Flexible ligand recognition of peroxisome proliferator-activated receptor-γ (PPARγ)

Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 11, 2010, Pages 3344-3347

  Yamagishi, Kenji ^a   Yamamoto, Keiko ^b   Mochizuki, Yuji ^a   Nakano, Tatsuya ^c   Yamada, Sachiko ^a,d   Tokiwa, Hiroaki ^a  

^a RIKKYO UNIVERSITY   (Japan)

^b SHOWA PHARMACEUTICAL UNIVERSITY   (Japan)

^c NATIONAL INSTITUTE OF HEALTH SCIENCES   (Japan)

^d NIHON UNIVERSITY   (Japan)

Author keywords

Fragment molecular orbital; Hydrophobic residue; Ligand recognition; Peroxisome proliferator activated receptor ; PPAR

Indexed keywords

FARGLITAZAR; LIGAND; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA; ROSIGLITAZONE; THIAZOLIDINE DERIVATIVE;

ARTICLE; BINDING AFFINITY; DRUG STRUCTURE; LIGAND BINDING; PHARMACOPHORE;

LIGANDS; MODELS, MOLECULAR; PPAR GAMMA;

EID: 77953292378     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.04.031     Document Type: Article

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