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Volumn 199, Issue 11, 2009, Pages 1575-1582

In vivo and in vitro efficacy of amodiaquine against Plasmodium falciparum in an area of Continued Use of 4-aminoquinolines in East Africa

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOQUINOLINE; AMODIAQUINE; ARTEMETHER PLUS BENFLUMETOL; DEETHYLAMODIAQUINE;

EID: 67650656234     PISSN: 00221899     EISSN: None     Source Type: Journal    
DOI: 10.1086/598862     Document Type: Article
Times cited : (25)

References (48)
  • 1
    • 0022646867 scopus 로고
    • Frequency of severe neutropenia associated with amodiaquine prophylaxis against malaria
    • Hatton CS, Peto TE, Bunch C, et al. Frequency of severe neutropenia associated with amodiaquine prophylaxis against malaria. Lancet 1986; 1:411-4.
    • (1986) Lancet , vol.1 , pp. 411-414
    • Hatton, C.S.1    Peto, T.E.2    Bunch, C.3
  • 3
    • 0029807475 scopus 로고    scopus 로고
    • Systematic review of amodiaquine treatment in uncomplicated malaria
    • Olliaro P, Nevill C, LeBras J, et al. Systematic review of amodiaquine treatment in uncomplicated malaria. Lancet 1996; 348:1196-201.
    • (1996) Lancet , vol.348 , pp. 1196-1201
    • Olliaro, P.1    Nevill, C.2    LeBras, J.3
  • 4
    • 67650649105 scopus 로고    scopus 로고
    • WHO Expert Committee on Malaria
    • World Health Organization WHO, Geneva: WHO
    • World Health Organization (WHO). WHO Expert Committee on Malaria, twentieth report. Vol 30. Geneva: WHO, 2000.
    • (2000) twentieth report , vol.30
  • 5
    • 0025986905 scopus 로고
    • Efficacy of amodiaquine against chloroquine-resistant malaria in Cameroon
    • Fadat G, Le Bras J, Hengy C, Louis JP, Gimou MM, Verdier F. Efficacy of amodiaquine against chloroquine-resistant malaria in Cameroon. Lancet 1991; 338:1092.
    • (1991) Lancet , vol.338 , pp. 1092
    • Fadat, G.1    Le Bras, J.2    Hengy, C.3    Louis, J.P.4    Gimou, M.M.5    Verdier, F.6
  • 6
    • 0033385917 scopus 로고    scopus 로고
    • Amodiaquine remains effective for treating uncomplicated malaria in West and Central Africa
    • Brasseur P, Guiguemde R, Diallo S, et al. Amodiaquine remains effective for treating uncomplicated malaria in West and Central Africa. Trans R Soc Trop Med Hyg 1999; 93:645-50.
    • (1999) Trans R Soc Trop Med Hyg , vol.93 , pp. 645-650
    • Brasseur, P.1    Guiguemde, R.2    Diallo, S.3
  • 7
    • 67650681498 scopus 로고    scopus 로고
    • World Health Organization WHO, Geneva: WHO
    • World Health Organization (WHO). Antimalarial treatment policies. Vol 2008. Geneva: WHO, 2007.
    • (2007) Antimalarial treatment policies , vol.2008
  • 9
    • 39449114525 scopus 로고    scopus 로고
    • Translation of artemether-lumefantrine treatment policy into paediatric clinical practice: An early experience from Kenya
    • Zurovac D, Njogu J, Akhwale W, Hamer DH, Snow RW. Translation of artemether-lumefantrine treatment policy into paediatric clinical practice: an early experience from Kenya. Trop Med Int Health 2008; 13:99-107.
    • (2008) Trop Med Int Health , vol.13 , pp. 99-107
    • Zurovac, D.1    Njogu, J.2    Akhwale, W.3    Hamer, D.H.4    Snow, R.W.5
  • 10
    • 0142215646 scopus 로고    scopus 로고
    • East African Network for Monitoring Antimalarial Treatment. The efficacy of antimalarial monotherapies, sulphadoxine-pyrimethamine and amodiaquine in East Africa: implications for sub-regional policy. Trop Med Int Health 2003; 8:860-7.
    • East African Network for Monitoring Antimalarial Treatment. The efficacy of antimalarial monotherapies, sulphadoxine-pyrimethamine and amodiaquine in East Africa: implications for sub-regional policy. Trop Med Int Health 2003; 8:860-7.
  • 11
    • 0345550447 scopus 로고    scopus 로고
    • Atovaquone and proguanil versus amodiaquine for the treatment of Plasmodium falciparum malaria in African infants and young children
    • Borrmann S, Faucher JF, Bagaphou T, et al. Atovaquone and proguanil versus amodiaquine for the treatment of Plasmodium falciparum malaria in African infants and young children. Clin Infect Dis 2003; 37: 1441-7.
    • (2003) Clin Infect Dis , vol.37 , pp. 1441-1447
    • Borrmann, S.1    Faucher, J.F.2    Bagaphou, T.3
  • 12
    • 17844404530 scopus 로고    scopus 로고
    • Amodiaquine alone, amodiaquine+sulfadoxine-pyrimethamine, amodiaquine+artesunate, and artemether-lumefantrine for outpatient treatment of malaria in Tanzanian children: A four-arm randomised effectiveness trial
    • Mutabingwa TK, Anthony D, Heller A, et al. Amodiaquine alone, amodiaquine+sulfadoxine-pyrimethamine, amodiaquine+artesunate, and artemether-lumefantrine for outpatient treatment of malaria in Tanzanian children: a four-arm randomised effectiveness trial. Lancet 2005; 365:1474-80.
    • (2005) Lancet , vol.365 , pp. 1474-1480
    • Mutabingwa, T.K.1    Anthony, D.2    Heller, A.3
  • 13
    • 33751379062 scopus 로고    scopus 로고
    • Amodiaquine resistance is not related to rare findings of pfmdrl gene amplifications in Kenya
    • Holmgren G, Bjorkman A, Gil JP. Amodiaquine resistance is not related to rare findings of pfmdrl gene amplifications in Kenya. Trop Med Int Health 2006; 11:1808-12.
    • (2006) Trop Med Int Health , vol.11 , pp. 1808-1812
    • Holmgren, G.1    Bjorkman, A.2    Gil, J.P.3
  • 14
    • 0037140198 scopus 로고    scopus 로고
    • Amodiaquine-artesunate versus amodiaquine for uncomplicated Plasmodium falciparum malaria in African children: A randomised, multicentre trial
    • Adjuik M, Agnamey P, Babiker A, et al. Amodiaquine-artesunate versus amodiaquine for uncomplicated Plasmodium falciparum malaria in African children: a randomised, multicentre trial. Lancet 2002; 359:1365-72.
    • (2002) Lancet , vol.359 , pp. 1365-1372
    • Adjuik, M.1    Agnamey, P.2    Babiker, A.3
  • 15
    • 33646472123 scopus 로고    scopus 로고
    • In-vitro susceptibility of Plasmodium falciparum to monodesethylamodiaquine, dihydroartemisinin and quinine in an area of high chloroquine resistance in Rwanda
    • Tinto H, Rwagacondo C, Karema C, et al. In-vitro susceptibility of Plasmodium falciparum to monodesethylamodiaquine, dihydroartemisinin and quinine in an area of high chloroquine resistance in Rwanda. Trans R Soc Trop Med Hyg 2006; 100:509-14.
    • (2006) Trans R Soc Trop Med Hyg , vol.100 , pp. 509-514
    • Tinto, H.1    Rwagacondo, C.2    Karema, C.3
  • 16
    • 0242267910 scopus 로고    scopus 로고
    • Isoquine and related amodiaquine analogues: A new generation of improved 4-aminoquinoline antimalarials
    • O'Neill PM, Mukhtar A, Stocks PA, et al. Isoquine and related amodiaquine analogues: a new generation of improved 4-aminoquinoline antimalarials. J Med Chem 2003; 46:4933-45.
    • (2003) J Med Chem , vol.46 , pp. 4933-4945
    • O'Neill, P.M.1    Mukhtar, A.2    Stocks, P.A.3
  • 17
    • 0042737835 scopus 로고    scopus 로고
    • Spatial and temporal heterogeneity of Anopheles mosquitoes and Plasmodium falciparum transmission along the Kenyan coast
    • Mbogo CM, Mwangangi JM, Nzovu J, et al. Spatial and temporal heterogeneity of Anopheles mosquitoes and Plasmodium falciparum transmission along the Kenyan coast. Am J Trop Med Hyg 2003; 68:734-42.
    • (2003) Am J Trop Med Hyg , vol.68 , pp. 734-742
    • Mbogo, C.M.1    Mwangangi, J.M.2    Nzovu, J.3
  • 18
    • 54849434602 scopus 로고    scopus 로고
    • Effect of a fall in malaria transmission on morbidity and mortality in Kilifi, Kenya
    • O'Meara WP, Bejon P, Mwangi TW, et al. Effect of a fall in malaria transmission on morbidity and mortality in Kilifi, Kenya. Lancet 2008; 372:1555-62.
    • (2008) Lancet , vol.372 , pp. 1555-1562
    • O'Meara, W.P.1    Bejon, P.2    Mwangi, T.W.3
  • 19
  • 20
    • 0029008630 scopus 로고
    • Indicators of life-threatening malaria in African children
    • Marsh K, Forster D, Waruiru C, et al. Indicators of life-threatening malaria in African children. N Engl J Med 1995; 332:1399-404.
    • (1995) N Engl J Med , vol.332 , pp. 1399-1404
    • Marsh, K.1    Forster, D.2    Waruiru, C.3
  • 22
    • 0027332108 scopus 로고
    • Plasmodium falciparum: A rapid technique for genotyping the merozoite surface protein 2
    • Felger I, Tavul L, Beck HP. Plasmodium falciparum: a rapid technique for genotyping the merozoite surface protein 2. Exp Parasitol 1993; 77:372-5.
    • (1993) Exp Parasitol , vol.77 , pp. 372-375
    • Felger, I.1    Tavul, L.2    Beck, H.P.3
  • 23
    • 0018606732 scopus 로고
    • Quantitative assessment of antimalarial activity in vitro by a semiautomated microdilution technique
    • Desjardins RE, Canfield CJ, Haynes JD, Chulay JD. Quantitative assessment of antimalarial activity in vitro by a semiautomated microdilution technique. Antimicrob Agents Chemother 1979; 16:710-8.
    • (1979) Antimicrob Agents Chemother , vol.16 , pp. 710-718
    • Desjardins, R.E.1    Canfield, C.J.2    Haynes, J.D.3    Chulay, J.D.4
  • 24
    • 0021028710 scopus 로고
    • Plasmodium falciparum: Effect of time in continuous culture on binding to human endothelial cells and amelanotic melanoma cells
    • Udeinya IJ, Graves PM, Carter R, Aikawa M, Miller LH. Plasmodium falciparum: effect of time in continuous culture on binding to human endothelial cells and amelanotic melanoma cells. Exp Parasitol 1983; 56: 207-14.
    • (1983) Exp Parasitol , vol.56 , pp. 207-214
    • Udeinya, I.J.1    Graves, P.M.2    Carter, R.3    Aikawa, M.4    Miller, L.H.5
  • 25
    • 0027535450 scopus 로고
    • In vitro activity of monodesethylamodiaquine and amopyroquine against African isolates and clones of Plasmodium falciparum
    • Basco LK, Le Bras J. In vitro activity of monodesethylamodiaquine and amopyroquine against African isolates and clones of Plasmodium falciparum. Am J Trop Med Hyg 1993; 48:120-5.
    • (1993) Am J Trop Med Hyg , vol.48 , pp. 120-125
    • Basco, L.K.1    Le Bras, J.2
  • 26
    • 33746898151 scopus 로고    scopus 로고
    • National Institute of Allergy and Infectious Diseases NIAID, Bethesda, MD: NIAID
    • National Institute of Allergy and Infectious Diseases (NIAID). Pediatric toxicity tables. Bethesda, MD: NIAID, 2003.
    • (2003) Pediatric toxicity tables
  • 27
    • 0023056632 scopus 로고
    • Isolation, characterization and standardization of a major metabolite of amodiaquine by chromatographic and spectroscopic methods
    • Churchill FC, Mount DL, Patchen LC, Bjorkman A. Isolation, characterization and standardization of a major metabolite of amodiaquine by chromatographic and spectroscopic methods. J Chromatogr 1986; 377: 307-18.
    • (1986) J Chromatogr , vol.377 , pp. 307-318
    • Churchill, F.C.1    Mount, D.L.2    Patchen, L.C.3    Bjorkman, A.4
  • 28
    • 0023628910 scopus 로고
    • Disposition of monodesethylamodiaquine after a single oral dose of amodiaquine and three regimens for prophylaxis against Plasmodium falciparum malaria
    • Pussard E, Verdier F, Faurisson F, Scherrmann JM, Le Bras J, Blayo MC. Disposition of monodesethylamodiaquine after a single oral dose of amodiaquine and three regimens for prophylaxis against Plasmodium falciparum malaria. Eur J Clin Pharmacol 1987; 33:409-14.
    • (1987) Eur J Clin Pharmacol , vol.33 , pp. 409-414
    • Pussard, E.1    Verdier, F.2    Faurisson, F.3    Scherrmann, J.M.4    Le Bras, J.5    Blayo, M.C.6
  • 29
    • 34748818756 scopus 로고    scopus 로고
    • Population pharmacokinetics of amodiaquine and desethylamodiaquine in pediatric patients with uncomplicated falciparum malaria
    • Hietala SF, Bhattarai A, Msellem M, et al. Population pharmacokinetics of amodiaquine and desethylamodiaquine in pediatric patients with uncomplicated falciparum malaria. J Pharmacokinet Pharmacodyn 2007; 34:669-86.
    • (2007) J Pharmacokinet Pharmacodyn , vol.34 , pp. 669-686
    • Hietala, S.F.1    Bhattarai, A.2    Msellem, M.3
  • 30
    • 0024544340 scopus 로고
    • A comparison of the in vitro activities of amodiaquine and desethylamodiaquine against isolates of Plasmodium falciparum
    • Childs GE, Boudreau EF, Milhous WK, et al. A comparison of the in vitro activities of amodiaquine and desethylamodiaquine against isolates of Plasmodium falciparum. Am J Trop Med Hyg 1989; 40:7-11.
    • (1989) Am J Trop Med Hyg , vol.40 , pp. 7-11
    • Childs, G.E.1    Boudreau, E.F.2    Milhous, W.K.3
  • 33
    • 0030007219 scopus 로고    scopus 로고
    • Pharmacokinetics of quinine, chloroquine and amodiaquine: Clinical implications
    • Krishna S, White NJ. Pharmacokinetics of quinine, chloroquine and amodiaquine: clinical implications. Clin Pharmacokinet 1996; 30:263-99.
    • (1996) Clin Pharmacokinet , vol.30 , pp. 263-299
    • Krishna, S.1    White, N.J.2
  • 34
    • 0036207647 scopus 로고    scopus 로고
    • In vitro activities of ferrochloroquine against 55 Senegalese isolates of Plasmodium falciparum in comparison with those of standard antimalarial drugs
    • Pradines B, Tall A, Rogier C, et al. In vitro activities of ferrochloroquine against 55 Senegalese isolates of Plasmodium falciparum in comparison with those of standard antimalarial drugs. Trop Med Int Health 2002; 7:265-70.
    • (2002) Trop Med Int Health , vol.7 , pp. 265-270
    • Pradines, B.1    Tall, A.2    Rogier, C.3
  • 35
    • 7844249022 scopus 로고    scopus 로고
    • In vitro susceptibility of Gabonese wild isolates of Plasmodium falciparum to artemether, and comparison with chloroquine, quinine, halofantrine and amodiaquine
    • Pradines B, Mabika Mamfoumbi M, Parzy D, et al. In vitro susceptibility of Gabonese wild isolates of Plasmodium falciparum to artemether, and comparison with chloroquine, quinine, halofantrine and amodiaquine. Parasitology 1998; 117:541-5.
    • (1998) Parasitology , vol.117 , pp. 541-545
    • Pradines, B.1    Mabika Mamfoumbi, M.2    Parzy, D.3
  • 36
    • 33750577489 scopus 로고    scopus 로고
    • Polymorphisms in pfcrt, pfmdrl, dhfr genes and in vitro responses to antimalarials in Plasmodium falciparum isolates from Bangui, Central African Republic
    • Menard D, Yapou F, Manirakiza A, Djalle D, Matsika-Claquin MD, Talarmin A. Polymorphisms in pfcrt, pfmdrl, dhfr genes and in vitro responses to antimalarials in Plasmodium falciparum isolates from Bangui, Central African Republic. Am J Trop Med Hyg 2006; 75:381-7.
    • (2006) Am J Trop Med Hyg , vol.75 , pp. 381-387
    • Menard, D.1    Yapou, F.2    Manirakiza, A.3    Djalle, D.4    Matsika-Claquin, M.D.5    Talarmin, A.6
  • 37
    • 0022403153 scopus 로고
    • Intravenous amodiaquine and oral amodiaquine/erythromycin in the treatment of chloroquineresistant falciparum malaria
    • Looareesuwan S, Phillips RE, White NJ, et al. Intravenous amodiaquine and oral amodiaquine/erythromycin in the treatment of chloroquineresistant falciparum malaria. Lancet 1985; 2:805-8.
    • (1985) Lancet , vol.2 , pp. 805-808
    • Looareesuwan, S.1    Phillips, R.E.2    White, N.J.3
  • 38
    • 34249699738 scopus 로고    scopus 로고
    • Combination therapy for uncomplicated falciparum malaria in Ugandan children: A randomized trial
    • Dorsey G, Staedke S, Clark TD, et al. Combination therapy for uncomplicated falciparum malaria in Ugandan children: a randomized trial. JAMA 2007; 297:2210-9.
    • (2007) JAMA , vol.297 , pp. 2210-2219
    • Dorsey, G.1    Staedke, S.2    Clark, T.D.3
  • 40
    • 42949156655 scopus 로고    scopus 로고
    • Effects of Plasmodium falciparum parasite population size and patient age on early and late parasitological outcomes of antimalarial treatment in children
    • Borrmann S, Matsiegui PB, Missinou MA, Kremsner PG. Effects of Plasmodium falciparum parasite population size and patient age on early and late parasitological outcomes of antimalarial treatment in children. Antimicrob Agents Chemother 2008; 52:1799-805.
    • (2008) Antimicrob Agents Chemother , vol.52 , pp. 1799-1805
    • Borrmann, S.1    Matsiegui, P.B.2    Missinou, M.A.3    Kremsner, P.G.4
  • 41
    • 35248823116 scopus 로고    scopus 로고
    • World Antimalarial Resistance Network (WARN) II: In vitro antimalarial drug susceptibility
    • Bacon DJ, Jambou R, Fandeur T, et al. World Antimalarial Resistance Network (WARN) II: in vitro antimalarial drug susceptibility. Malar J 2007; 6:120.
    • (2007) Malar J , vol.6 , pp. 120
    • Bacon, D.J.1    Jambou, R.2    Fandeur, T.3
  • 42
    • 0037068963 scopus 로고    scopus 로고
    • Chlorproguanil-dapsone versus sulfadoxine-pyrimethamine for sequential episodes of uncomplicated falciparum malaria in Kenya and Malawi: A randomised clinical trial
    • Sulo J, Chimpeni P, Hatcher J, et al. Chlorproguanil-dapsone versus sulfadoxine-pyrimethamine for sequential episodes of uncomplicated falciparum malaria in Kenya and Malawi: a randomised clinical trial. Lancet 2002; 360:1136-43.
    • (2002) Lancet , vol.360 , pp. 1136-1143
    • Sulo, J.1    Chimpeni, P.2    Hatcher, J.3
  • 43
    • 33847717147 scopus 로고    scopus 로고
    • Molecular epidemiology of malaria in Cameroon. XXIV. Trends of in vitro antimalarial drug responses in Yaounde, Cameroon
    • Basco LK, Ringwald P. Molecular epidemiology of malaria in Cameroon. XXIV. Trends of in vitro antimalarial drug responses in Yaounde, Cameroon. Am J Trop Med Hyg 2007; 76:20-6.
    • (2007) Am J Trop Med Hyg , vol.76 , pp. 20-26
    • Basco, L.K.1    Ringwald, P.2
  • 44
    • 24144461306 scopus 로고    scopus 로고
    • Short-course regimens of artesunate-fosmidomycin in treatment of uncomplicated Plasmodium falciparum malaria
    • Borrmann S, Adegnika AA, Moussavou F, et al. Short-course regimens of artesunate-fosmidomycin in treatment of uncomplicated Plasmodium falciparum malaria. Antimicrob Agents Chemother 2005; 49:3749-54.
    • (2005) Antimicrob Agents Chemother , vol.49 , pp. 3749-3754
    • Borrmann, S.1    Adegnika, A.A.2    Moussavou, F.3
  • 45
    • 17144379315 scopus 로고    scopus 로고
    • Efficacy and safety of artemether-lumefantrine (Coartem) tablets (six-dose regimen) in African infants and children with acute, uncomplicated falciparum malaria
    • Falade C, Makanga M, Premji Z, Ortmann CE, Stockmeyer M, de Palacios PI. Efficacy and safety of artemether-lumefantrine (Coartem) tablets (six-dose regimen) in African infants and children with acute, uncomplicated falciparum malaria. Trans R Soc Trop Med Hyg 2005; 99: 459-67.
    • (2005) Trans R Soc Trop Med Hyg , vol.99 , pp. 459-467
    • Falade, C.1    Makanga, M.2    Premji, Z.3    Ortmann, C.E.4    Stockmeyer, M.5    de Palacios, P.I.6
  • 46
    • 45349085051 scopus 로고    scopus 로고
    • Sulfadoxine-pyrimethaminebased combinations for malaria: A randomised blinded trial to compare efficacy, safety and selection of resistance in Malawi
    • Bell DJ, Nyirongo SK, Mukaka M, et al. Sulfadoxine-pyrimethaminebased combinations for malaria: a randomised blinded trial to compare efficacy, safety and selection of resistance in Malawi. PLoS ONE 2008; 3:e1578.
    • (2008) PLoS ONE , vol.3
    • Bell, D.J.1    Nyirongo, S.K.2    Mukaka, M.3
  • 47
    • 0032410803 scopus 로고    scopus 로고
    • Metabolism-dependent neutrophil cytotoxicity of amodiaquine: A comparison with pyronaridine and related antimalarial drugs
    • Naisbitt DJ, Williams DP, O'Neill PM, et al. Metabolism-dependent neutrophil cytotoxicity of amodiaquine: a comparison with pyronaridine and related antimalarial drugs. Chem Res Toxicol 1998; 11:1586-95.
    • (1998) Chem Res Toxicol , vol.11 , pp. 1586-1595
    • Naisbitt, D.J.1    Williams, D.P.2    O'Neill, P.M.3
  • 48
    • 0024523935 scopus 로고
    • Drug-protein conjugatesXVIII. Detection of antibodies towards the antimalarial amodiaquine and its quinone imine metabolite in man and the rat
    • Christie G, Breckenridge AM, Park BK. Drug-protein conjugatesXVIII. Detection of antibodies towards the antimalarial amodiaquine and its quinone imine metabolite in man and the rat. Biochem Pharmacol 1989; 38:1451-8.
    • (1989) Biochem Pharmacol , vol.38 , pp. 1451-1458
    • Christie, G.1    Breckenridge, A.M.2    Park, B.K.3


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