Mild and selective synthesis of an aryl boronic ester by equilibration of mixtures of boronic and borinic acid derivatives

Organic Process Research and Development

Volumn 12, Issue 6, 2008, Pages 1265-1268

  Hawkins, Vanessa F ^a   Wilkinson, Mark C ^a   Whiting, Matthew ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 58149131534     PISSN: 10836160     EISSN: 1520586X     Source Type: Journal    
DOI: 10.1021/op800169s     Document Type: Article

References (6)

1. For leading references see: (a) Hall, D. G. Boronic Acids; Wiley: New York, 2005.
2. For leading references see: (a) De-Meijere, A.; Diederich, F. Metal Catalyzed Cross Coupling Reactions; Wiley; New York, 2004.
3. Brown, H. C.; Cole, T. E. Organometallics 1983, 2, 1316-1319.
4. Li, W.; Nelson, D. P.; Jensen, M. S.; Hoerrner, R. S.; Cai, D.; Larsen, R. D.; Reider, P. J. Org. Chem. 2002, 67, 5394-5397.
5. Gadamasetti, K. G. Process Chemistry in the Pharmaceutical Industry; Marcel Dekker: New York, 1999.
6. Winkle, D. D.; Schaab, K. M. Org. Process Res. Dev. 2001, 5, 450-451.