1,3,5-Triazepan-2,6-diones as conformationally constrained dipeptide mimetics. in silico guided identification of sPLA2 inhibitors

Advances in Experimental Medicine and Biology

Volumn 611, Issue , 2009, Pages 201-202

  Guichard, Gilles ^a   Léna, Gersande ^a   Boeglin, Joel ^a   Muller, Pascal ^b   Boilard, Eric ^c   Lambeau, Gérard ^c   Rognan, Didier ^b   Didierjean, Claude ^d  

^a INSTITUT DE BIOLOGIE MOLÉCULAIRE ET CELLULAIRE   (France)

^b CNRS   (France)

^c INSTITUT DE PHARMACOLOGIE MOLÉCULAIRE ET CELLULAIRE   (France)

^d UNIVERSITÉ DE LORRAINE   (France)

Author keywords

[No Author keywords available]

Indexed keywords

1,3,5 TRIAZEPAM 2,6 DIONE; PEPTIDOMIMETIC AGENT; PHOSPHOLIPASE A2; PHOSPHOLIPASE A2 INHIBITOR; UNCLASSIFIED DRUG; DIPEPTIDE; ENZYME INHIBITOR; TRIAZINE DERIVATIVE;

ARTICLE; COMPUTER MODEL; DRUG CONFORMATION; DRUG IDENTIFICATION; DRUG PROTEIN BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; PRIORITY JOURNAL; CHEMICAL STRUCTURE; CHEMISTRY; DRUG ANTAGONISM; MOLECULAR MIMICRY; PROTEIN CONFORMATION;

DIPEPTIDES; ENZYME INHIBITORS; MODELS, MOLECULAR; MOLECULAR MIMICRY; PHOSPHOLIPASES A2; PROTEIN CONFORMATION; TRIAZINES;

EID: 66349119940     PISSN: 00652598     EISSN: None     Source Type: Book Series    
DOI: 10.1007/978-0-387-73657-0_92     Document Type: Article

References (5)

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