A route to the γ-secretase inhibitor [2,3,4-3H]BMS299897 via an α-phenylselenide derivative

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 53, Issue 1, 2010, Pages 44-46

  Malmquist, Jonas ^a   Bernlind, Alexandra ^a   Ström, Peter ^a  

^a ASTRAZENECA R AND D   (Sweden)

Author keywords

Secretase; Wilkinson's catalyst

Indexed keywords

BASIC HYDROLYSIS; DOUBLE BONDS; METHYL ESTERS; SECRETASES; SELENIDES; SPECIFIC ACTIVITY; WILKINSON'S CATALYST; Γ-SECRETASE INHIBITORS;

CATALYSTS;

4 [2 [1 [4 CHLORO N (2,5 DIFLUOROPHENYL)PHENYLSULFONAMIDO]ETHYL] 5 FLUOROPHENYL]BUTANOIC ACID H 3; ALIPHATIC COMPOUND; BMS 299897; RADIOPHARMACEUTICAL AGENT; SELENIDE; TRITIUM; UNCLASSIFIED DRUG;

ARTICLE; AUTORADIOGRAPHY; CHEMICAL BOND; DRUG SYNTHESIS; HALOGENATION; REDUCTION;

EID: 76149110453     PISSN: 03624803     EISSN: 10991344     Source Type: Journal    
DOI: 10.1002/jlcr.1719     Document Type: Article

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