The absolute configuration plays an important role in muscarinic activity of BGT-A and its analogs

Bioorganic and Medicinal Chemistry

Volumn 16, Issue 24, 2008, Pages 10251-10256

  Niu, Yin Yao ^a   Zhu, Liang ^a   Cui, Yong Yao ^a   Liu, Hui Zhong ^a   Chen, Hong Zhuan ^a   Lu, Yang ^a  

^a SHANGHAI JIAO TONG UNIVERSITY SCHOOL OF MEDICINE   (China)

Author keywords

Absolute configuration; Analogs of Baogongteng A; Enantiomers; Muscarinic agonist and antagonist; Mydriatic and myotic

Indexed keywords

BAOGONGTENG A; MUSCARINIC RECEPTOR; NORTROPANE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; DRUG ACTIVITY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; ENANTIOMER; FEMALE; GUINEA PIG; MALE; NONHUMAN;

ANIMALS; FEMALE; GUINEA PIGS; MALE; MOTOR ACTIVITY; MUSCARINIC AGONISTS; MUSCLE, SKELETAL; RABBITS; RATS; RECEPTORS, MUSCARINIC; STEREOISOMERISM; SUBMANDIBULAR GLAND; TROPANES;

EID: 56349126563     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2008.10.047     Document Type: Article

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