Novel derivatives of ISO-1 as potent inhibitors of MIF biological function

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 16, 2009, Pages 4773-4776

  Balachandran, Sarala ^a   Rodge, Atish ^a   Gadekar, Pradip K ^a   Yadav, Vitthal N ^a   Kamath, Divya ^a   Chetrapal Kunwar, Anshu ^a   Bhatt, Pooja ^a   Srinivasan, Shaila ^a   Sharma, Somesh ^a   Vishwakarma, Ram A ^a   Dagia, Nilesh M ^a  

^a Piramal Enterprises Limited   (India)

Author keywords

Amide; Anti inflammatory; ISO 1; MIF; Oxadiazole; Phthalimide

Indexed keywords

1,2,4 OXADIAZOLE DERIVATIVE; AMIDE; INTERLEUKIN 1BETA; INTERLEUKIN 6; ISO 1; ISOXAZOLE DERIVATIVE; MACROPHAGE MIGRATION INHIBITION FACTOR; PHTHALIMIDE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG EFFECT; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME INHIBITION; HUMAN; HUMAN CELL; PERIPHERAL BLOOD MONONUCLEAR CELL; REACTION ANALYSIS; STRUCTURE ANALYSIS;

AMIDES; ANTI-INFLAMMATORY AGENTS; CELL LINE; HUMANS; INTERLEUKIN-1BETA; INTERLEUKIN-6; ISOXAZOLES; OXADIAZOLES; PHTHALIMIDES; RECEPTORS, IMMUNOLOGIC;

EID: 67749099598     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2009.06.052     Document Type: Article

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