Reversed-phase TLC study of the lipophilicity of some 3-hydroxy-1,2- benzisoxazoles substituted in the benzene ring

Acta Chromatographica

Volumn 21, Issue 2, 2009, Pages 251-258

  Slawik T ^a   Skibinski R ^a   Paw, B ^a   Dzialo G ^a  

^a MEDICAL UNIVERSITY OF LUBLIN   (Poland)

Author keywords

1,2 benzisothiazolones; 3 hydroxy 1,2 benzisoxazoles; Calculated partition coefficients; Lipophilicity; Retention R M 0 ; RP TLC

Indexed keywords

EID: 67650504843     PISSN: 12332356     EISSN: 20835736     Source Type: Journal    
DOI: 10.1556/AChrom.21.2009.2.5     Document Type: Article

References (27)

1. A. Leo, C. Hansch, D. Elkins, Chem. Rev., 71, 525, (1971)
2. T. Fujita, J. Iwasa, C. Hansch, J. Am. Chem Soc., 86, 5175, (1964)
3. R. F. Rekker, R. Mannhold, Calculation of Drug Lipophilicity, The Hydrophobic Fragmental Constant Approach VCH, Weinheim, 1992
4. L. G. Danielsson, Y. H. Zhang, Trends Anal. Chem., 15, 188, (1996)
5. T. Hartmann, J. Schmitt, Drug Discovery Today, Technologies, 1, 431, (2004)
6. M. E. Morgan, L. Kui, B. Anderson, J. Pharm. Sci, 87, 238, (1998)
7. A. Persona, Z. Fekner, B. Marczewska, T. Sławik, XLV Conference of Polish Chemical Society vol II 870, Kraków, (2002)
8. G. Bouchard, P. A. Carrupt, B. Testa. V. Gobry, H. H. Girault, Chem Eur. J., 8, 3478, (2002)
9. J. Østergaard, S. H. Hansen, H. Larsen, Ch. Shou, N. H. H. Heegard, Electrophoresis, 24, 1078, (2003)
10. M. Bajda, A. Bucki, J. Szlȩk, M. Szwaczkiewicz, M. Świerczek, B. Malawska, Biomed. Chromatogr. DOJ: 10.1002/bmc (2007)
11. T. Ba̧czek, M. Markuszewski, R. Kaliszan, M. A. van Straten, H. A. Claessens; J. High Resol. Chromatogr., 23, 667, (2000)
12. J. Kresta, P. Kastner, J. Klimeš, V. Klimešowa, J. Liq. Chromatogr. Rel. Technolog., 27, 2539, (2004)
13. D. Matosiuk, K. Jóźwiak, J. Planar Chromatogr., 13, 130, (2000)
14. S. Boryczka, K. Kulig, B. Malawska, J. Planar Chromatogr., 16, 117, (2003)
15. K. Kulig, B. Malawska, Biomed. Chromatogr., 17, 1, (2003)
16. T. Sławik, B. Paw, J. Planar Chromatogr., 16, 442, (2003)
17. I. V. Tetko, V. J. Tanchuk, VCC - Lab, 2002, http://146.107.217.178/ servlets/ vcc.lab?action-alogps
18. C. Bertaccini, M. Impiccatore, T. Vitali, Pharmacol. Res. Commun., 3, 385, (1971); Chem. Abstr., 77, 70117, (1972)
19. M. Impiccatore, T. Vitali, G. Bertaccini, Boll. Soc. Ital. Biol. Sper., 47, 296, (1971); Chem. Abstr., 76, 254, (1972)
20. H. Böshagen, Chem. Ber., 100, 954, (1967)
21. T. Sławik, E. Domagalina, Acta Polon. Pharm., XLI, 625, (1984)
22. T. Braumann, J. Chromatogr., 323, 191, (1986)
23. K Dross, R. F. Rekker, G. de Viers, R. Mannhold, Quant. Struct. Act. Relat, 17, 549, (1998)
24. P. Kästern, L. Klimeš, P. Velenovska, V. Klimešowa, J. Planar Chromatogr., 15, 200, (2002)
25. A. Pyka, M. Dołowy, J. Liq. Chromatogr. Rel. Technol, 28, 293, (2005)
26. T. Sławik, C. Kowalski, J. Chromatogr. A, 952, 295, (2002)
27. M. Daszykowski, B. Walczak, D.L. Massart, Chemom. Intell. Lab. Syst. 65, 97, (2003)