Thermodynamic relationships between nateglinide polymorphs

Journal of Pharmaceutical and Biomedical Analysis

Volumn 50, Issue 5, 2009, Pages 764-770

  Bruni, G ^a   Berbenni, V ^a   Milanese, C ^a   Girella, A ^a   Cardini, A ^b   Vigano E ^b   Lanfranconi, S ^b   Marini, A ^a  

^a UNIVERSITY OF PAVIA   (Italy)

^b AMSA SpA   (Italy)

Author keywords

DSC; Monotropy; Nateglinide; Physico chemical characterization; Polymorphism

Indexed keywords

NATEGLINIDE;

ARTICLE; CONTROLLED STUDY; CRYSTALLIZATION; DRUG STRUCTURE; MELTING POINT; PHYSICAL CHEMISTRY; PRIORITY JOURNAL; SCANNING ELECTRON MICROSCOPY; THERMODYNAMICS; THERMOSTABILITY; X RAY DIFFRACTION;

CHEMISTRY, PHARMACEUTICAL; CHEMISTRY, PHYSICAL; CRYSTALLIZATION; CRYSTALLOGRAPHY, X-RAY; CYCLOHEXANES; HOT TEMPERATURE; HYPOGLYCEMIC AGENTS; MICROSCOPY, ELECTRON, SCANNING; MODELS, CHEMICAL; MOLECULAR STRUCTURE; PHENYLALANINE; SPECTROPHOTOMETRY; SPECTROPHOTOMETRY, INFRARED; SPECTROSCOPY, FOURIER TRANSFORM INFRARED; TECHNOLOGY, PHARMACEUTICAL; TEMPERATURE; THERMODYNAMICS;

EID: 70349184934     PISSN: 07317085     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jpba.2009.06.017     Document Type: Article

References (7)

1. Lieder T.R. FDA approves nateglinide for treatment of type 2 diabetes. Am. J. Health Syst. Pharm. 58 (2001) 285-288
2. Li G., Xu Q.W., Mo X.Y., Chen J.Y., and Su G.Q. Study on stability of nateglinide polymorphism. Chin. Chem. Lett. 14 (2003) 730-733
3. Marini A., Berbenni V., Bruni G., Margheritis C., and Orlandi A. Physico-chemical study of the solid forms of a new drug. J. Pharm Sci. 90 (2001) 2131-2140
4. Marini A., Berbenni V., Bruni G., Sinistri C., Maggioni A., Orlandi A., and Villa M. Physico-chemical characterization of a novel tricyclic β-lactam antibiotic. J. Pharm. Sci. 89 (2000) 232-240
5. Hilfiker R. Polymorphism in the Pharmaceutical Industry (2006), Wiley-VCH (Chapters 1 and 2)
6. Burger A., and Ramberger R. On the polymorphism of pharmaceuticals and other organic molecular crystals. II. Applicability of thermodynamic rules. Mikrochim Acta II (1979) 273-316
7. Yu L. Inferring thermodynamic stability relationship of polymorphs from melting data. J. Pharm. Sci. 84 (1995) 966-974