Synthesis and in vitro cysticidal activity of new benzimidazole derivatives

European Journal of Medicinal Chemistry

Volumn 44, Issue 4, 2009, Pages 1794-1800

  Palomares Alonso, Francisca ^a,b   Jung Cook, Helgi ^a,b   Pérez Villanueva, Jaime ^b   Piliado, Juan Carlos ^a   Rodríguez Morales, Sergio ^b   Palencia Hernández, Guadalupe ^a   López Balbiaux, Nayeli ^b   Hernández Campos, Alicia ^b   Castillo, Rafael ^b   Hernández Luis, Francisco ^b  

^a NATIONAL INSTITUTE OF NEUROLOGY AND NEUROSURGERY   (Mexico)

^b UNIVERSIDAD NACIONAL AUTÓNOMA DE MÉXICO   (Mexico)

Author keywords

Benzimidazole analogues; Cysticidal activity; Molecular modelling

Indexed keywords

4 NITROBENZYL 2 [(METHOXYCARBONYL)AMINO] 1H BENZIMIDAZOLE 5 CARBOXYLATE; ALBENDAZOLE SULFOXIDE; BENZIMIDAZOLE DERIVATIVE; CARBAMIC ACID DERIVATIVE; METHYL [1 METHYL 5 (PROPYLTHIO) 1H BENZIMIDAZOL 2 YL]CARBAMATE; METHYL [1 METHYL 6 (PROPYLTHIO) 1H BENZIMIDAZOL 2 YL]CARBAMATE; METHYL [5 (PIPERIDIN 1 YLCARBONYL) 1H BENZIMIDAZOL 2 YL]CARBAMATE; METHYL [5 [(METHYLAMINO)CARBONYL] 1H BENZIMIDAZOL 2 YL]CARBAMATE; METHYL METHYL[5 (PROPYLTHIO) 1H BENZIMIDAZOL 2 YL]CARBAMATE; UNCLASSIFIED DRUG;

ANTIMICROBIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; CYSTICIDAL ACTIVITY; DRUG EFFICACY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; IN VITRO STUDY; MALE; MOUSE; NONHUMAN; TAENIA CRASSICEPS;

ALBENDAZOLE; ANIMALS; ANTHELMINTICS; BENZIMIDAZOLES; DRUG DESIGN; MODELS, MOLECULAR; REFERENCE STANDARDS; TAENIA;

EID: 61349184552     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2008.05.005     Document Type: Article

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