Peptides based on CcdB protein as novel inhibitors of bacterial topoisomerases

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 23, 2008, Pages 6161-6164

  Trovatti, Eliane ^a   Cotrim, Camila A ^a   Garrido, Saulo S ^a   Barros, Ronaldo S ^a   Marchetto, Reinaldo ^a  

^a SÃO PAULO STATE UNIVERSITY UNESP   (Brazil)

Author keywords

CcdB toxin; DNA gyrase; Peptides; Topoisomerase IV

Indexed keywords

CCDB TOXIN; CCDBET1 TOXIN; CCDBET2 TOXIN; CCDBET2M TOXIN; CCDBET3 TOXIN; CCDBET4 TOXIN; CIPROFLOXACIN; DNA TOPOISOMERASE (ATP HYDROLYSING); DNA TOPOISOMERASE IV; SYNTHETIC PEPTIDE; UNCLASSIFIED DRUG;

AMINO ACID SEQUENCE; ARTICLE; CONCENTRATION RESPONSE; DNA SUPERCOILING; ENZYME INHIBITION; ESCHERICHIA COLI; MUTATION; NONHUMAN; PEPTIDE SYNTHESIS; PLASMID; PROTEIN PROTEIN INTERACTION; STRUCTURE ACTIVITY RELATION; TOXIN STRUCTURE; WILD TYPE;

AMINO ACIDS; BACTERIAL PROTEINS; BACTERIAL TOXINS; DNA GYRASE; DNA TOPOISOMERASE IV; DNA TOPOISOMERASES, TYPE II; ESCHERICHIA COLI; PEPTIDES; PROTEIN CONFORMATION; STRUCTURE-ACTIVITY RELATIONSHIP;

BACTERIA (MICROORGANISMS); ESCHERICHIA COLI;

EID: 55549141128     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.10.008     Document Type: Article

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