Synthesis, reactivity and biological evaluation of novel halogenated tripentones

Bioorganic and Medicinal Chemistry

Volumn 17, Issue 22, 2009, Pages 7783-7788

  Perri, Vittoria ^a   Rochais, Christophe ^a   Cresteil, Thierry ^b   Dallemagne, Patrick ^a   Rault, Sylvain ^a  

^a CENTRE D ETUDES ET DE RECHERCHE SUR LE MÉDICAMENT DE NORMANDIE   (France)

^b INSTITUT DE CHIMIE DES SUBSTANCES NATURELLES   (France)

Author keywords

Fused ring systems; Metallo catalysed cross coupling; Tripentones

Indexed keywords

ANTINEOPLASTIC AGENT; PYRROLIZINE DERIVATIVE; TRIPENTONE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; CROSS COUPLING REACTION; DRUG ACTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; HALOGENATION; HUMAN; HUMAN CELL;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CROSS-LINKING REAGENTS; DRUG EVALUATION, PRECLINICAL; HUMANS; HYDROCARBONS, HALOGENATED; PYRROLIZIDINE ALKALOIDS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 71749120415     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2009.09.027     Document Type: Article

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