The effects of some permeability enhancers on the percutaneous absorption of lidocaine

Pakistan Journal of Pharmaceutical Sciences

Volumn 23, Issue 1, 2010, Pages 83-88

  Mohammadi Samani, Soliman ^a   Jamshidzadeh, Akram ^a   Montaseri, Hashem ^a   Rangbar Zahedani, Mojgan ^a   Kianrad, Roshan ^a  

^a SHIRAZ UNIVERSITY OF MEDICAL SCIENCES   (Iran)

Author keywords

DMSO; Lidocaine; Permeability enhancer; Surfactants; Terpene

Indexed keywords

CYCLOHEXANOL; DIMETHYL SULFOXIDE; LIDOCAINE; POLYSORBATE 20; POLYSORBATE 80; TERPENE DERIVATIVE; TERPIN HYDRATE;

ANIMAL TISSUE; ANTINOCICEPTION; ARTICLE; CONTROLLED STUDY; DRUG ABSORPTION; DRUG EFFECT; DRUG FORMULATION; DRUG PENETRATION; GUINEA PIG; NONHUMAN; SKIN ABSORPTION; SKIN PENETRATION;

ADMINISTRATION, CUTANEOUS; ANESTHETICS, LOCAL; ANIMALS; CYCLOHEXANOLS; CYCLOHEXENES; DIMETHYL SULFOXIDE; DRUG INTERACTIONS; LIDOCAINE; MONOTERPENES; PAIN; PERMEABILITY; POLYSORBATES; RATS; SKIN; SKIN ABSORPTION;

EID: 75649137320     PISSN: 1011601X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (21)

1. Barry BW (1987). Mode of action of penetration enhancers in human skin. Journal of Controlled Release, 6(1): 85-97.
2. Barry BW (2001a). Is transdermal drug delivery research still important today? Drug Discov. Today, 6(19): 967-971.
3. Barry BW (2001b). Novel mechanisms and devices to enable successful transdermal drug delivery. Eur. J. Pharm. Sci., 14(2): 101-114.
4. Brechner VL, Cohen DD and Pretsky I (1967). Dermal anesthesia by the topical application of tetracaine base dissolved in dimethyl sulfoxide. Ann. NY Acad. Sci., 141(1): 524-531.
5. Cornwella PA and Barry BW (1993). The routes of penetration of ions and 5-fluorouracil across human skin and the mechanisms of action of terpene skin penetration enhancers. International Journal of Pharmaceutics, 94(1-3): 189-194.
6. Embery G and Dugard PH (1971). The isolation of dimethyl sulfoxide soluble components from human epidermal preparations: A possible mechanism of action of dimethyl sulfoxide in effecting percutaneous migration phenomena. J. Invest. Dermatol., 57(5): 308-311.
7. Evrard D, Touitou E, Kolusheva S, Fishov Y and Jelinek R (2001). A new colorimetric assay for studying and rapid screening of membrane penetration enhancers. Pharm. Res., 18(7): 943-949.
8. Gajraj NM, Pennant JH and Watcha MF (1994). Eutectic mixture of local anesthetics (EMLA) cream. Anesth. Analg., 78(3): 574-583.
9. Jakobson B and Nilsson A (1985). Methemoglobinemia associated with a prilocaine-lidocaine cream and trimetoprim-sulphamethoxazole. A case report. Acta Anaesthesiol. Scand., 29(4): 453-455.
10. Juhlin L and Evers H (1990). EMLA: A new topical anesthetic. Adv. Dermatol., 5: 75-91; Discussion 92.
11. Kang L, Jun HW and Mani N (2001). Preparation and characterization of two-phase melt systems of lidocaine. Int. J. Pharm., 222(1): 35-44.
12. Kang L, Jun HW and McCall JW (2000). Physicochemical studies of lidocaine-menthol binary systems for enhanced membrane transport. Int. J. Pharm., 206(1-2): 35-42.
13. Karande P, Jain A and Mitragotri S (2006). Insights into synergistic interactions in binary mixtures of chemical permeation enhancers for transdermal drug delivery. J. Control Release, 115(1): 85-93.
14. Lener EV, Bucalo BD, Kist DA and Moy RL (1997). Topical anesthetic agents in dermatologic surgery. A review. Dermatol. Surg., 23(8): 673-683.
15. Lim PF, Liu XY, Kang L, Ho PC, Chan YW and Chan SY (2006). Limonene GP1/PG organogel as a vehicle in transdermal delivery of haloperidol. Int. J. Pharm., 311(1-2): 157-164.
16. Liu H, Li S, Wang Y, Yao H and Zhang Y (2006). Effect of vehicles and enhancers on the topical delivery of cyclosporin A. Int. J. Pharm., 311(1-2): 182-186.
17. Lopez A, Llinares F, Cortell C and Herraez M (2000). Comparative enhancer effects of Span20 with Tween20 and Azone on the in vitro percutaneous penetration of compounds with different lipophilicities. Int. J. Pharm., 202(1-2): 133-140.
18. Nokhodchi A, Sharabiani K, Rashidi MR and Ghafourian T (2007). The effect of terpene concentrations on the skin penetration of diclofenac sodium. Int. J. Pharm., 335(1-2): 97-105.
19. Nokhodchi A, Shokri J, Dashbolaghi A, Hassan-Zadeh D, Ghafourian T and Barzegar-Jalali M (2003). The enhancement effect of surfactants on the penetration of lorazepam through rat skin. Int. J. Pharm., 250(2): 359-369.
20. Nortier YL, van de Haven JA, Koks CH and Beijnen JH (1995). Preparation and stability testing of a hydrogel for topical analgesia. Pharm. World Sci., 17(6): 214-217.
21. Owen JA, Tasker RA and Nakatsu K (1984). A simple, less stressful rat restrainer. Experientia, 40(3): 306-308.