Development of an automated synthesis system for preparation of glucuronides using a solid-phase extraction column loaded with microsomes

Chemical and Pharmaceutical Bulletin

Volumn 58, Issue 3, 2010, Pages 354-358

  Kashima, Yousuke ^a   Kitade, Takashi ^b   Kashima, Yuuko ^a   Okabayashi, Yoshito ^a  

^a SHIONOGI AND CO LTD   (Japan)

^b M and S Instruments Inc   (Japan)

Author keywords

Automated synthesis; Glucuronide; Microsome: Microsome immobilized solid phase extraction column

Indexed keywords

BETA CYCLODEXTRIN; DIPALMITOYLPHOSPHATIDYLCHOLINE; ESTRADIOL; GLUCURONIC ACID; GLUCURONIDE; GLUCURONOSYLTRANSFERASE; MEFENAMIC ACID; OCTADECYLSILICON DIOXIDE; PHOSPHOLIPID; SILICON DIOXIDE; UNCLASSIFIED DRUG; URIDINE DIPHOSPHATE;

ANIMAL TISSUE; AQUEOUS SOLUTION; ARTICLE; AUTOMATION; CATALYSIS; DRUG ISOLATION; DRUG SYNTHESIS; ELUTION; ENZYME ACTIVITY; GLUCURONIDATION; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; LIVER MICROSOME; NONHUMAN; SOLID PHASE EXTRACTION;

ANIMALS; DOGS; FEMALE; GLUCURONIDES; LIVER; MICROSOMES; MOLECULAR CONFORMATION; PHOSPHOLIPIDS; SILICON DIOXIDE; SOLID PHASE EXTRACTION; STEREOISOMERISM; SURFACE PROPERTIES;

EID: 77649253971     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.58.354     Document Type: Article

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