The first asymmetric synthesis of a 4-aryl-substituted 5-carboxy-3,4-dihydropyridin-2-one derivative

Tetrahedron Letters

Volumn 51, Issue 12, 2010, Pages 1554-1557

  Huang, Xiaojun ^a   Zhu, Jiang ^a   Broadbent, Scott ^a  

^a ROCHE BIOSCIENCE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 (4 FLUOROPHENYL) 1,4,5,6 TETRAHYDRO 6 OXO 3 PYRIDINECARBOXYLIC ACID; DIHYDROPYRIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CATALYSIS; CATALYST; CHEMICAL ANALYSIS; CHEMICAL MODIFICATION; CHEMICAL REACTION; CHEMICAL STRUCTURE; CYCLIZATION; DRUG SYNTHESIS;

EID: 76449093041     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2010.01.049     Document Type: Article

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15. 3: C, 62.65; H, 4.85; N, 5.62. Found: C, 62.78; H, 4.77; N, 5.64.
16. 3: C, 61.28; H, 4.29; N, 5.95. Found: C, 61.05; H, 4.21; N, 6.03.