Anti-oxidant and anti-bacterial activities of novel N′-arylmethylidene-2-(3, 4-dimethyl-5, 5-dioxidopyrazolo[4,3-c][1,2]benzothiazin-2(4H)-yl) acetohydrazides

European Journal of Medicinal Chemistry

Volumn 45, Issue 2, 2010, Pages 698-704

  Ahmad, Matloob ^a,b   Siddiqui, Hamid Latif ^b   Zia ur Rehman, Muhammad ^a   Parvez, Masood ^c  

^a APPLIED CHEMISTRY RESEARCH CENTRE   (Pakistan)

^b UNIVERSITY OF THE PUNJAB   (Pakistan)

^c UNIVERSITY OF CALGARY   (Canada)

Author keywords

1,2 Benzothiazine 1,1 dioxides; Anti bacterial activity; Anti oxidant activity; Pyrazolo 4,3 c 1,2 benzothiazine 5,5 dioxide

Indexed keywords

2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL] N' (PHENYLMETHYLIDEN)ACETOHYDRAZIDE; 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL] N' (PYRIDIN 2 YLMETHYLIDEN)ACETOHYDRAZIDE; 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL] N' (PYRIDIN 3 YLMETHYLIDEN)ACETOHYDRAZIDE; 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL] N' (THIOPHEN 2 YLMETHYLIDEN)ACETOHYDRAZIDE; 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL] N' (THIOPHEN 3 YLMETHYLIDEN)ACETOHYDRAZIDE; 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL] N' [(2 NITROPHENYL)METHYLIDEN]ACETOHYDRAZIDE; 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL] N' [(3 NITROPHENYL)METHYLIDEN]ACETOHYDRAZIDE; 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL] N' [(4 NITROPHENYL)METHYLIDEN]ACETOHYDRAZIDE; [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL] N [(4 FLUOROPHENYL)METHYLIDEN]ACETOHYDRAZIDE; ACETOHYDRAZIDE; ALDEHYDE; ANTIINFECTIVE AGENT; ANTIOXIDANT; CHLOROACETIC ACID; HYDRAZINE; N [(3,4 DICHLOROPHENYL)METHYLIDENE] 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL]ACETOHYDRAZIDE; N' [(2 CHLOROPHENYL)METHYLIDENE] 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL]ACETOHYDRAZIDE; N' [(2,4 DICHLOROPHENYL)METHYLIDENE] 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL]ACETOHYDRAZIDE; N' [(2,4 DIHYDROXYPHENYL)METHYLIDENE] 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL]ACETOHYDRAZIDE; N' [(2,4 DIMETHOXYPHENYL)METHYLIDENE] 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL]ACETOHYDRAZIDE; N' [(3 ETHOXY 4 HYDROXY)METHYLIDENE] 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL]ACETOHYDRAZIDE; N' [(3 METHOXYPHENYL)METHYLIDENE] 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL]ACETOHYDRAZIDE; N' [(4 CHLOROPHENYL)METHYLIDENE] 2 [3,4 DIMETHYL 5,5 DIOXIDOPYRAZOLO[4,3 C][1,2]BENZOTHIAZIN 1(4H) YL]ACETOHYDRAZIDE; SACCHARIN; UNCLASSIFIED DRUG;

ALKYLATION; ANTIBACTERIAL ACTIVITY; ANTIOXIDANT ACTIVITY; ARTICLE; BACILLUS SUBTILIS; CHEMICAL REACTION; CONTROLLED STUDY; CYCLIZATION; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; METHYLATION; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; POLYMERIZATION; REACTION TIME; RING OPENING; STEREOCHEMISTRY; ULTRASOUND;

ANTI-BACTERIAL AGENTS; ANTIOXIDANTS; BACTERIA; FREE RADICALS; HUMANS; MICROBIAL SENSITIVITY TESTS; STEREOISOMERISM; THIAZINES;

EID: 73549117438     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2009.11.016     Document Type: Article

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