Preparation and prodrug studies of quercetin pentabenzensulfonate

Yakugaku Zasshi

Volumn 128, Issue 12, 2008, Pages 1845-1849

  Peng, You ^a,b   Deng, Zeyuan ^a   Wang, Chunfeng ^b  

^a NANCHANG UNIVERSITY   (China)

^b JIUJIANG UNIVERSITY   (China)

Author keywords

Benzensulfonate; Crystal structure; Hydrolysis; Partition coefficient; Prodrug

Indexed keywords

QUERCETIN; QUERCETIN DERIVATIVE; QUERCETIN PENTABENZENSULFONATE; UNCLASSIFIED DRUG;

ARTICLE; DRUG BIOAVAILABILITY; DRUG DESIGN; DRUG HALF LIFE; DRUG SOLUBILITY; DRUG STRUCTURE; DRUG SYNTHESIS; HYDROLYSIS; PARTITION COEFFICIENT; X RAY;

BENZENESULFONATES; BIOLOGICAL AVAILABILITY; HALF-LIFE; HYDROLYSIS; LIPIDS; MOLECULAR CONFORMATION; PRODRUGS; QUERCETIN; SOLUBILITY; WATER;

EID: 57149091984     PISSN: 00316903     EISSN: 13475231     Source Type: Journal    
DOI: 10.1248/yakushi.128.1845     Document Type: Article

References (15)

1. Kiihnau J., World. Rev. Nutr. Diet., 24, 117-191 (1976).
2. Calias P., Galanopoulos T., Alarcao M., Khayat A., Graves D., Antoniades H. N., d'Alarcao M., Carbohydr. Res., 292, 83-90 (1996).
3. Avila M. A., Velasco J. A., Cansado J., Notario V., Cancer Res., 54, 2424-2428 (1994).
4. Scambia G., Benedetti Panici P., Ranelletti F. O., Ferrandina G., DeVincenzo R., Piantelli M., Masciullo V., Bonanno G., Isola G., Mancuso S., Int. J. Cancer, 57, 211-215 (1994).
5. Yoshida M., Yamamoto M., Nikaido T., Cancer Res., 52, 6676-6681 (1992).
6. Agullo G., Gamet L., Besson C., Demigne, C., Remesy C., Cancer Lett., 87, 55-63 (1994).
7. Li M., Han X. W., Yu B., Tetrahedron Lett., 43, 9467-9470 (2002).
8. Mulholland P. J., Ferry D. R., Anderson D., Hussain S. A., Young A. M., Cook J. E., Hodgkin E., Seymour L. W., Kerr D. J., ESMO, 12, 245-248 (2001).
9. Peng Y., Deng Z. Y., Lang S. J., Xiong D. M., Acta Crystallogr., E63, 4787 (2007).
10. Bruker AXS, Inc., SMART (Version 5.628) and SAINT (Version 6.02). Bruker AXS, Inc., Madison, Wisconsin, USA, 1998.
11. Sheldrick, G. M., SADABS, Program for Empirical Absorption Correction of Area Detector, University of Göttingen, Germany, 1996.
12. Sheldrick, G. M. SHELXTL V5.1 "Software Reference Manual", Bruker AXS, Inc., Madison, Wisconsin, USA.
13. Wang S. Y., Du Z. L., Li R. X., Wu D. C., Tai Y. L., "The Global Seabuckthorn Research and Development", 2, 12-15 (2004).
14. Gugler R., Leschik M., Dengler H., J. Eur. J. Clin. Pharmacol., 9, 229-234 (1975).
15. Adamson A. W., "A Textbook of Physical Chemistry", 3rd ed., Los Angeles, 1986, p. 541.