Fluorine-18 labeled galactosyl-neoglycoalbumin for imaging the hepatic asialoglycoprotein receptor

Bioorganic and Medicinal Chemistry

Volumn 17, Issue 21, 2009, Pages 7510-7516

  Yang, Wenjiang ^a   Mou, Tiantian ^a   Peng, Cheng ^b   Wu, Zhanhong ^c   Zhang, Xianzhong ^a   Li, Fang ^c   Ma, Yunchuan ^b  

^a BEIJING NORMAL UNIVERSITY   (China)

^b CAPITAL MEDICAL UNIVERSITY   (China)

^c PEKING UNION MEDICAL COLLEGE HOSPITAL   (China)

Author keywords

Asialoglycoprotein receptor; NGA; Pet imaging

Indexed keywords

ASIALOGLYCOPROTEIN RECEPTOR; BLOCKING AGENT; CRYPTAND 2.2.2; FLUORINE 18; GALACTOSYLNEOGLYCOALBUMIN TC 99M; RADIOISOTOPE; TRACER; ALBUMINOID; FLUORINE; GALACTOSYL NEOGLYCOALBUMIN; GALACTOSYL-NEOGLYCOALBUMIN; RADIOPHARMACEUTICAL AGENT;

ARTICLE; COLUMN CHROMATOGRAPHY; CONJUGATION; CONTROLLED STUDY; DRUG BINDING; DRUG DISTRIBUTION; DRUG EFFICACY; DRUG PURIFICATION; DRUG STABILITY; EX VIVO STUDY; FEMALE; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IMAGE QUALITY; IN VIVO STUDY; ISOTOPE LABELING; LIVER FUNCTION; MOUSE; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; QUANTITATIVE ANALYSIS; RADIOASSAY; RADIOCHEMISTRY; RAT; REACTION TIME; SCINTISCANNING; ANIMAL; CHEMISTRY; LIVER; METABOLISM; SYNTHESIS; TISSUE DISTRIBUTION;

MAMMALIA; MUS; RATTUS;

ALBUMINS; ANIMALS; ASIALOGLYCOPROTEIN RECEPTOR; FLUORINE RADIOISOTOPES; LIVER; MICE; POSITRON-EMISSION TOMOGRAPHY; RADIOPHARMACEUTICALS; RATS; TISSUE DISTRIBUTION;

EID: 73949093807     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2009.09.017     Document Type: Article

References (20)

1. Kokudo, N.; Vera, D. R.; Makuuchi, M. Nucl. Med. Biol. 2003, 30, 845.
2. Stadalnik, R. C.; Vera. D. R. Nucl. Med. Biol. 2001, 28, 499.
3. Vera, D. R.; Stadalnik, R. C.; Krohn, K. A. J. Nucl. Med. 1985, 26, 1157.
4. Kubota, Y.; Kojima, M.; Hazama, H.; Kawa, S.; Nakazawa, M.; Nishiyama, Y.; Nakagawa, S.; Murase. T.; Okuno, H.; Naitoh, Y., et aljpnj. Nucl. Med. 1986, 23, 899.
5. Torizuka, K.; Ha-Kawa. S. K.; Ikekubo, K.; Suga, Y.; Tanaka, Y.; Hino, M.; Ito, H.; Yamamoto, K.: Yonekura, Y. Jpn. J. Nucl. Med. 1991, 28, 1321.
6. Wakisaka, K.; Arano, Y.; Uezono, T.; Akizawa, H.; Ono, M.; Kawai, K.; Ohomomo, Y.; Nakayama, M.; Saji, H. J. Med. Chem. 1997, 40, 2643.
7. Arano, Y.; Mukai, T.; Akizawa, H.; Uezono. T.; Motonarl, H.; Wakisaka, K.; Kairiyama, C.; Yokoyama, A. Nucl. Med. Biol. 1995, 22, 555.
8. Vera, D. R. J. Nucl. Med. 1992, 33, 1160.
9. Guhlke, S.; Coenen, H. H.; Stöcklin, G. Appl. Radiat. Isot. 1994, 45, 715.
10. Zhang. X.; Cai, W.; Cao. F.; Schreibmann, E.; Wu. Y.; Wu, J. C.; Xing, L.; Chen, X. J. Nucl. Med. 2006, 47, 492.
11. Zhang, X.; Xiong, Z.; Wu, Y.; Cai, W.; Tseng, J. R.; Gambhir, S. S.; Chen, X. J. Nucl. Med. 2006, 47, 113.
12. DuBois, M.; Gilles, K. A.; Hamilton, J. K.; Rebers, P. A; Smith, F. Anal. Chem. 1956, 28, 350.
13. Ametamey, S. M.; Honer, M.; Schubiger, P. A. Chem. Rev. 2008, 108, 1501.
14. Gore, S.: Morris, A. I.: Gilmore, I. T.; Maltby, P. J.; Thornback, J. R.; Billington, D. J. Nucl. Med. 1991, 32, 506.
15. Duncan, J. R.; Welch, M. J. J. Nucl. Med. 1993, 34, 1728.
16. Arano, Y.; Mukai, T.; Uezono, T.; Wakisaka, K.; Motonari, H.; Akizawa, H.; Taoka, Y.; Yokoyama, A. J. Nucl. Med. 1994, 35, 890.
17. Ono, M.; Arano, Y.; Uehara, T.; Fujioka, Y.; Ogawa, K.; Namba, S.; Mukai, T.; Nakayama, M.; Saji. H. Bioconjugate Chem. 1999, 10, 386.
18. Hwang, E.-. H.; Taki, J.; Shuke, N.; Nakajima, K.; Kinuya, S.; Konishi, S.; Michigishi, T.; Aburano, T.; Tonami, N. J. Nucl. Med. 1999, 40, 1644.
19. Sugai, Y.; Komatani, A.; Hosoya. T.; Yamaguchi, K. J. Nucl. Med. 2000, 41, 421.
20. Shuke, N.; Okizaki, A.; Kino, S.; Sato. J.; Ishikawa, Y.; Zhao, C.; Kinuya, S.; Watanabe, N.; Yokoyama, K.; Aburano, T. J. Nucl. Med. 2003, 44, 475.