro M et al. Comparative antimicrobial activity and post-antibiotic effect of azithromycin, clarithromycin and roxithromycin against some respiratory pathogens. Int J Antimicrob Agents 1996; 7: 181-6.
    • (1996) Int J Antimicrob Agents , vol.7 , pp. 181-186
    • Ferrara, A.1    Dos, S.C.2    Cimbro, M.3
  • 8
    • 0023503132 scopus 로고
    • Spectrum and mode of action of azithromycin (CP-62,993), a new 15-membered-ring macrolide with improved potency against gram-negative organisms
    • Retsema J, Girard A, Schelkly W et al. Spectrum and mode of action of azithromycin (CP-62,993), a new 15-membered-ring macrolide with improved potency against gram-negative organisms. Antimicrob Agents Chemother 1987; 31: 1939-47.
    • (1987) Antimicrob Agents Chemother , vol.31 , pp. 1939-1947
    • Retsema, J.1    Girard, A.2    Schelkly, W.3
  • 9
    • 0037378762 scopus 로고    scopus 로고
    • Activity of and resistance to moxifloxacin in Staphylococcus aureus
    • Ince D, Zhang X, Hooper DC. Activity of and resistance to moxifloxacin in Staphylococcus aureus. Antimicrob Agents Chemother 2003; 47: 1410-5.
    • (2003) Antimicrob Agents Chemother , vol.47 , pp. 1410-1415
    • Ince, D.1    Zhang, X.2    Hooper, D.C.3
  • 10
    • 33744502866 scopus 로고    scopus 로고
    • Activity of gatifloxacin in an in vitro pharmacokinetic-pharmacodynamic model against Staphylococcus aureus strains either susceptible to ciprofloxacin or exhibiting various levels and mechanisms of ciprofloxacin resistance
    • Ba BB, Arpin C, Vidaillac C et al. Activity of gatifloxacin in an in vitro pharmacokinetic-pharmacodynamic model against Staphylococcus aureus strains either susceptible to ciprofloxacin or exhibiting various levels and mechanisms of ciprofloxacin resistance. Antimicrob Agents Chemother 2006; 50: 1931-6.
    • (2006) Antimicrob Agents Chemother , vol.50 , pp. 1931-1936
    • Ba, B.B.1    Arpin, C.2    Vidaillac, C.3
  • 11
    • 0033998520 scopus 로고    scopus 로고
    • Activities and postantibiotic effects of gemifloxacin compared to those of 11 other agents against Haemophilus influenzae and Moraxella catarrhalis
    • Davies TA, Kelly LM, Hoellman DB et al. Activities and postantibiotic effects of gemifloxacin compared to those of 11 other agents against Haemophilus influenzae and Moraxella catarrhalis. Antimicrob Agents Chemother 2000; 44: 633-9.
    • (2000) Antimicrob Agents Chemother , vol.44 , pp. 633-639
    • Davies, T.A.1    Kelly, L.M.2    Hoellman, D.B.3
  • 12
    • 0038172604 scopus 로고    scopus 로고
    • Detection of mutations in quinolone resistance-determining regions in levofloxacin and methicillin-resistant Staphylococcus aureus: effects of the mutations on fluoroquinolone MICs
    • Horii T, Suzuki Y, Monji A et al. Detection of mutations in quinolone resistance-determining regions in levofloxacin and methicillin-resistant Staphylococcus aureus: effects of the mutations on fluoroquinolone MICs. Diagn Microbiol Infect Dis 2003; 46: 139-45.
    • (2003) Diagn Microbiol Infect Dis , vol.46 , pp. 139-145
    • Horii, T.1    Suzuki, Y.2    Monji, A.3
  • 13
    • 0036095939 scopus 로고    scopus 로고
    • In vitro activities of novel nonfluorinated quinolones PGE 9262932 and PGE 9509924 against clinical isolates of Staphylococcus aureus and Streptococcus pneumoniae with defined mutations in DNA gyrase and topoisomerase IV
    • Jones ME, Critchley IA, Karlowsky JA et al. In vitro activities of novel nonfluorinated quinolones PGE 9262932 and PGE 9509924 against clinical isolates of Staphylococcus aureus and Streptococcus pneumoniae with defined mutations in DNA gyrase and topoisomerase IV. Antimicrob Agents Chemother 2002; 46: 1651-7.
    • (2002) Antimicrob Agents Chemother , vol.46 , pp. 1651-1657
    • Jones, M.E.1    Critchley, I.A.2    Karlowsky, J.A.3
  • 14
    • 34247101013 scopus 로고    scopus 로고
    • Fluoroquinolone resistance in Streptococcus pneumoniae: area under the concentration-time curve/MIC ratio and resistance development with gatifloxacin, gemifloxacin, levofloxacin, and moxifloxacin
    • LaPlante KL, Rybak MJ, Tsuji B et al. Fluoroquinolone resistance in Streptococcus pneumoniae: area under the concentration-time curve/MIC ratio and resistance development with gatifloxacin, gemifloxacin, levofloxacin, and moxifloxacin. Antimicrob Agents Chemother 2007; 51: 1315-20.
    • (2007) Antimicrob Agents Chemother , vol.51 , pp. 1315-1320
    • LaPlante, K.L.1    Rybak, M.J.2    Tsuji, B.3
  • 15
    • 0031728829 scopus 로고    scopus 로고
    • Alteration in the GyrA subunit of DNA gyrase and the ParC subunit of DNA topoisomerase IV in quinolone-resistant clinical isolates of Staphylococcus epidermidis
    • Li Z, Deguchi T, Yasuda M et al. Alteration in the GyrA subunit of DNA gyrase and the ParC subunit of DNA topoisomerase IV in quinolone-resistant clinical isolates of Staphylococcus epidermidis. Antimicrob Agents Chemother 1998; 42: 3293-5.
    • (1998) Antimicrob Agents Chemother , vol.42 , pp. 3293-3295
    • Li, Z.1    Deguchi, T.2    Yasuda, M.3
  • 16
    • 4344607734 scopus 로고    scopus 로고
    • Quinolone-resistant Haemophilus influenzae in a long-term-care facility: nucleotide sequence characterization of alterations in the genes encoding DNA gyrase and DNA topoisomerase IV
    • Li X, Mariano N, Rahal JJ et al. Quinolone-resistant Haemophilus influenzae in a long-term-care facility: nucleotide sequence characterization of alterations in the genes encoding DNA gyrase and DNA topoisomerase IV. Antimicrob Agents Chemother 2004; 48: 3570-2.
    • (2004) Antimicrob Agents Chemother , vol.48 , pp. 3570-3572
    • Li, X.1    Mariano, N.2    Rahal, J.J.3
  • 17
    • 12144287623 scopus 로고    scopus 로고
    • Laboratory detection of Haemophilus influenzae with decreased susceptibility to nalidixic acid, ciprofloxacin, levofloxacin, and moxifloxacin due to GyrA and ParC mutations
    • Perez-Vazquez M, Roman F, Aracil B et al. Laboratory detection of Haemophilus influenzae with decreased susceptibility to nalidixic acid, ciprofloxacin, levofloxacin, and moxifloxacin due to GyrA and ParC mutations. J Clin Microbiol 2004; 42: 1185-91.
    • (2004) J Clin Microbiol , vol.42 , pp. 1185-1191
    • Perez-Vazquez, M.1    Roman, F.2    Aracil, B.3
  • 18
    • 45249101344 scopus 로고    scopus 로고
    • Mutations in the quinolone resistance determining region in Staphylococcus epidermidis recovered from conjunctiva and their association with susceptibility to various fluoroquinolones
    • Yamada M, Yoshida J, Hatou S et al. Mutations in the quinolone resistance determining region in Staphylococcus epidermidis recovered from conjunctiva and their association with susceptibility to various fluoroquinolones. Br J Ophthalmol 2008; 92: 848-51.
    • (2008) Br J Ophthalmol , vol.92 , pp. 848-851
    • Yamada, M.1    Yoshida, J.2    Hatou, S.3
  • 19
    • 60649093308 scopus 로고    scopus 로고
    • Target specificity of the new fluoroquinolone besifloxacin in Streptococcus pneumoniae Staphylococcus aureus and Escherichia coli
    • Cambau E, Matrat S, Pan XS et al. Target specificity of the new fluoroquinolone besifloxacin in Streptococcus pneumoniae, Staphylococcus aureus and Escherichia coli. J Antimicrob Chemother 2009; 63: 443-50.
    • (2009) J Antimicrob Chemother , vol.63 , pp. 443-450
    • Cambau, E.1    Matrat, S.2    Pan, X.S.3
  • 20
    • 68549092580 scopus 로고    scopus 로고
    • Ocular pharmacokinetics of besifloxacin following topical administration to rabbits, monkeys, and humans
    • Proksch JW, Granvil CP, Mermet-Siou R et al. Ocular pharmacokinetics of besifloxacin following topical administration to rabbits, monkeys, and humans. J Ocul Pharmacol Ther 2009; 25: 335-44.
    • (2009) J Ocul Pharmacol Ther , vol.25 , pp. 335-344
    • Proksch, J.W.1    Granvil, C.P.2    Mermet-Siou, R.3
  • 21
    • 34250800221 scopus 로고    scopus 로고
    • Nonclinical pharmacodynamics, pharmacokinetics, and safety of BOL-303224-A, a novel fluoroquinolone antimicrobial agent for topical ophthalmic use
    • Ward KW, Lepage JF, Driot JY. Nonclinical pharmacodynamics, pharmacokinetics, and safety of BOL-303224-A, a novel fluoroquinolone antimicrobial agent for topical ophthalmic use. J Ocul Pharmacol Ther 2007; 23: 243-56.
    • (2007) J Ocul Pharmacol Ther , vol.23 , pp. 243-256
    • Ward, K.W.1    Lepage, J.F.2    Driot, J.Y.3
  • 22
    • 64849100973 scopus 로고    scopus 로고
    • Besifloxacin ophthalmic suspension 0.6% in patients with bacterial conjunctivitis: a multicenter, prospective, randomized, double-masked, vehicle-controlled 5-day efficacy and safety study
    • Karpecki P, DePaolis M, Hunter JA et al. Besifloxacin ophthalmic suspension 0.6% in patients with bacterial conjunctivitis: a multicenter, prospective, randomized, double-masked, vehicle-controlled, 5-day efficacy and safety study. Clin Ther 2009; 31: 514-26.
    • (2009) Clin Ther , vol.31 , pp. 514-526
    • Karpecki, P.1    DePaolis, M.2    Hunter, J.A.3
  • 23
    • 69349091130 scopus 로고    scopus 로고
    • Efficacy and safety of besifloxacin ophthalmic suspension 0.6% compared with moxifloxacin ophthalmic solution 0. 5% for treating bacterial conjunctivitis
    • McDonald MB, Protzko EE, Brunner LS et al. Efficacy and safety of besifloxacin ophthalmic suspension 0.6% compared with moxifloxacin ophthalmic solution 0.5% for treating bacterial conjunctivitis. Ophthalmology 2009; 116: 1615-23.
    • (2009) Ophthalmology , vol.116 , pp. 1615-1623
    • McDonald, M.B.1    Protzko, E.E.2    Brunner, L.S.3
  • 24
    • 67649400450 scopus 로고    scopus 로고
    • Phase III efficacy and safety study of besifloxacin ophthalmic suspension 0.6% in the treatment of bacterial conjunctivitis
    • Tepedino ME, Heller WH, Usner DW et al. Phase III efficacy and safety study of besifloxacin ophthalmic suspension 0.6% in the treatment of bacterial conjunctivitis. Curr Med Res Opin 2009; 25: 1159-69.
    • (2009) Curr Med Res Opin , vol.25 , pp. 1159-1169
    • Tepedino, M.E.1    Heller, W.H.2    Usner, D.W.3
  • 26
    • 3342984904 scopus 로고    scopus 로고
    • In vitro activities of mutant prevention concentration-targeted concentrations of fluoroquinolones against Staphylococcus aureus in a pharmacodynamic model
    • Allen GP, Kaatz GW, Rybak MJ. In vitro activities of mutant prevention concentration-targeted concentrations of fluoroquinolones against Staphylococcus aureus in a pharmacodynamic model. Int J Antimicrob Agents 2004; 24: 150-60.
    • (2004) Int J Antimicrob Agents , vol.24 , pp. 150-160
    • Allen, G.P.1    Kaatz, G.W.2    Rybak, M.J.3
  • 27
    • 3343024520 scopus 로고    scopus 로고
    • Comparison of minimal inhibitory and mutant prevention drug concentrations of 4 fluoroquinolones against clinical isolates of methicillin-susceptible and -resistant Staphylococcus aureus
    • Metzler K, Hansen GM, Hedlin P et al. Comparison of minimal inhibitory and mutant prevention drug concentrations of 4 fluoroquinolones against clinical isolates of methicillin-susceptible and -resistant Staphylococcus aureus. Int J Antimicrob Agents 2004; 24: 161-7.
    • (2004) Int J Antimicrob Agents , vol.24 , pp. 161-167
    • Metzler, K.1    Hansen, G.M.2    Hedlin, P.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.