Structure of human protein kinase CK2α2 with a potent indazole-derivative inhibitor

Acta Crystallographica Section F: Structural Biology and Crystallization Communications

Volumn 65, Issue 2, 2009, Pages 75-79

  Nakaniwa, Tetsuko ^a   Kinoshita, Takayoshi ^a   Sekiguchi, Yusuke ^a   Tada, Toshiji ^a   Nakanishi, Isao ^b,c   Kitaura, Kazuo ^c   Suzuki, Yamato ^c   Ohno, Hiroaki ^c   Hirasawa, Akira ^c   Tsujimoto, Gozoh ^c  

^a Osaka Prefecture University   (Japan)

^b KINKI UNIVERSITY   (Japan)

^c KYOTO UNIVERSITY   (Japan)

Author keywords

Casein kinase 2; CK2 inhibitors; CK2 2; Selective kinase inhibitors

Indexed keywords

CASEIN KINASE II; INDAZOLE DERIVATIVE; ISOENZYME; PROTEIN KINASE; PROTEIN KINASE INHIBITOR;

ARTICLE; CHEMISTRY; COMPARATIVE STUDY; DRUG ANTAGONISM; HUMAN; METABOLISM; PHYSIOLOGY; PROTEIN SECONDARY STRUCTURE; X RAY CRYSTALLOGRAPHY;

CASEIN KINASE II; CRYSTALLOGRAPHY, X-RAY; HUMANS; INDAZOLES; ISOENZYMES; PROTEIN KINASE INHIBITORS; PROTEIN KINASES; PROTEIN STRUCTURE, SECONDARY;

EID: 59749086318     PISSN: 17443091     EISSN: 17443091     Source Type: Journal    
DOI: 10.1107/S1744309108043194     Document Type: Article

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