Fragment screening using surface plasmon resonance optical biosensor technology

Yakugaku Zasshi

Volumn 130, Issue 3, 2010, Pages 341-348

  Miura, Takaaki ^a  

^a CHUGAI PHARMACEUTICAL CO LTD   (Japan)

Author keywords

Fragment screening; Promiscuous binder; Surface plasmon resonance

Indexed keywords

BINDING ASSAY; BINDING COMPETITION; FRAGMENT SCREENING; MOLECULAR INTERACTION; NUCLEAR MAGNETIC RESONANCE; OPTICAL BIOSENSOR; PRACTICE GUIDELINE; REVIEW; SCREENING; STOICHIOMETRY; SURFACE PLASMON RESONANCE; X RAY CRYSTALLOGRAPHY;

BIOSENSING TECHNIQUES; DRUG DISCOVERY; DRUG EVALUATION, PRECLINICAL; PROTEIN BINDING; SURFACE PLASMON RESONANCE;

EID: 77649253758     PISSN: 00316903     EISSN: 13475231     Source Type: Journal    
DOI: 10.1248/yakushi.130.341     Document Type: Review

References (10)

1. Kawada S., "Seitaibusshitsu Sougo Sayou no Real Time Kaiseki Jikken Hou," ed. by Nagata K., Handa H., Springer-Verlag, Tokyo, 1998, pp13-26.
2. Day Y. S., Baird C. L.,Rich R. L., Myszka D. G., Protein Sci., 11, 1017-1025 (2002).
3. Frostell-Karlsson A., Remaeus A., Roos H., Andersson K., Borg P., Hämäläinen M., Karlsson R., J. Med. Chem., 43, 1986-1992 (2000).
4. Rich R. L., Myszka D. G., J. Mol. Recognit., 21, 355-400 (2008).
5. Hajduk P. J., Greer J., Nat. Rev. Drug. Discov., 6, 211-219 (2007).
6. Perspicace S., Banner D., Benz J., Muller F., Schlatter D., Huber W., J. Biomol. Screen., 14, 337-349 (2009).
7. Nordstroäm H., Gossas T., Hämäläinen M. D., Källbrad P., Nystroäm S., Wallberg H., Danielson U. H., J. Med. Chem., 51, 3449-3459 (2008).
8. Hämäläinen M. D., Zhukov A., Ivarsson M., Fex T., Gottfries J., Karlsson R., Björsne M., J. Biomol. Screen., 13, 202-209 (2008).
9. Hajduk P. J., J. Med. Chem., 49, 6972-6976 (2006).
10. Giannetti A. M., Koch B. D., Browner M. F., J. Med. Chem., 51, 574-580 (2008).