Synthesis of functionalized amino acid derivatives as new pharmacophores for designing anticancer agents

Journal of Enzyme Inhibition and Medicinal Chemistry

Volumn 24, Issue 3, 2009, Pages 763-770

  Kumar, Vivek ^a   Mudgal, Mukesh M ^a   Rani, Nidhi ^a   Jha, Amrita ^a   Jaggi, Manu ^a   Singh, Anu T ^a   Sanna, Vinod K ^a   Singh, Pratibha ^a   Sharma, Pramod K ^b   Irchhaiya, Raghuveer ^b   Burman, Anand C ^a  

^a DABUR RESEARCH FOUNDATION   (India)

^b BUNDELKHAND UNIVERSITY   (India)

Author keywords

Anticancer; Carboxamide; Functionalized amino acid

Indexed keywords

1 N (3' CHLORO 4' FLUORO)PHENYL 3 AMINO 2 HYDROXY 3 PHENYLPROPANE 1 CARBOXAMIDE; 1 N (4' CYANO)PHENYL 3 AMINO 2 HYDROXY 3 PHENYLPROPANE 1 CARBOXAMIDE; 1 N (4' FLUORO)PHENYL 3 AMINO 2 HYDROXY 3 PHENYLPROPANE 1 CARBOXAMIDE; 1 N (4' METHOXY)PHENYL 3 AMINO 2 HYDROXY 3 PHENYLPROPANE 1 CARBOXAMIDE; 1 N CYCLOHEXYL 3 AMINO 2 HYDROXY 3 PHENYLPROPANE 1 CARBOXAMIDE; 1 N CYCLOPENTYL 3 AMINO 2 HYDROXY 3 PHENYLPROPANE 1 CARBOXAMIDE; 1 N CYCLOPROPYL 3 AMINO 2 HYDROXY 3 PHENYLPROPANE 1 CARBOXAMIDE; 1 N ISOPROPYL 3 AMINO 2 HYDROXY 3 PHENYLPROPANE 1 CARBOXAMIDE; 1 N PHENYL 3 AMINO 2 HYDROXY 3 PHENYLPROPANE 1 CARBOXAMIDE; 5 N (3' CHLORO 4' FLUORO)PHENYL 3 N' TERT BUTOXYCARBONYL2,2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N (4' CYANO)PHENYL 3 N' TERT BUTOXYCARBONYL 2,2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N (4' FLUORO)PHENYL 3 N' TERT BUTOXYCARBONYL 2,2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N (4' METHOXY)PHENYL 3 N' TERT BUTOXYCARBONYL 2,2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N 2' PYRIDINE 3 N' TERT BUTOXYCARBONYL 2, 2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N 2' THIAZOLE 3 N' TERT BUTOXYCARBONYL 2, 2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N 3' PYRIDINE 3 N' TERT BUTOXYCARBONYL 2, 2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N 4' PYRIDINE 3 N' TERT BUTOXYCARBONYL 2, 2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N BENZYL 3 N' TERT BUTOXYCARBONYL 2,2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N CYCLOHEXYL 3 N' TERT BUTOXYCARBONYL 2,2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N CYCLOPENTYL 3 N' TERT BUTOXYCARBONYL 2,2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N CYCLOPROPYL 3 N' TERT BUTOXYCARBONYL 2,2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N ISOPROPYL 3 N' TERT BUTOXYCARBONYL 2,2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N MORPHOLINE 3 N' TERT BUTOXYCARBONYL 2, 2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N PHENYL 3 N' TERT BUTOXYCARBONYL 2,2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N PIPERIDINE 3 N' TERT BUTOXYCARBONYL 2, 2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; 5 N PYRROLODINE 3 N' TERT BUTOXYCARBONYL 2, 2 DIMETHYL 4 PHENYL OXAZOLIDINE 5 CARBOXAMIDE; AMIDE; AMINO ACID DERIVATIVE; ANTINEOPLASTIC AGENT; UNCLASSIFIED DRUG; UNINDEXED DRUG; AMINO ACID;

ANIMAL CELL; ARTICLE; CANCER CELL CULTURE; CYTOTOXICITY; DRUG SYNTHESIS; FEMALE; HUMAN; HUMAN CELL; IC 50; IN VITRO STUDY; MOUSE; MOUTH CANCER; NONHUMAN; OVARY CANCER; PHARMACOPHORE; PRIORITY JOURNAL; CELL LINE; CHEMISTRY; CYTOLOGY; DRUG DESIGN; DRUG EFFECTS; DRUG SCREENING; FIBROBLAST; IC50; MOUTH TUMOR; OVARY TUMOR; PATHOLOGY; SYNTHESIS; TUMOR CELL LINE;

AMIDES; AMINO ACIDS; ANTINEOPLASTIC AGENTS; CELL LINE; CELL LINE, TUMOR; DRUG DESIGN; DRUG SCREENING ASSAYS, ANTITUMOR; FEMALE; FIBROBLASTS; HUMANS; INHIBITORY CONCENTRATION 50; MOUTH NEOPLASMS; OVARIAN NEOPLASMS;

EID: 70749159280     PISSN: 14756366     EISSN: 14756374     Source Type: Journal    
DOI: 10.1080/14756360802362975     Document Type: Article

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