Mapping of suramin binding sites on the group IIA human secreted phospholipase A2

Bioorganic Chemistry

Volumn 37, Issue 2, 2009, Pages 41-45

  Vieira, Davi Serradella ^a   Aragão, Elisangela Aparecida ^a   Lourenzoni, Marcos Roberto ^a   Ward, Richard J ^a  

^a UNIVERSITY OF SÃO PAULO   (Brazil)

Author keywords

Isothermal titration calorimetry; Molecular dynamics

Indexed keywords

PHOSPHOLIPASE A2; PHOSPHOLIPASE A2 GROUP IIA; SURAMIN; UNCLASSIFIED DRUG;

ARTICLE; BINDING SITE; CONTROLLED STUDY; CRYSTAL STRUCTURE; DRUG PROTEIN BINDING; ELECTRICITY; ENZYME ACTIVITY; ENZYME RELEASE; HUMAN; HYDROLYSIS; HYDROPHOBICITY; ISOTHERMAL TITRATION CALORIMETRY; MOLECULAR DYNAMICS; NUCLEOTIDE SEQUENCE; PHOSPHOLIPID MEMBRANE; PRIORITY JOURNAL;

ANTINEMATODAL AGENTS; BINDING SITES; CALORIMETRY; COMPUTER SIMULATION; GROUP II PHOSPHOLIPASES A2; HUMANS; MODELS, MOLECULAR; PROTEIN CONFORMATION; PROTEIN STRUCTURE, TERTIARY; RECOMBINANT PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP; SURAMIN; THERMODYNAMICS;

EID: 62949180597     PISSN: 00452068     EISSN: 10902120     Source Type: Journal    
DOI: 10.1016/j.bioorg.2009.01.002     Document Type: Article

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