Surface solid dispersion of glimepiride for enhancement of dissolution rate

International Journal of PharmTech Research

Volumn 1, Issue 3, 2009, Pages 822-831

  Kiran, T ^a   Shastri, Nalini ^a   Ramakrishna, Sistla ^b   MSadanandam, ^a  

^a Sri Venkateshwara College of Pharmacy   (India)

^b INDIAN INSTITUTE OF CHEMICAL TECHNOLOGY   (India)

Author keywords

Avicel PH 101; Croscarmellose; Crospovidone; Glimepiride; Potato starch; Pre gelatinized starch; Presence absence model; Sodium starch glycolate; Solvent deposition; Surface Solid Dispersion

Indexed keywords

CROSCARMELLOSE SODIUM; CROSPOVIDONE; DRUG CARRIER; GLIMEPIRIDE; STARCH; STARCH GLYCOLATE SODIUM;

ARTICLE; CONTROLLED STUDY; DIFFERENTIAL SCANNING CALORIMETRY; DISPERSION; DRUG GRANULATION; DRUG MIXTURE; DRUG SOLUBILITY; GAS CHROMATOGRAPHY; INFRARED SPECTROSCOPY; SCANNING ELECTRON MICROSCOPY; TABLET FORMULATION; X RAY POWDER DIFFRACTION;

EID: 77953445452     PISSN: None     EISSN: 09744304     Source Type: Journal    
DOI: None     Document Type: Article

References (19)

1. Yalkowsky, S.H., (1981). Techniques of Solubilization of drugs, vol 12, Marcel Dekker Inc., New York.
2. Serajuddin, A.T.M., (1999). Solid dispersion of poorly water soluble-soluble drugs: early promises, subsequent problems, and recent breakthroughs. J. Pharm. Sci., 88, 1058-1066.
3. Ford, J.L., (1986). The current status of solid dispersions. Pharm. Acta Helv., 53, 93-98.
4. Williams, A.C., Timmins, P., Lu, M., & Forbes, R.T., (2005). Disorder and dissolution enhancement: Deposition of ibuprofen on to insoluble polymers. Eur. J. Pharm. Sci., 26, 288-294.
5. Westerberg, M., Jonsson, B., & Nystrom, C., (1986). Physicochemical aspects of drug release. IV. The effect of carrier particle properties on the dissolution rate from ordered mixtures. Int. J. Pharm., 18, 23-31.
6. Yang, K.Y., Glemza, R., & Jarowski, C.I., (1979). Effects of amorphous silicon dioxides on drug dissolution. J. Pharm. Sci., 68, 560-565.
7. Barzegar-Jalali, M., Maleki, N., Garjani, A., Khandar, A.A., Haji-Hosseinloo, M., Jabbari, R., & Dastmalchi, S., (2002). Enhancement of dissolution rate and anti-infammatory effects of piroxicam using solvent deposition technique. Drug Dev. Ind. Pharm., 28(6), 681-686.
8. Charumanee, S., Okonoki, S., & Sirithunyalug, J., (2004), Improvement of dissolution rate of piroxicam by surface solid dispersions. CMU Journal, 3(2), 77-84.
9. Sharma, S., Sher, P., Badve, S., & Pawar, A.P., (2005). Adsorption of meloxicam on porous calcium silicate: Characterization and tablet formulation. AAPS PharmSciTech., 6(4), E618-E625.
10. Chowdary, K.P.R., & Rao, Sk. S., (2000). Investigation of dissolution enhancement of itraconazole by solid dispersion in superdisintegrants. Drug Dev. Ind. Pharm., 26(1), 1207-1211.
11. Giunchedi, P., Scalia, S., Maggi, L., & Conte, U., (1996). Ursodeoxycholic acid: improvement of dissolution behaviour and its HPLC determination. Int. J. Pharm., 130, 41-47.
12. Massimo, M.B., (2003). Glimepiride in type 2 diabetes mellitus: a review of the worldwide therapeutic experience. Clin. Ther. 25, 799-816.
13. Frick A., Möller, H., & Wirbitzki, E., (1998). Biopharmaceutical characterization of oral immediate release drug products. In vivo/in vitro comparison of phenoxy methyl penicillin potassium, glimepiride and levofloxacin. Eur. J. Pharm. Biopharm., 46, 305-311.
14. Ammar, H.O., Salama, H.A., Ghorab M., & Mahmoud, A.A., (2006). Formulation and biological evaluation of glimepiride-cyclodextrin-polymer systems, Int. J. Pharm., 309, 129-138
15. rd Pharmaceutical Powder X-ray Diffraction Symposium 2004, USA at http://www.icdd.com/ppxrd/03/reginfo/Abstract-ysrKrishnaiah.pdf.
16. Lewis, G.A., Mathieu, D., & Phan-Tan-Luu, R., (1991) Pharmaceutical Experimental design, vol no 92, Marcel Dekker Inc., New York, pg 28- 37.
17. Anderson, N.H., Johnston, D., & Vojvodic, P.R., (1990) Dissolution testing using continuous multicomponent UV analysis to correct for excipients interference, J. Pharm. Biomed. Anal., 8(10-12), 987-989.
18. Khan, K.A., (1975). The concept of dissolution efficiency. J.Pharm.Pharmacol., 27, 48-49.
19. Babu, P.S., Ramu, A., Sasidhar, R., & Vidyadhara, S., (2008). Enhancement of dissolution rate of glimepiride using new carriers. The Indian Pharmacist, 69(3), 65-68.