Diversity-oriented synthesis of substituted pyrazolo-[4,3-d][1,2,3]triazin-4-ones

Heterocycles

Volumn 78, Issue 1, 2009, Pages 71-91

  Meibom, Daniel ^a   Bauser, Marcus ^a   Meier, Heinrich ^a   Schneider, Dirk ^a   Svenstrup, Niels ^a   Haebich, Dieter ^a  

^a BAYER PHARMA AG   (Germany)

Author keywords

Amidation Cyclization; Methoxycarbonylation; Parallel Synthesis; Sonogashira Coupling; Suzuki Coupling

Indexed keywords

EID: 62549113444     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/COM-08-11482     Document Type: Article

References (13)

1. Cheng C.C., and Zee-Cheng R.K.-Y. Drugs of the future 11 (1986) 121
2. Baraldi P.G., Simoni D., Periotto V., Manfredini S., Guarneri M., Manservigi R., Cassai E., and Bertolasi V. J. Med. Chem. 27 (1984) 986
3. Baraldi P.G., Cacciari B., Dalpiaz A., Dionisotti S., Zocchi C., Pineda de las Infantas M.J., Spalluto G., and Varani K. Drug Res. 46 (1996) 365
4. Manfredini S., Bazzanini R., Baraldi P.G., Guarneri M., Simoni D., Marongiu M.E., Pani A., Tramontano E., and La Colla P. J. Med. Chem. 35 (1992) 917
5. Baraldi P.G., Casolari A., Guarneri M., Manfredini S., Pollini G.P., Simoni D., and Zanirato V. Synthesis 1 (1988) 78
6. Baraldi P.G., Garuti L., and Roberti M. Synthesis 12 (1994) 1437
7. Long R.A., Gerster J.F., and Townsend L.B. J. Heterocycl. Chem. 7 (1970) 863
8. Buchanan J.G., Stobie A., and Wightman H. J. Chem. Soc., Perkin Trans. 1 (1981) 2374
9. Gil C., Schwoegler A., and Braese S. J. Comb. Chem. 6 (2004) 38
10. Hrelia P., Fimognari C., Maffei F., Brighenti B., Garuti L., Burnelli S., and Cantelli-Forti G. Mutation Research 397 (1998) 293
11. Baraldi P.G., Cacciari B., Leoni A., Recanatini M., Roberti M., Rossi M., Manfredini S., Periotto V., and Simoni D. Il Farmaco 46 (1991) 1337
12. Svenstrup N., Freiberg C., Lohrmann E., Bauser M., Meibom D., Meier H., and Schiffer G. DE 10 2005 021 963 A1 (2005)
13. Bartlett S., and Nelson A. Org. Biomol. Chem. 2 (2004) 2874