Synthesis and functionalization of the 3-(1, 3, 4-oxadiazol-2-yl)-1H- indoles

Chemistry of Heterocyclic Compounds

Volumn 45, Issue 10, 2009, Pages 1270-1275

  Alyab'ev, S B ^a   Kravchenko, D V ^a   Ivashchenko, A V ^a  

^a Chemical Diversity Research Institute   (Russian Federation)

Author keywords

3 (1, 3, 4 oxadiazol 2 yl) 1H indoles; 3 (1, 3, 4 oxadiazol 2 yl) 1H indol 1 yl acetic acids; Amide library; Intramolecular cyclization; Orthoesters

Indexed keywords

EID: 77249117282     PISSN: 00093122     EISSN: 15738353     Source Type: Journal    
DOI: 10.1007/s10593-010-0418-0     Document Type: Article

References (13)

1. J. S. Biradar and S. Y. Manjunath, Indian J. Chem., 43B, 141 (2004).
2. C. J. Swain, R. Baker, C. Kneen, J. Moseley, and J. Saunders, J. Med. Chem., 34, 140 (1991).
3. I. Nicolaou and V. J. Demopoulos, J. Med. Chem., 46, 417 (2003).
4. D. E. Mais, F. Mohamadi, G. P. Dube, W. L. Kurtz, and K. A. Brune, Eur. J. Med. Chem., 26, 821 (1991).
5. A. M. Korolev, E. I. Lazhko, and M. N. Preobrazhenskaya, Khim.-Farm. Zh., 25, No. 11, 42 (1991).
6. P. E. Cross, R. P. Dickinson, M. J. Parry, and M. J. Randall, J. Med. Chem., 29, 342 (1986).
7. V. I. Kelarev and G. A. Shvekhgeimer, Khim. Geterotsikl. Soedin., 343 (1982).
8. V. I. Kelarev and G. A. Shvekhgeimer Chem. Heterocycl. Comp., 18, 258 (1982).
9. V. A. Monge, M. M. Rabbani, and E. Fernandez-Alvarez, Bol. Soc. Quim. Peru, 49, No. 2, 120 (1983).
10. R. A. Karakhanov, V. I. Kelarev, A. S. Kokosova, I. M. Nasyrov, and Z. Ya. Kuznetsova (Kusnetsova); in: Proc. Fifth Conf. Appl. Chem. Unit. Oper. and Process, Balatonfured, September 3-7, 1989: 405th Event Eur. Fed. Chem., vol. 2, Budapest (1989); p. 446.
11. A. H. Farghaly Abdel-Rahman, J. Chin. Chem. Soc., 51, No. 1, 147 (2004).
12. C. J. Swain, R. Baker, C. Kneen, J. Moseley, and J. Saunders, J. Med. Chem., 34, 140 (1991).
13. O. Ottoni, R. Cruz, and R. Alves, Tetrahedron, 54, 13915 (1998).