Synthesis and anti-inflammatory activity of some novel biphenyl-4- carboxylic acid 5-(arylidene)-2-(aryl)-4-oxothiazolidin-3-yl amides

Acta Poloniae Pharmaceutica - Drug Research

Volumn 67, Issue 1, 2010, Pages 63-67

  Deep, Aakash ^a   Jain, Sandeep ^b   Sharma, Prabodh Chander ^c  

^a GVM College of Pharmacy   (India)

^b GURU JAMBHESHWAR UNIVERSITY OF SCIENCE AND TECHNOLOGY   (India)

^c KURUKSHETRA UNIVERSITY   (India)

Author keywords

4 thiazolidinone; Anti inflammatory activity; Biphenyl; Synthesis

Indexed keywords

ACETIC ACID; ALDEHYDE; AMIDE; ANTIINFLAMMATORY AGENT; BIPHENYL 4 CARBOXYLIC ACID (5 BENZYLIDENE 4 OXO 2 PHENYLTHIAZOLIDIN 3YL)AMIDE; BIPHENYL 4 CARBOXYLIC ACID [2 (3 BROMOPHENYL) 5 (3 NITROBENZYLIDENE) 4 OXO THIAZOLIDIN 3 YL]AMIDE; BIPHENYL 4 CARBOXYLIC ACID [2 (3 BROMOPHENYL) 5 (4 CHLOROBENZYLIDENE) 4 OXO THIAZOLIDIN 3 YL]AMIDE; BIPHENYL 4 CARBOXYLIC ACID [2 (3 BROMOPHENYL) 5 (4 METHOXYBENZYLIDENE) 4 OXO THIAZOLIDIN 3 YL]AMIDE; BIPHENYL 4 CARBOXYLIC ACID [5 (3 BROMOBENZYLIDENE) 2 (3 BROMOPHENYL) 4 OXO THIAZOLIDIN 3 YL]AMIDE; BIPHENYL 4 CARBOXYLIC ACID [5 (3 BROMOBENZYLINE) 4 OXO 2 PHENYLTHIAZOLIDIN 3YL)AMIDE; BIPHENYL 4 CARBOXYLIC ACID [5 (3 NITROBENZYLIDENE) 4 OXO 2 PHENYLTHIAZOLIDIN 3YL)AMIDE; BIPHENYL 4 CARBOXYLIC ACID [5 (4 CHLOROBENZYLINE) 4 OXO 2 PHENYLTHIAZOLIDIN 3YL)AMIDE; BIPHENYL 4 CARBOXYLIC ACID [5 (4 FLUOROPHENYL) 5 (3 NITROBENZYLIDENE) 4 OXO THIAZOLIDIN 3 YL]AMIDE; BIPHENYL 4 CARBOXYLIC ACID [5 (4 METHOXYBENZYLINE) 4 OXO 2 PHENYLTHIAZOLIDIN 3YL)AMIDE; BIPHENYL 4 CARBOXYLIC ACID [5 BENZYLIDENE 2 (3 BROMOPHENYL) 4 OXOTHIAZOLIDIN 3YL)AMIDE; BIPHENYL 4 CARBOXYLIC ACID [5 BENZYLIDENE 2 (4 FLUOROPHENYL) 4 OXO THIAZOLIDIN 3 YL]AMIDE; CARRAGEENAN; HYDRAZONE DERIVATIVE; THIOGLYCOLIC ACID; UNCLASSIFIED DRUG; ZINC CHLORIDE;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIINFLAMMATORY ACTIVITY; ARTICLE; CATALYSIS; CHEMICAL REACTION; CONTROLLED STUDY; DRUG ACTIVITY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; INFRARED RADIATION; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; RAT;

ANIMALS; ANTI-INFLAMMATORY AGENTS; CARRAGEENAN; DISEASE MODELS, ANIMAL; FEMALE; INFLAMMATION; MAGNETIC RESONANCE SPECTROSCOPY; MALE; MOLECULAR STRUCTURE; RATS; SPECTROSCOPY, FOURIER TRANSFORM INFRARED; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 76749144263     PISSN: 00016837     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (14)

1. Bruke A., Smyth E. M., FitzGerald G. A.: in Goodman and Gilman's The Pharmacological Basis of Therapeutics, Bruton L. L. Ed., p. 671-716, McGraw Hill Co., New York 2006.
2. Samir B., Wesam K., Ahmed A. F.: Eur. J. Med. Chem. 42, 948 (2007).
3. Shah T. J., Desai V.A.: ARKIVOC (xiv) 218 (2007).
4. Vicini P., Geronikaki A., Anastasia K., Incerti M., Zani F.: Bioorg. Med. Chem., 14, 3859 (2006).
5. Sharma R., Nagda D. P., Talesara G. L.: ARKIVOC (i), 1, (2006).
6. Handan A., Oznur A., Seher B., Gulten O., Melten U., Dilek S.: Turk. J. Chem. 29, 425 (2005).
7. Knutsen L.J.S., Hobbs C.J., Earnshaw C.G., et al.: Bioorg. Med. Chem. Lett. 17, 662, (2007).
8. Ottana R., Maccari R., Barreca M. L., et al.: Bioorg. Med. Chem. 13, 4243 (2005).
9. Goel B., Ram T., Tyagi R., Bansal E., Kumar A., Mukherjee D., Sinha J.M.: Eur. J. Med. Chem. 34, 265 (1999).
10. Balzarini J., Orzeszko B., Maurin J.K., Orzeszko A.: Eur. J. Med. Chem. 42, 993 (2007).
11. Mujeebur Rahman V.P., Mukhtar S., Ansari W.H.: Eur. J. Med. Chem. 40, 173 (2005).
12. Gursoy A., Terzioglu N.: Turk. J. Chem. 29, 247 (2005).
13. Andres C. J., Bronson J. J., D'Andrea S. V., Deshpande M. S., et al.: Bioorg. Med. Chem. Lett. 10, 715 (2000).
14. Winter C. A., Fisley E. A. Nuss G. W.: Proc. Soc. Exp. Biol. Med. 111, 544 (1962).